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BMF-500

Phase 1

Acute Myeloid Leukemia | Small molecule | Oncology |Biomea Fusion, Inc.|Last Updated: Feb 23, 2026

Target and mechanism

Molecular targetFLT3
Target classGene
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDDMC
Total Trials1
Total Enrollment35

FDA Designations

No designations recorded

Clinical trial landscape

BMF-500 · 1 trial · 1 indication

Phase 1 1
NCT05918692A Phase 1 Study of BMF-500 in Adults With Acute LeukemiaAcute Myeloid Leukemia
ACTIVE NOT_RECRUITING35 Analytics
PHASE1ACTIVE NOT_RECRUITING
A Phase 1 Study of BMF-500 in Adults With Acute Leukemia
Acute Myeloid LeukemiaUnlock trial analytics

Study Endpoints

Primary Endpoints

Evaluate the safety and tolerability of BMF-500 by incidence of Treatment Emergent Adverse Events (TEAEs).
At the end of each 28 Day cycle for a maximum of 32 cycles

Assessed by the NCI CTCAE version 5.0.

Evaluate the safety and tolerability of BMF-500 by incidence of Serious Adverse Events (SAEs).
At the end of each 28 Day cycle for a maximum of 32 cycles

Assessed by the NCI CTCAE version 5.0.

Determine the recommended Phase 2 Dose (RP2D) of BMF-500.
At the end of 28 day Dose-Limiting Toxicities (DLT) observation Period

Safety, as determined by Dose-Limiting Toxicities (clinically significant Adverse Event) within each dose level assessed NCI CTCAE version 5.0.

Secondary Endpoints

Determine the pharmacokinetics of BMF-500.
At the end of each cycle (each cycle is 28 days in duration) for 7 cycles
Evaluate the efficacy of BMF-500
At the end of each cycle (each cycle is 28 days in duration) for a maximum of 32 cycles
Assess additional evidence of antitumor activity per investigator assessment as per corresponding response criteria.
At the end of each cycle (each cycle is 28 days in duration) for a maximum of 32 cycles
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Arm A: Escalation PhaseEXPERIMENTALBMF-500 taken twice daily by participants who are not receiving drugs that inhibit CYP3A4 activity.
Arm B: Escalation PhaseEXPERIMENTALBMF-500 taken twice daily by participants who are receiving necessary azole antifungals that are Strong CYP3A4 inhibitors.
Arm C: Escalation PhaseEXPERIMENTALBMF-500 taken twice daily by participants who are receiving necessary azole antifungals that are moderate CYP3A4 inhibitors.

Interventions

NameTypeDescription
BMF-500DRUGInvestigational Product
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites14

Key Inclusion Criteria: * Age ≥ 18 years. * Individuals with histologically or pathologically confirmed diagnosis of relapsed or refractory AML with documented FLT3 mutation, and/or Individuals with histologically or pathologically confirmed diagnosis of their malignancy with wild-type FLT3 (includ...

Countries:United States
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Frequently asked questions about BMF-500

What is BMF-500 used for?

BMF-500 is an investigational small molecule being developed for the treatment of Acute Myeloid Leukemia (AML). It is currently in Phase 1 clinical development and has not been approved by the FDA. The drug is being studied in adult patients with acute leukemia.

What does BMF-500 target?

BMF-500 targets FLT3, a gene that is frequently mutated in Acute Myeloid Leukemia. By targeting FLT3, the drug aims to interfere with the signaling pathways that drive the growth of leukemia cells. This mechanism is being evaluated in early-stage clinical trials.

Who makes BMF-500?

BMF-500 is being developed by Biomea Fusion, Inc., a biopharmaceutical company. The company's stock is traded under the ticker symbol BMEA. Biomea Fusion is conducting clinical trials to evaluate the safety and efficacy of BMF-500 in patients with acute leukemia.

What phase is BMF-500 in?

BMF-500 is currently in Phase 1 clinical development. It is an investigational drug, meaning it has not yet received FDA approval. The ongoing Phase 1 trial is designed to assess the safety, tolerability, and preliminary efficacy of BMF-500 in adults with acute leukemia.

What clinical trials is BMF-500 in?

BMF-500 is being studied in a Phase 1 clinical trial with the identifier NCT05918692. The trial, titled 'A Phase 1 Study of BMF-500 in Adults With Acute Leukemia,' is active but not recruiting participants. It is enrolling approximately 35 patients in the United States.

Is BMF-500 the same as any other drug?

No, BMF-500 is a unique investigational compound developed by Biomea Fusion. It is not known to have any alternative names. The drug is being studied specifically for its potential role in treating Acute Myeloid Leukemia and is in early-stage clinical development.