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SAR439459

Phase 1

Malignant Solid Tumor | Monoclonal antibody | Oncology |Sanofi|Last Updated: Aug 7, 2024

Target and mechanism

Molecular targetTGFb
Target classProtein
ModalityMonoclonal antibody

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLEDDMC
Total Trials1
Total Enrollment161

FDA Designations

No designations recorded

Clinical trial landscape

SAR439459 · 1 trial · 1 indication

Phase 1 1
NCT03192345A First-in-human Study of the Safety, Pharmacokinetics, Pharmacodynamics and Anti-tumor Activity of SAR439459 Monotherapy and Combination of SAR439459 and Cemiplimab in Patients With Advanced Solid TumorsMalignant Solid Tumor
COMPLETED161 Analytics
PHASE1COMPLETED
A First-in-human Study of the Safety, Pharmacokinetics, Pharmacodynamics and Anti-tumor Activity of SAR439459 Monotherapy and Combination of SAR439459 and Cemiplimab in Patients With Advanced Solid Tumors
Malignant Solid TumorUnlock trial analytics

Study Endpoints

Primary Endpoints

Incidence of Dose Limiting Toxicities (DLTs)
Through the end of 1 or 2 cycles, total duration up to 6 weeks (for Part 1A each cycle is 2 weeks; for Part 1B each cycle is 2 or 3 weeks)

Incidence of DLTs at Cycle 1 and/or 2 in Parts 1A and 1B.

Objective Response Rate (ORR) for Part 2B
Continuous throughout study assessment (up to approximately 1 year)

Efficacy as documented by ORR will be assessed by evaluation of antitumor response information according to RECIST 1.1 (Part 2B).

Secondary Endpoints

Overall safety profile
Continuous throughout study assessment (up to approximately 1 year)
Progression free survival (PFS)
Continuous throughout study assessment (up to approximately 1 year)
Time to progression (TTP)
Continuous throughout study assessment (up to approximately 1 year)
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Dose Escalation SAR439459 monotherapyEXPERIMENTALSAR439459 administered intravenously every 2 weeks in a 14-day cycle with escalating doses
Dose Expansion SAR439459 monotherapyEXPERIMENTALSAR439459 administered intravenously every 3 weeks in a 21-day cycle with the previously determined recommended doses as the patients will be randomized to 2 different doses
Dose Escalation SAR439459 + cemiplimab combinationEXPERIMENTALSAR439459 + cemiplimab combination administered intravenously every 2 weeks in a 14-day cycle or every 3 weeks in a 21-day cycle with escalating SAR439459 doses and cemiplimab
Dose Expansion SAR439459 + cemiplimab combinationEXPERIMENTALSAR439459 + cemiplimab combination administered intravenously every 3 weeks in a 21-day cycle with previously determined SAR439459 doses and cemiplimab

Interventions

NameTypeDescription
SAR439459BIOLOGICALPharmaceutical form: powder for solution for infusion Route of administration: intravenous infusion
Cemiplimab REGN2810DRUGPharmaceutical form: solution for infusion Route of administration: intravenous infusion
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites34

Inclusion criteria: Dose escalation (Part 1A and Part 1B) * Patients with histologically confirmed, advanced unresectable or metastatic solid tumor whom in the opinion of the Investigator does not have a suitable alternative therapy. Dose expansion (Part 2A) * Patients with histologically confir...

Countries:United StatesAustraliaBelgiumCanadaEstoniaFranceGermanyItalyNetherlandsSouth KoreaSpainTaiwanUnited Kingdom
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Frequently asked questions about SAR439459

What is SAR439459 used for?

SAR439459 is an investigational monoclonal antibody being studied for the treatment of malignant solid tumors. It is currently in Phase 1 clinical development, meaning it has not yet been approved by regulatory authorities and remains under investigation for safety and efficacy.

What does SAR439459 target?

SAR439459 targets TGFb, a protein involved in tumor growth and immune regulation. By binding to TGFb, the antibody is designed to modulate its activity, which may have anti-tumor effects. This mechanism is being evaluated in the context of advanced solid tumors.

Who makes SAR439459?

SAR439459 is being developed by Sanofi, a global biopharmaceutical company listed on the stock exchange under the ticker symbol SNY. Sanofi is conducting clinical trials to evaluate the safety and efficacy of this investigational drug in patients with malignant solid tumors.

What phase is SAR439459 in?

SAR439459 is in Phase 1 clinical development. This early-stage trial is designed to assess the safety, pharmacokinetics, pharmacodynamics, and anti-tumor activity of the drug. It is an investigational agent and has not yet received regulatory approval for any indication.

What clinical trials is SAR439459 in?

SAR439459 has been studied in a Phase 1 clinical trial registered as NCT03192345. This first-in-human study evaluated SAR439459 as a monotherapy and in combination with cemiplimab in patients with advanced solid tumors. The trial was completed and enrolled 161 participants across multiple countries.

Is SAR439459 the same as any other drug?

SAR439459 is a distinct investigational monoclonal antibody developed by Sanofi. It is being studied alone and in combination with cemiplimab, which is a separate PD-1 inhibitor. No alternative names for SAR439459 have been reported in the clinical trial information.