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zenocutuzumab

Phase 2

Solid Tumours Harboring NRG1 Fusion | Small molecule | Oncology |cbdMD, Inc.|Last Updated: Apr 29, 2025

Target and mechanism

Molecular targetERBB2, ERBB3
Target classInhibitor
ModalitySmall molecule

Also known as zenocutuzumab (MCLA-128)

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment250

FDA Designations

No designations recorded

Clinical trial landscape

zenocutuzumab · 1 trial · 4 indications

Phase 2 1
NCT02912949A Study of Zenocutuzumab (MCLA-128) in Patients With Solid Tumors Harboring an NRG1 Fusion (eNRGy)Solid Tumours Harboring NRG1 Fusion
ACTIVE NOT_RECRUITING250 Analytics
PHASE2ACTIVE NOT_RECRUITING
A Study of Zenocutuzumab (MCLA-128) in Patients With Solid Tumors Harboring an NRG1 Fusion (eNRGy)
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Study Endpoints

Primary Endpoints

Objective overall response rate (ORR) as per local investigator's assessment
36 months

Evaluation of clinical benefit assessed by RECIST v1.1 determining objective overall response rate (ORR)

Duration of response per RECIST v1.1 as per local Investigator's assessment.
36 Months

To assess durability of anti-tumor activity of MCLA-128 in patients with NRG1 fusions as assessed locally

Secondary Endpoints

Overall response rate as per Blinded Independent Central Review (BICR)
36 months
Clinical Benefit Rate (CBR) of zenocutuzumab (MCLA-128) assessed locally and BICR
36 months
Duration of Response as per BICR
36 months
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part 2 Pancreatic adenocarcinoma harboring NRG1 fusionEXPERIMENTALParticipants will receive intravenous infusion of 750 mg of zenocutuzumab (MCLA-128) (the recommended Phase 2 dose (RP2D)) every 2 weeks.
Part 2 NSCLC cancer harboring NRG1 fusionEXPERIMENTALParticipants will receive intravenous infusion of 750 mg of zenocutuzumab (MCLA-128) (the recommended Phase 2 dose (RP2D)) every 2 weeks.
Part 2 Solid tumour (basket) harboring NRG1 fusionEXPERIMENTALParticipants will receive intravenous infusion of 750 mg of zenocutuzumab (MCLA-128) (the recommended Phase 2 dose (RP2D)) every 2 weeks.

Interventions

NameTypeDescription
zenocutuzumab (MCLA-128)DRUGfull length IgG1 bispecific antibody targeting HER2 and HER3
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites64

Inclusion Criteria: * At least one measurable lesion according to RECIST v1.1 OR evaluable disease for a limited number of patients (up to 15) in Group H; * Performance status of ECOG 0 - 2; * Estimated life expectancy of at least 12 weeks; * Toxicities incurred as a result of previous anti-cancer ...

Countries:United StatesAustriaBelgiumCanadaDenmarkFranceGermanyIsraelItalyJapanNetherlandsNorwaySingaporeSouth KoreaSpainSwedenTaiwanUnited Kingdom
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Frequently asked questions about zenocutuzumab

What is zenocutuzumab used for?

Zenocutuzumab is an investigational antibody being studied for the treatment of solid tumors harboring an NRG1 fusion, including non-small cell lung cancer and pancreatic cancer with this genetic alteration. It is currently in Phase 2 clinical development and has not been approved by regulatory authorities.

What does zenocutuzumab target?

Zenocutuzumab is a monoclonal antibody (a -mab) designed to target tumors that harbor an NRG1 fusion. It is being evaluated in biomarker-selected patients whose cancers carry this specific genetic alteration, which is the basis for its mechanism of action in treating these solid tumors.

Who is developing zenocutuzumab?

Zenocutuzumab is being developed by cbdMD, Inc., a company traded on the stock exchange under the ticker YCBD. The drug is currently in Phase 2 clinical trials for solid tumors harboring an NRG1 fusion.

What phase is zenocutuzumab in?

Zenocutuzumab is in Phase 2 clinical development. It is an investigational drug being studied in patients with solid tumors harboring an NRG1 fusion, and it has not yet received FDA approval. The ongoing trial is active but not recruiting participants.

What clinical trials is zenocutuzumab in?

Zenocutuzumab is being studied in a single Phase 2 clinical trial with the identifier NCT02912949, titled "A Study of Zenocutuzumab (MCLA-128) in Patients With Solid Tumors Harboring an NRG1 Fusion (eNRGy)." The trial is active but not recruiting and has an enrollment of 250 participants across multiple countries.

Is zenocutuzumab the same as MCLA-128?

Yes, zenocutuzumab is also known as MCLA-128. The drug is being studied under this alternative name in clinical trials, including the eNRGy study (NCT02912949), which evaluates zenocutuzumab (MCLA-128) in patients with solid tumors harboring an NRG1 fusion.