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palbociclib isethionate

Phase 1

Healthy | Small molecule | Other |Pfizer, Inc.|Last Updated: Mar 17, 2014

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
UNCONTROLLED
Total Trials1
Total Enrollment36
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02041273Relative Bioavailability Of Palbociclib (PD-0332991) Under Fed And Fasted ConditionsPHASE1 COMPLETED 36Jan 1, 2014Mar 1, 2014Mar 17, 20141 United States
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Study Endpoints
Primary Endpoints
Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUC (0 - 8)]
7 days

AUC (0 - 8)= Area under the plasma concentration versus time curve (AUC) from time zero (pre-dose) to extrapolated infinite time (0 - 8). It is obtained from AUC (0 - t) plus AUC (t - 8).

Maximum Observed Plasma Concentration (Cmax)
7 days
Secondary Endpoints
Area Under the Curve From Time Zero to Last Quantifiable Concentration (AUClast)
7 days
Apparent Oral Clearance (CL/F)
7 days
Plasma Decay Half-Life (t1/2)
7 days
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Study Design & Arms
AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Palbociclib given to healthy volunteersEXPERIMENTAL -
Interventions
NameTypeDescription
palbociclib isethionate (phase 1 and 2 studies)DRUG125 mg palbociclib isethionate salt under overnight fasting conditions
palbociclib commercial free base capsuleDRUG125 mg palbociclib commercial free base capsule under fed conditions ( moderate fat meal)
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male subjects and/or female subjects of non-childbearing potential between the ages of 18 and 55 years. * Evidence of a personally signed and dated informed consent document indicating that the subject has been informed of all pertinent aspects of the study. Exclusion...

Countries:United States
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