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BHV-1510

Phase 1

Solid Tumor | Small molecule | Oncology |Biohaven Ltd.|Last Updated: Mar 11, 2026

Target and mechanism

Molecular targetTrop2
Target classProtein
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment500

FDA Designations

No designations recorded

Clinical trial landscape

BHV-1510 · 1 trial · 1 indication

Phase 1 1
NCT06384807A Phase 1/2 Study of BHV-1510 (Previously PBI-410) in Advanced Solid TumorsSolid Tumor
RECRUITING500 Analytics
PHASE1RECRUITING
A Phase 1/2 Study of BHV-1510 (Previously PBI-410) in Advanced Solid Tumors
Solid TumorUnlock trial analytics

Study Endpoints

Primary Endpoints

Phase 1: Number of patients with adverse events (AEs)
Through study completion, estimated as an average of 47 months

Description: Incidence and severity of AEs, serious adverse events (SAEs) and dose limiting toxicities (DLTs). Severity of AEs will be assessed according to the NCI CTCAE v5.0. This applies to both the BHV-1510 monotherapy arm and BHV-1510 in combination with Cemiplimab arm.

Phase 1: Recommended doses or schedules for expansion (RDEs) and maximum tolerated dose (MTD)
Approximately 15 months

Based on tolerability and preliminary antitumor activity. This applies to both the BHV-1510 monotherapy arm and BHV-1510 in combination with Cemiplimab arm.

Phase 2: Objective Response Rate (ORR) for BHV-1510 for monotherapy and in combination with cemiplimab
Through study completion, estimated as an average of 47 months

Assessed by Response Evaluation Criteria in Solid Tumors (RECIST) v 1.1.

Phase 2: Number of patients with AEs for BHV-1510 for monotherapy and in combination with cemiplimab
Through study completion, estimated as an average of 47 months

Incidence and severity of AEs, SAEs and DLTs. Severity of AEs will be assessed according to the NCI CTCAE v5.0

Phase 2: Duration of Response (DoR) for BHV-1510 for monotherapy and in combination with cemiplimab
Through study completion, estimated as an average of 47 months

Assessed by RECIST v 1.1

Secondary Endpoints

Phase 1 and 2: Maximum Plasma Concentration (Cmax) of BHV-1510, total antibody and payload (BHC-0080269)
Up to 8 timepoints, but not exceeding, 22 days in Cycles 1 and 3
Phase 1 and 2: Area Under the Concentration versus time Curve from the end of infusion to the last measurable concentration (AUClast) of BHV-1510, total antibody and payload
Up to 8 timepoints, but not exceeding, 22 days in Cycles 1 and 3
Phase 1 and 2: Area Under the Concentration versus time curve extrapolated to infinity (AUCinf) of BHV-1510, total antibody and payload
Up to 8 timepoints, but not exceeding, 22 days in Cycle 1
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BHV-1510 Monotherapy Dose EscalationEXPERIMENTAL -
BHV-1510 in combination with Cemiplimab dose escalationEXPERIMENTAL -

Interventions

NameTypeDescription
BHV-1510DRUGBHV-1510 will be administered on Day 1 every 3 weeks
CemiplimabDRUGcemiplimab (350mg) will be administered as an IV infusion on Day 1 every 3 weeks
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites17

Key Inclusion Criteria: * Male or female participants aged ≥18 years. * Unresectable, incurable, locally advanced or metastatic epithelial-origin solid tumor that is refractory to standard therapies, or has no approved standard therapies, or no approved standard therapies at its current treatment s...

Countries:United States
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Competitive Landscape -Other Solid Tumors 9 trials (matched to "Solid Tumor")

Frequently asked questions about BHV-1510

What is BHV-1510 used for?

BHV-1510 is an investigational small molecule being developed for the treatment of solid tumors. It is currently in Phase 1 clinical development, and the drug is being studied in patients with advanced solid tumors. BHV-1510 is not yet approved by the FDA and remains in clinical trials.

What does BHV-1510 target?

BHV-1510 targets Trop2, a protein that is overexpressed in many solid tumors. By targeting Trop2, the drug aims to interfere with tumor growth. This mechanism is being evaluated in a Phase 1/2 clinical trial for advanced solid tumors.

Who is developing BHV-1510?

BHV-1510 is being developed by Biohaven Ltd., a biopharmaceutical company. The company is conducting clinical trials to evaluate the safety and efficacy of BHV-1510 in patients with solid tumors. Biohaven is listed on the stock exchange under the ticker symbol BHVN.

What phase is BHV-1510 in?

BHV-1510 is in Phase 1 clinical development. The drug is being studied in a Phase 1/2 trial for advanced solid tumors, and the trial is currently recruiting participants. BHV-1510 is an investigational drug and has not been approved by regulatory authorities.

What clinical trials is BHV-1510 in?

BHV-1510 is being studied in a Phase 1/2 clinical trial with the identifier NCT06384807. This trial is recruiting patients with advanced solid tumors in the United States, with an enrollment target of 500 participants. The study is open to adults aged 18 years and older.

Is BHV-1510 the same as PBI-410?

Yes, BHV-1510 was previously known as PBI-410. The clinical trial NCT06384807, titled 'A Phase 1/2 Study of BHV-1510 (Previously PBI-410) in Advanced Solid Tumors,' confirms that the drug was renamed. Both names refer to the same investigational small molecule targeting Trop2.