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TH-302

Phase 1

Solid Tumor | Small molecule | Oncology |Merck & Company, Inc.|Last Updated: Jun 10, 2016

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDDMC
Total Trials1
Total Enrollment10

FDA Designations

No designations recorded

Clinical trial landscape

TH-302 · 1 trial · 1 indication

Phase 1 1
NCT02076230A Phase 1 TH-302 Mass Balance TrialSolid Tumor
COMPLETED10 Analytics
PHASE1COMPLETED
A Phase 1 TH-302 Mass Balance Trial
Solid TumorUnlock trial analytics

Study Endpoints

Primary Endpoints

Pharmacokinetics profile in plasma: Cmax, Tmax, AUC (0-t), lambda_z, t1/2, AUC (0-infinity), CL, Vss, Vz, MRT for TH-302 and its active metabolite Br-IPM
Days 1 and 8 of Cycle 1
Pharmacokinetics profile in excreta: Cumulative Ae (0-t), Ae (0-infinity), percent radioactive dose excreted in urine and feces, AeUF, CLR, CLNR for TH-302 and its active metabolite Br-IPM
Day 1 of Cycle 1

Secondary Endpoints

Number of subjects with Treatment-emergent adverse events (TEAEs)
Baseline up to Day 30 after the last dose of study treatment
Blood to plasma ratio of total 14C-radioactivity
Days 1 and 8 of Cycle 1
Total and free plasma concentrations of TH-302 in plasma
Day 1 of Cycle 1
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
[14C] TH-302 (Label 1)EXPERIMENTAL -
[14C] TH-302 (Label 2)EXPERIMENTAL -

Interventions

NameTypeDescription
[14C] TH-302 (Label 1)DRUG\[14C\]-labeled TH-302 (Label 1) will be administered as intravenous infusion over 30 minutes on Day 1 of Part A.
[14C] TH-302 (Label 2)DRUG\[14C\]-labeled TH-302 (Label 2) will be administered as intravenous infusion over 30 minutes on Day 1 of Part A.
Unlabeled TH-302DRUGUnlabeled TH-302 will be administered along with labeled TH-302 at the dose of 340 milligram per square meter (mg/m\^2) as intravenous infusion over 30 minutes on Day 1 of Part A, followed by recommended Phase 2 dose (RP2D) of 480 mg/m\^2 as monotherapy infusion over 30 minutes on Days 8 and 15 of Part A; and on Days 1, 8 and 15 of Part B, until progression of the disease, unacceptable toxicity, withdrawal of consent by the subject, loss to follow up, or death.
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Eligibility Criteria

Age Range18 Years to 70 Years
SexMALE
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Male subject with pathologically or cytologically confirmed solid tumor which is locally advanced or metastatic, and either refractory to the standard therapy or for which no effective standard therapy is available * Subject has measurable and evaluable disease as RECIST versi...

Countries:Germany
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Competitive Landscape -Other Solid Tumors 9 trials (matched to "Solid Tumor")

Frequently asked questions about TH-302

What is TH-302 used for?

TH-302 is an investigational small molecule being studied for the treatment of solid tumors. It is in Phase 1 clinical development as a potential oncology therapy.

Who is developing TH-302?

TH-302 is being developed by Merck & Company, Inc. (NYSE: MRK). The drug is currently in Phase 1 clinical trials for solid tumors.

What phase is TH-302 in?

TH-302 is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed.

What clinical trials is TH-302 in?

TH-302 has one completed Phase 1 trial, NCT02076230, titled "A Phase 1 TH-302 Mass Balance Trial." This trial enrolled 10 male participants aged 18 years and older with solid tumors and was conducted in Germany.

Is TH-302 being studied in a randomized trial?

No, the completed Phase 1 trial of TH-302 (NCT02076230) was not randomized and was not double-blind. It was a controlled study that enrolled 10 participants with solid tumors.