Recent Updates
Recently added Catalysts

Rivaroxaban Xarelto, BAY59-7939

Phase 1

Thrombosis | Small molecule | Cardiovascular |Bayer AG|Last Updated: Apr 16, 2019

Target and mechanism

Molecular targetF10
Target classInhibitor
ModalitySmall molecule

Also known as Rivaroxaban (Xarelto, BAY59-7939

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

UNCONTROLLEDDMC
Total Trials1
Total Enrollment47

FDA Designations

No designations recorded

Clinical trial landscape

Rivaroxaban Xarelto, BAY59-7939 · 1 trial · 1 indication

Phase 1 1
NCT02497716Phase I Study on Rivaroxaban Granules for Oral Suspension Formulation in ChildrenThrombosis
COMPLETED47 Analytics
PHASE1COMPLETED
Phase I Study on Rivaroxaban Granules for Oral Suspension Formulation in Children
ThrombosisUnlock trial analytics

Study Endpoints

Primary Endpoints

AUC (area under the curve)
4x within 8 hrs post study drug administrationh and 1x between 24-28h after administration

Only PK will be tested in central lab

Cmax (maximum observed drug concentration)
4x within 8 hrs post study drug administrationh and 1x between 24-28h after administration

Only PK will be tested in central lab

Secondary Endpoints

Prothrombin time (PT)
Pre-administration, if not done within the past 10 days, and then 24-28 hours after drug administration
Activated partial thromboplastin time (aPTT)
Pre-administration, if not done within the past 10 days, and then 24-28 hours after drug administration
Composite of major bleeding and clinically relevant non-major bleeding
From dose administration until follow up call on day 8+3
Unlock Study Endpoints

Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeOTHER

Treatment Arms

ArmTypeDescription
RivaroxabanEXPERIMENTALSingle arm, open label study

Interventions

NameTypeDescription
Rivaroxaban (Xarelto, BAY59-7939DRUGSingle dose of reconstituted rivaroxaban granules
Unlock Study Design Details

Eligibility Criteria

Age Range2 Months to 12 Years
SexALL
Healthy VolunteersNo
Study Sites21

Inclusion Criteria: * Children with an age ≥2 months and weight between 3 and \<12 kg, who have completed anticoagulant treatment at least 10 days prior to the planned study drug administration. * Gestational age at birth of at least 37 weeks * Oral feeding/ nasogastric/ gastric feeding for at...

Countries:United StatesBelgiumCanadaFinlandFranceHungaryItalySpain
Unlock Eligibility Criteria

Competitive Landscape -Thrombosis and Embolism 22 trials (matched to "Thrombosis")

Top 2 of 9 competitors

Unlock Competitive Intelligence

Frequently asked questions about Rivaroxaban Xarelto, BAY59-7939

What is Rivaroxaban used for?

Rivaroxaban is used for the treatment of thrombosis, a condition involving blood clots. It is a small molecule drug developed by Bayer AG under the ticker BAYRY. The clinical program includes a Phase 1 study in children with thrombosis, evaluating an oral suspension granule formulation.

What does Rivaroxaban target?

Rivaroxaban targets coagulation factor Xa, also known as F10. It acts as an inhibitor of this enzyme, which plays a central role in the blood coagulation cascade. By inhibiting factor Xa, rivaroxaban reduces thrombin generation and clot formation.

Who makes Rivaroxaban?

Rivaroxaban is developed by Bayer AG, which trades under the ticker BAYRY. Bayer AG is the company responsible for the clinical development of the drug, including the Phase 1 trial in pediatric patients with thrombosis.

What phase is Rivaroxaban in?

Rivaroxaban is in Phase 1 clinical development for thrombosis. The only listed trial is a completed Phase 1 study. It is an investigational drug and has not been approved by the FDA for this indication based on the available information.

What clinical trials is Rivaroxaban in?

Rivaroxaban has been studied in a Phase 1 trial, NCT02497716, titled 'Phase I Study on Rivaroxaban Granules for Oral Suspension Formulation in Children.' The trial enrolled 47 participants with thrombosis across the United States, Belgium, Canada, Finland, France, Hungary, Italy, and Spain, and is completed.

Is Rivaroxaban the same as Xarelto or BAY59-7939?

Yes, Rivaroxaban is also known as Xarelto and BAY59-7939. These are alternative names for the same drug substance. Rivaroxaban is the international nonproprietary name, Xarelto is a brand name, and BAY59-7939 is a development code used by Bayer AG.