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DIVALPROEX, USP

Phase 1

Healthy | Small molecule | Other |Viatris Inc.|Last Updated: Aug 18, 2010

Target and mechanism

Molecular targetALDH5A1
Target classInhibitor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLEDBiomarker
Total Trials2
Total Enrollment37

FDA Designations

No designations recorded

Clinical trial landscape

DIVALPROEX, USP · 2 trials · 1 indication

Phase 1 2
NCT01183676Fed Bioequivalence Study of Divalproex Sodium Delayed-Release Tablets, 500 mgHealthy
COMPLETED20 Analytics
NCT01184391Bioequivalence Study of Divalproex Sodium Delayed-Release Tablets, 500 mgHealthy
COMPLETED17 Analytics
PHASE1COMPLETED
Fed Bioequivalence Study of Divalproex Sodium Delayed-Release Tablets, 500 mg
HealthyUnlock trial analytics
PHASE1COMPLETED
Bioequivalence Study of Divalproex Sodium Delayed-Release Tablets, 500 mg
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax
30 days

Maximum plasma concentration (micrograms/mL)

AUCL
30 days

Area under the concentration time curve from time zero to the last measurable time point. (micrograms x mL/hour)

AUCI
30 days

Area under the concentration time curve from time zero to infinity (micrograms x mL/hour)

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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER

Treatment Arms

ArmTypeDescription
Divalproex SodiumEXPERIMENTALDIVALPROEX SODIUM DELAYED-RELEASE TABLETS, USP, 500 MG - Mylan Pharmaceuticals Inc
Depakote TabletsACTIVE_COMPARATORDEPAKOTE® Tablets, 500 MG Abbott Laboratories
Test: Divalproex SodiumEXPERIMENTALDIVALPROEX SODIUM DELAYED-RELEASE TABLETS, USP, 500 MG
Reference: Depakote TabletsACTIVE_COMPARATORDEPAKOTE® Tablets, 500 MG Abbott Laboratories

Interventions

NameTypeDescription
DEPAKOTE® Tablets, 500 MGDRUG1 x 500 mg Tablet, under fed conditions
DIVALPROEX SODIUM DELAYED-RELEASE TABLETS, USP, 500 MGDRUG1 x 500 mg Tablet, under fed conditions
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Age: 18 years and older. 2. Sex: Females not of child bearing potential and males. * No hormonal contraceptives or hormonal replacement therapies are permitted in this study. * Women will not be considered of childbearing potential if one of the following is reported a...

Countries:United States
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Frequently asked questions about DIVALPROEX, USP

What is DIVALPROEX, USP?

DIVALPROEX, USP is a small molecule drug developed by Viatris Inc. (ticker VTRS). It is being studied in Phase 1 clinical trials in healthy adult volunteers. The drug is also known as divalproex sodium delayed-release tablets, USP, 500 mg.

What does DIVALPROEX, USP target?

DIVALPROEX, USP targets ALDH5A1 and acts as an inhibitor of this enzyme. ALDH5A1 is the molecular target of the drug, and its inhibition is the basis for its pharmacological activity in the studied setting.

Who makes DIVALPROEX, USP?

DIVALPROEX, USP is developed by Viatris Inc., which trades under the ticker symbol VTRS. Viatris is the company responsible for the clinical development of this drug candidate.

What phase is DIVALPROEX, USP in?

DIVALPROEX, USP is in Phase 1 clinical development. It is an investigational drug and has not been approved by the FDA for any indication. The Phase 1 trials have been completed, and no active trials are currently listed.

What clinical trials is DIVALPROEX, USP in?

DIVALPROEX, USP has been evaluated in two completed Phase 1 trials: NCT01184391, a bioequivalence study of divalproex sodium delayed-release tablets, 500 mg, with 17 participants, and NCT01183676, a fed bioequivalence study of the same formulation, with 20 participants. Both enrolled healthy adults in the United States.