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Febuxostat IR

Phase 3

Gout | Small molecule | Musculoskeletal |Takeda Pharmaceutical Company Limited|Last Updated: Nov 3, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDDMCBiomarker
Total Trials2
Total Enrollment1,979
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02139046Efficacy and Safety of Extended Release and Immediate Release Febuxostat in Participants With GoutPHASE3 COMPLETED 1,790Apr 1, 2014Nov 1, 2015Nov 3, 2016192 United States
NCT02128490Efficacy and Safety of Extended Release and Immediate Release Febuxostat in Participants With Gout and Moderate Renal ImpairmentPHASE2 COMPLETED 189May 1, 2014Oct 1, 2015Nov 3, 201689 United States
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Study Endpoints
Primary Endpoints
Percentage of Participants With Serum Urate <5.0 mg/dL at Month 3
Month 3
Secondary Endpoints
Percentage of Participants With at Least One Gout Flare Requiring Treatment
Baseline to Month 3
Percentage of Participants With Serum Urate <6.0 mg/dL at Month 3
Month 3
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Febuxostat IR 40 mgACTIVE_COMPARATORFebuxostat Immediate Release (IR) 40 mg over-encapsulated tablet, orally, once daily, and colchicine 0.6 mg tablet, orally, every day (for participants with estimated glomerular filtration rate (eGFR) ≥ 60 mL/min) or every other day (if eGFR ≥ 15 - ≤ 59 mL/min), or, alternatively, if colchicine is not tolerated and the subject's eGFR is ≥ 50 mL/min, naproxen 250 mg tablets, orally, twice a day and lansoprazole 15 mg capsule, orally once daily, for 3 months.
Febuxostat IR 80 mgACTIVE_COMPARATORFebuxostat IR 80 mg over-encapsulated tablet, orally, once daily, and colchicine 0.6 mg tablet, orally, every day or every other day, or, alternatively, if colchicine is not tolerated and the subject's eGFR is ≥ 50 mL/min, naproxen 250 mg tablets, orally, twice a day and lansoprazole 15 mg capsule, orally once daily, for 3 months.
Febuxostat XR 40 mgEXPERIMENTALFebuxostat Extended Release (XR) 40 mg over-encapsulated capsule, orally, once daily, and colchicine 0.6 mg tablet, orally, every day or every other day, or, alternatively, if colchicine is not tolerated and the subject's eGFR is ≥ 50 mL/min, naproxen 250 mg tablets, orally, twice a day and lansoprazole 15 mg capsule, orally once daily, for 3 months.
Febuxostat XR 80 mgEXPERIMENTALFebuxostat XR 80 mg over-encapsulated capsule, orally, once daily, and colchicine 0.6 mg tablet, orally, every day or every other day, or, alternatively, if colchicine is not tolerated and the subject's eGFR is ≥ 50 mL/min, naproxen 250 mg tablets, orally, twice a day and lansoprazole 15 mg capsule, orally once daily, for 3 months.
PlaceboPLACEBO_COMPARATORFebuxostat placebo-matching capsule, orally, once daily, and colchicine 0.6 mg tablet, orally, every day or every other day, or, alternatively, if colchicine is not tolerated and the subject's eGFR is ≥ 50 mL/min, naproxen 250 mg tablets, orally, twice a day and lansoprazole 15 mg capsule, orally once daily, for 3 months.
Interventions
NameTypeDescription
Febuxostat IRDRUGFebuxostat IR over-encapsulated tablets
Febuxostat XRDRUGFebuxostat XR over-encapsulated capsules
Febuxostat placeboDRUGFebuxostat placebo-matching capsules
ColchicineDRUGColchicine tablets
NaproxenDRUGNaproxen tablets
LansoprazoleDRUGLansoprazole capsules
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites192

Inclusion Criteria: 1. In the opinion of the investigator, the participant is capable of understanding and complying with protocol requirements. 2. The participant or, when applicable, the participant's legally acceptable representative signs and dates a written, informed consent form and any requi...

Countries:United States
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Competitive Landscape -Gout 5 trials