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XPF-001

Phase 2

Dental Pain | Small molecule | Pain |Xenon Pharmaceuticals Inc.|Last Updated: Jul 16, 2012

Success Probability
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Market & Valuation
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment61
FDA Designations
No designations recorded
Clinical trial landscape

XPF-001 · 3 trials · 4 indications

Phase 2 1Phase 1 2
NCT00954356Safety and Efficacy Study of XPF-001 to Treat Pain Following Wisdom Tooth ExtractionDental Pain
COMPLETED61 Analytics
PHASE2COMPLETED
Safety and Efficacy Study of XPF-001 to Treat Pain Following Wisdom Tooth Extraction
Dental PainUnlock trial analytics
Study Endpoints
Primary Endpoints
Total Pain Relief at 6 Hours Post Dose (TOTPAR 6)
6 hours post dose

The primary efficacy variable was total pain relief at the 6-hour observation (TOTPAR 6); TOTPAR 6 is an area calculation incorporating time and relief scores over the 6 hours following dosing and was calculated using Simpson's trapezoidal rule. The higher the LS Means scores, the more pain relief was obtained. Relief (REL) scores were measured at multiple timepoints after dosing, using a 5 point categorical pain relief rating scale. (None = 0, A Little Relief = 1, Some = 2, A Lot = 3, Complete Relief = 4). The minimum possible TOTPAR 6 score = 0, maximum possible score = 24

Pain intensity difference (PID) in each treatment period based on an 11-point Pain Intensity-NRS (where 0 = No pain and 10 = worst pain you can imagine)
2 days
ECGs, Telemetry, Vital Signs, Physical Examinations, Laboratory Assessments and Adverse Events.
up to 14 days post dose
Secondary Endpoints
Total Pain Relief (TOTPAR) at 4 Hours Post Dose
4 hours
Total Pain Relief (TOTPAR) at 8 Hours Post Dose
8 hours
Total Pain Relief (TOTPAR) at 12 Hours Post Dose
12 hours
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
XPF-001EXPERIMENTAL -
PlaceboPLACEBO_COMPARATOR -
Matching PlaceboPLACEBO_COMPARATOR -
Cohort 1: Single dose of XPF-001EXPERIMENTAL -
Cohort 2: Single dose of XPF-001EXPERIMENTAL -
Cohort 3: Single dose of XPF-001EXPERIMENTAL -
Cohort 4: Single dose of XPF-001EXPERIMENTAL -
Cohort 5: Single dose of XPF-001EXPERIMENTAL -
Cohort A: Repeated doses of XPF-001EXPERIMENTAL -
Cohort B: Repeated doses of XPF-001EXPERIMENTAL -
Cohort C: Repeated doses of XPF-001EXPERIMENTAL -
Interventions
NameTypeDescription
XPF-001DRUGSingle oral administration of 500 mg XPF-001 capsules (5 x 100 mg capsules)
placeboDRUGSingle oral administration of 5 x 100 mg Placebo capsules.
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Eligibility Criteria
Age Range18 Years to 60 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Males (aged 18-60) and females of non-childbearing potential (aged 18-60; * BMI between 19.5 to 32.0 kg/m2; * Outpatient, scheduled to undergo surgical extraction of 2 or more impacted 3rd molars (with at least 1 partial bony mandibular extraction); * use of only the following...

Countries:United StatesNetherlandsCanada
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