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iNexin

Phase 1

Dry Eye Disease | Small molecule | Ophthalmology |United Therapeutics Corporation|Last Updated: Mar 4, 2022

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment30

FDA Designations

No designations recorded

Clinical trial landscape

iNexin · 1 trial · 1 indication

Phase 1 1
NCT05031806Evaluation of the Safety, Tolerability and Efficacy of iNexin™ for the Treatment of the Signs and Symptoms Associated With Dry Eye DiseaseDry Eye Disease
COMPLETED30 Analytics
PHASE1COMPLETED
Evaluation of the Safety, Tolerability and Efficacy of iNexin™ for the Treatment of the Signs and Symptoms Associated With Dry Eye Disease
Dry Eye DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Evaluation of the safety of iNexin™
Through study completion, an average of 24 days

Assessed using: Visual Acuity (VA) (ETDRS), Slit-lamp biomicroscopy, Adverse Event Query, Dilated Fundoscopy Interocular Pressure

Evaluation of the tolerability of iNexin™
Through study completion, an average of 24 days

Assessed using: Ora Calibra Drop Comfort Assessments

Secondary Endpoints

Comparison of the efficacy of iNexin™ to Vehicle for the treatment of the signs and symptoms associated with dry eye disease
Through study completion, an average of 24 days
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
iNexin™ (0.08% aCT1)EXPERIMENTAL36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle. During a 7-day study run-in period prior to randomization, all subjects will receive Vehicle eye drops (Vehicle) bilaterally BID (from Visit 1 to the evening before Visit 2).
iNexin™ (0.4% aCT1)EXPERIMENTAL36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle. During a 7-day study run-in period prior to randomization, all subjects will receive Vehicle eye drops (Vehicle) bilaterally BID (from Visit 1 to the evening before Visit 2).
iNexin™ (2.0% aCT1)EXPERIMENTAL36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle. During a 7-day study run-in period prior to randomization, all subjects will receive Vehicle eye drops (Vehicle) bilaterally BID (from Visit 1 to the evening before Visit 2).
Vehicle (eye drop formulation without aCT1)PLACEBO_COMPARATOR36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle. During a 7-day study run-in period prior to randomization, all subjects will receive Vehicle eye drops (Vehicle) bilaterally BID (from Visit 1 to the evening before Visit 2).

Interventions

NameTypeDescription
iNexin™ (0.08% aCT1)DRUG36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle.randomized 7:3 for each active concentration to Vehicle.
iNexin™ (0.4% aCT1)DRUG36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle.
iNexin™ (2.0% aCT1)DRUG36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle.
Vehicle (eye drop formulation without aCT1)DRUG36 eligible subjects will be randomized to Vehicle or one of three concentrations of iNexin™ to be administered bilaterally BID for 15 days (from Visit 2 to the evening of Visit 4). Subjects will be randomized 2:1 for each active concentration to Vehicle. During a 7-day study run-in period prior to randomization, all subjects will receive Vehicle eye drops (Vehicle) bilaterally BID (from Visit 1 to the evening before Visit 2).
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: Subjects must meet all the following requirements to be eligible for enrollment into the study. 1. Be at least 18 years of age; 2. Provide written informed consent; 3. Have a self-reported history of dry eye for at least 6 months prior to Visit 1; 4. Have a history of use or de...

Countries:United States
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Competitive Landscape -Dry Eye Disease 7 trials

Frequently asked questions about iNexin

What is iNexin used for?

iNexin is an investigational small molecule being developed for the treatment of dry eye disease. It is designed to address both the signs and symptoms associated with the condition. As of the latest available information, iNexin is in Phase 1 clinical development and has not been approved by regulatory authorities.

Who is developing iNexin?

iNexin is being developed by United Therapeutics Corporation, a publicly traded company listed on the NASDAQ under the ticker symbol UTHR. The company is conducting clinical research to evaluate the safety, tolerability, and efficacy of iNexin for dry eye disease.

What phase is iNexin in?

iNexin is currently in Phase 1 clinical development. A Phase 1 trial has been completed, which evaluated the safety, tolerability, and efficacy of iNexin in patients with dry eye disease. The drug remains investigational and is not yet approved for commercial use.

What clinical trials has iNexin been in?

iNexin has been studied in one completed Phase 1 clinical trial registered as NCT05031806. This trial, conducted in the United States, enrolled 30 participants with dry eye disease. The study was randomized, double-blind, and placebo-controlled, and it evaluated the safety, tolerability, and efficacy of iNexin for treating the signs and symptoms of dry eye disease.

Is iNexin FDA approved?

iNexin is not FDA approved. It is an investigational drug that has completed a Phase 1 clinical trial for dry eye disease. Further clinical development and regulatory review would be required before iNexin could be considered for approval.