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ZE46-0134

Phase 1

AML With Gene Mutations | Small molecule | Other |cbdMD, Inc.|Last Updated: Dec 31, 2025

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDBiomarker
Total Trials1
Total Enrollment150

FDA Designations

No designations recorded

Clinical trial landscape

ZE46-0134 · 1 trial · 1 indication

Phase 1 1
NCT06366789Dose Escalation and Expansion Study to Evaluate the Safety, PK, PD and Efficacy of ZE46-0134 in Adults With FLT3 Mutated or Spliceosome Mutated Relapsed or Refractory Acute Myeloid LeukemiaAML With Gene Mutations
RECRUITING150 Analytics
PHASE1RECRUITING
Dose Escalation and Expansion Study to Evaluate the Safety, PK, PD and Efficacy of ZE46-0134 in Adults With FLT3 Mutated or Spliceosome Mutated Relapsed or Refractory Acute Myeloid Leukemia
AML With Gene MutationsUnlock trial analytics

Study Endpoints

Primary Endpoints

The incidence of DLTs
From baseline to the End of Treatment (EOT) (Max 24 cycles, 28 days each)

To determine the maximum tolerated dose or biologically effective dose of ZE46-0134 in adults with FLT3 and spliceosome mutated relapsed and refractory AML.

Secondary Endpoints

Incidence of AE/SAE
From baseline to the EOT (Max 24 cycles, 28 days each)
Incidence of clinically significant abnormal laboratory results
From baseline to the EOT (Max 24 cycles, 28 days each)
Incidence of abnormal clinically significant ECG results
From baseline to the EOT (Max 24 cycles, 28 days each)
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ZE46-0134 Dose Level -1EXPERIMENTALOptional and would only be performed Dose Level 1 is poorly tolerated
ZE46-0134 Dose Level 1EXPERIMENTAL -
ZE46-0134 Dose Level 2EXPERIMENTAL -
ZE46-0134 Dose Level 3EXPERIMENTAL -
ZE46-0134 Dose Level 4EXPERIMENTAL -
ZE46-0134 Dose Level 5EXPERIMENTAL -
ZE46-0134 Selected dose 1EXPERIMENTALThe doses used in Part 2 of the study will be determined based on the data from Part 1 of the study and will not exceed a loading dose of 150 mg x 2 days and maintenance dose of 50 mg QD
ZE46-0134 Selected dose 2EXPERIMENTALThe doses used in Part 2 of the study will be determined based on the data from Part 1 of the study and will not exceed a loading dose of 150 mg x 2 days and maintenance dose of 50 mg QD
ZE46-0134 Dose Level 6EXPERIMENTAL -
ZE46-0134 Dose Level 7EXPERIMENTAL -
ZE46-0134 Dose Level 8EXPERIMENTAL -
ZE50-0134 (Group 2) Dose Level -1EXPERIMENTALOptional and would only be performed Dose Level 1 is poorly tolerated
ZE50-0134 (Group 2) Dose Level 1EXPERIMENTAL -
ZE50-0134 (Group 2) Dose Level 2EXPERIMENTAL -
ZE50-0134 (Group 2) Dose Level 3EXPERIMENTAL -
ZE50-0134 (Group 2) Dose Level 4EXPERIMENTAL -
ZE50-0134 (Group 2) Selected dose 1EXPERIMENTALThe doses used in Part 2 of the study will be determined based on the data from Part 1 of the study.
ZE50-0134 (Group 2) Selected dose 2EXPERIMENTALThe doses used in Part 2 of the study will be determined based on the data from Part 1 of the study.

Interventions

NameTypeDescription
ZE46-0134DRUGoral capsules QD
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites23

Inclusion Criteria: 1. Written Informed Consent must be obtained from the patient or legally authorized representative prior to any study-related procedures (including withdrawal of prohibited medication, if applicable). 2. Patient is ≥18 years of age at the time of obtaining informed consent. 3. P...

Countries:United StatesAustraliaSouth KoreaTaiwan
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Competitive Landscape -Genetic Mutations 6 trials (matched to "AML With Gene Mutations")

Frequently asked questions about ZE46-0134

What is ZE46-0134 used for?

ZE46-0134 is an investigational small molecule being developed for the treatment of acute myeloid leukemia (AML) with gene mutations, specifically in adults with FLT3 mutated or spliceosome mutated relapsed or refractory AML. It is currently in Phase 1 clinical development.

What does ZE46-0134 target?

ZE46-0134 is being studied in patients with FLT3 mutated or spliceosome mutated relapsed or refractory acute myeloid leukemia. The clinical trial evaluates its safety, pharmacokinetics, pharmacodynamics, and efficacy in this biomarker-selected patient population.

Who is developing ZE46-0134?

ZE46-0134 is being developed by cbdMD, Inc., a company traded on the NYSE American under the ticker symbol YCBD. The drug is currently in Phase 1 clinical development for AML with gene mutations.

What phase is ZE46-0134 in?

ZE46-0134 is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. A Phase 1 trial is currently recruiting participants to evaluate the drug in adults with relapsed or refractory acute myeloid leukemia.

What clinical trials is ZE46-0134 in?

ZE46-0134 is being studied in a Phase 1 clinical trial with the identifier NCT06366789. This is a dose escalation and expansion study evaluating the safety, pharmacokinetics, pharmacodynamics, and efficacy of ZE46-0134 in adults with FLT3 mutated or spliceosome mutated relapsed or refractory acute myeloid leukemia.

Where is the ZE46-0134 clinical trial being conducted?

The Phase 1 clinical trial of ZE46-0134 is being conducted in the United States, Australia, South Korea, and Taiwan. The trial is recruiting adults aged 18 years and older with relapsed or refractory acute myeloid leukemia with specific gene mutations.