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Sequence 1: PCI-32765

Phase 1

Healthy Volunteers | Small molecule | Other |Johnson & Johnson|Last Updated: Jul 15, 2014

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment52
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01820936A Study to Determine the Effect of Food on the Pharmacokinetics of PCI-32765PHASE1 COMPLETED 52Mar 1, 2013Jun 1, 2013Jul 15, 20141 United States
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Study Endpoints
Primary Endpoints
Area under the plasma concentration-time curve from time 0 to time the last quantifiable concentrations of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
Area under the plasma concentration-time curve from time 0 to infinite time of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
Maximum plasma concentration of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
Secondary Endpoints
Time to reach the maximum plasma concentration of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
Percentage of area under the plasma concentration-time curve from time 0 to infinite time obtained by extrapolation of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
Elimination half-life of PCI-32765
Predose; postdose at 30 minutes and 1, 1.5, 2, 3, 4, 6, 8, 12, 16, 24, 36, 48, and 72 hours
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Treatment A: PCI-32765EXPERIMENTAL420 mg capsules administered by mouth with 240 mL noncarbonated water 30 minutes after completing a high-fat breakfast
Treatment B: PCI-32765EXPERIMENTAL420 mg capsules administered by mouth with 240 mL noncarbonated water after fasting for at least 10 hours and 30 minutes before starting a high-fat breakfast
Treatment C: PCI-32765EXPERIMENTAL420 mg capsules administered by mouth with 240 mL noncarbonated water 2 hours after completing a high-fat breakfast
Treatment D: PCI-32765EXPERIMENTAL420 mg capsules administered with 240 mL noncarbonated water after fasting at least 10 hours
Treatment E: PCI-32765EXPERIMENTAL840 mg capsules administered with 240mL noncarbonated water 30 minutes after completing a high-fat breakfast
Interventions
NameTypeDescription
Sequence 1: PCI-32765DRUGPeriod 1 = Treatment D, Period 2 = Treatment C, Period 3 = Treatment A, Period 4 = Treatment B
Sequence 2: PCI-32765DRUGPeriod 1 = Treatment A, Period 2 = Treatment D, Period 3 = Treatment B, Period 4 = Treatment C
Sequence 3: PCI-32765DRUGPeriod 1 = Treatment B, Period 2 = Treatment A, Period 3 = Treatment C, Period 4 = Treatment D
Sequence 4: PCI-32765DRUGPeriod 1 = Treatment C, Period 2 = Treatment B, Period 3 = Treatment D, Period 4 = Treatment A
Sequence 5: PCI-32765DRUGAfter completion of the 4-way crossover, an additional separate cohort of 8 subjects were enrolled. These subjects participated in 1 treatment period to document safety and PK
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Women must be postmenopausal or documented as surgically sterile * Men must agree to use an adequate contraception method as deemed appropriate by the investigator during the study and for 3 months after receiving the last dose of study drug, and to not donate sperm during the...

Countries:United States
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