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ARV-806

Phase 1

KRAS G12D Mutation | Small molecule | Oncology |Arvinas, Inc.|Last Updated: Aug 19, 2026

Target and mechanism

Molecular targetKRAS G12D
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment159

FDA Designations

No designations recorded

Clinical trial landscape

ARV-806 · 1 trial · 2 indications

Phase 1 1
NCT07023731A Study to Evaluate ARV-806 in Adults With Advanced Cancer That Has the KRAS G12D MutationKRAS G12D Mutation
ACTIVE NOT_RECRUITING159 Analytics
PHASE1ACTIVE NOT_RECRUITING
A Study to Evaluate ARV-806 in Adults With Advanced Cancer That Has the KRAS G12D Mutation
KRAS G12D MutationUnlock trial analytics

Study Endpoints

Primary Endpoints

Part A (Phase 1): Number of dose-limiting toxicities (DLTs) of ARV-806
28 days from first ARV-806 administration

Number of participants within a dose escalation cohort with adverse events (AEs) meeting protocol defined dose limiting toxicities during cycle 1 (28 days).

Part A (Phase 1): Number of participants with AEs
From the study baseline to at least 28 days after last dose of ARV-806

AEs as characterized by type, frequency, severity (as graded by National Cancer Institute Common Terminology Criteria for Adverse Events \[NCI CTCAE\]), timing, seriousness, and relationship to study intervention as a measure of safety and tolerability

Part B (Phase 2): Overall Response Rate (ORR)
Approximately 2 years

ORR is a parameter measuring the anti-tumor activity of ARV-806. ORR is the percentage of participants for whom the study treatment resulted in a complete response or partial response of the disease under study. It is measured using CT/MRI and RECIST 1.1 criteria per investigator assessment.

Secondary Endpoints

Pharmacokinetics (PK) of ARV-806 (Part A): Area under the plasma or blood concentration-time profile during a dosing interval (AUCtau)
At predefined intervals throughout the treatment period, up to approximately 6 months after first dose of ARV-806
PK of ARV-806 (Part A): Area under the plasma or blood concentration time profile from time zero to the time of the last quantifiable concentration (Clast) (AUClast)
At predefined intervals throughout the treatment period, up to approximately 6 months after first dose of ARV-806
PK of ARV-806 (Part A): Maximum plasma or blood concentration (Cmax)
At predefined intervals throughout the treatment period, up to approximately 6 months after first dose of ARV-806
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Phase 1/Part A Monotherapy (Dose Escalation)EXPERIMENTALParticipants will receive ARV-806 at the assigned doses and regimen (weekly or every 2 weeks).
Phase 2/Part B Monotherapy (Dose Expansion)EXPERIMENTALParticipants will receive ARV-806 at one of up to 2 dose levels/regimens selected from Part A)

Interventions

NameTypeDescription
ARV-806DRUGIntravenous infusion at assigned dose and dosing schedule
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites14

Inclusion Criteria: Part A: * Histological or cytological diagnosis of unresectable or metastatic solid tumor malignancy, AND * Must have evidence of KRAS G12D mutation in tumor tissue or blood (circulating tumor deoxyribonucleic acid \[ctDNA\]), AND * Must have received prior standard-of-care (SO...

Countries:United States
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Competitive Landscape -Genetic Mutations 6 trials (matched to "KRAS G12D Mutation")

Recent Changes (Last 90 Days)

LOWAug 20, 2026NCT07023731primaryCompletionDate: changed
LOWAug 20, 2026NCT07023731primaryCompletionDate: changed
LOWAug 20, 2026NCT07023731primaryCompletionDate: changed
LOWAug 20, 2026NCT07023731primaryCompletionDate: changed
MEDIUMJul 2, 2026NCT07023731Status: RECRUITING → ACTIVE_NOT_RECRUITING
MEDIUMJul 2, 2026NCT07023731Status: RECRUITING → ACTIVE_NOT_RECRUITING

Frequently asked questions about ARV-806

What is ARV-806 used for?

ARV-806 is an investigational small molecule being developed for the treatment of advanced solid cancers that have the KRAS G12D mutation. It is currently in Phase 1 clinical development and has not been approved by the FDA.

What does ARV-806 target?

ARV-806 targets the KRAS G12D mutation, a specific genetic alteration found in certain cancers. By targeting this mutation, the drug aims to address tumors that carry this particular KRAS variant.

Who makes ARV-806?

ARV-806 is being developed by Arvinas, Inc., a biopharmaceutical company traded on NASDAQ under the ticker symbol ARVN. The company is conducting clinical trials to evaluate the drug's safety and efficacy.

What phase is ARV-806 in?

ARV-806 is in Phase 1 clinical development. It is an investigational drug, meaning it has not yet been approved by regulatory authorities and is still being studied in clinical trials.

What clinical trials is ARV-806 in?

ARV-806 is being studied in a Phase 1 clinical trial with the identifier NCT07023731. This trial evaluates the drug in adults with advanced cancer that has the KRAS G12D mutation, with an enrollment of 159 participants in the United States.