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Tofacitinib/g

Phase 2

Dermatitis, Atopic | Small molecule | Dermatology |Pfizer, Inc.|Last Updated: Nov 25, 2015

Target and mechanism

Molecular targetJAK3, JAK1, JAK2, TYK2
Target classInhibitor
ModalitySmall molecule

Also known as tofacitinib

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment69

FDA Designations

No designations recorded

Clinical trial landscape

Tofacitinib/g · 2 trials · 3 indications

Phase 2 2
NCT02001181Tofacitinib Ointment For Atopic Dermatitis (Atopic Eczema)Dermatitis, Atopic
COMPLETED69 Analytics
NCT01831466Tofacitinib Ointment For Chronic Plaque PsoriasisPsoriasis Vulgaris
COMPLETED476 Analytics
PHASE2COMPLETED
Tofacitinib Ointment For Atopic Dermatitis (Atopic Eczema)
Dermatitis, AtopicUnlock trial analytics
PHASE2COMPLETED
Tofacitinib Ointment For Chronic Plaque Psoriasis
Psoriasis VulgarisUnlock trial analytics

Study Endpoints

Primary Endpoints

Percent Change From Baseline in Eczema Area and Severity Index (EASI) Total Score at Week 4
Baseline (pre-dose on Day 1) and Week 4

The EASI quantifies the severity of a participant's atopic dermatitis based on both lesion severity and the percent of BSA affected. The EASI is a composite scoring by the atopic dermatitis clinical evaluator of the degree of erythema, induration/papulation, excoriation, and lichenification (each scored separately) for each of 4 body regions, with adjustment for the percent of BSA involved for each body region and for the proportion of the body region to the whole body. The EASI score can vary in increments of 0.1 and range from 0.0 to 72.0, with higher scores representing greater severity of atopic dermatitis. What is reported is the percent change from baseline in EASI scores.

Percentage of Participants Achieving a PGA-C Response of Clear (0) or Almost Clear (1) and Greater Than or Equal to (≥) 2 Grade/Point Improvement From Baseline at Week 12
Baseline, Week 12

Clinical signs of plaque psoriasis (erythema \[E\], induration \[I\], and scaling \[S\]) were scored separately according to a 5-point severity scale (0 to 4) to provide PGA subscores, which described the overall severity of each clinical sign. The PGA-C was a static assessment; i.e., without regard to a previous assessment. The PGA subscores are then summed and averaged after which the total average was rounded to the nearest whole number to determine the PGA-C score and category. A higher score indicated a higher level of severity. 0 is equal to (=) cleared except for any residual discoloration and 1=almost clear, majority of lesions had individual scores for E+I+S that when summed, averaged, and rounded equaled 1.

Percentage of Participants Achieving a PGA-C Response of Clear (0) or Almost Clear (1) and ≥2 Grade/Point Improvement From Baseline at Week 8
Baseline, Week 8

Clinical signs of plaque psoriasis (E, I, and S) were scored separately according to a 5-point severity scale (0 to 4) to provide PGA subscores, which described the overall severity of each clinical sign. The PGA-C was a static assessment; i.e., without regard to a previous assessment. The PGA subscores are then summed and averaged after which the total average was rounded to the nearest whole number to determine the PGA-C score and category. A higher score indicated a higher level of severity. 0 is equal to (=) cleared except for any residual discoloration and 1=almost clear, majority of lesions had individual scores for E+I+S that when summed, averaged, and rounded equaled 1.

Secondary Endpoints

Proportion of Participants Achieving Physician's Global Assessment (PGA) Response of Clear or Almost Clear at Week 4
Week 4
Proportion of Participants With Response of Clear or Almost Clear and Greater Than or Equal to (>=) 2 Grade/Point Improvement From Baseline at Week 4
Baseline (pre-dose on Day 1) and Week 4
Percent Change From Baseline in Body Surface Area (BSA) Efficacy at Week 4
Baseline (pre-dose on Day 1) and Week 4
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Treatment group AEXPERIMENTAL -
Treatment BPLACEBO_COMPARATOR -
Treatment Group BEXPERIMENTAL -
Treatment Group CPLACEBO_COMPARATOR -
Treatment Group DEXPERIMENTAL -
Treatment Group EEXPERIMENTAL -
Treatment Group FPLACEBO_COMPARATOR -

Interventions

NameTypeDescription
Tofacitinib ointment 20mg/gDRUGTofacitinib ointment 20mg/g twice daily (BID) for 4 weeks
Placebo ointment (Vehicle)DRUGPlacebo ointment (vehicle) twice daily (BID) for 4 weeks
tofacitinib ointment 20 mg/gDRUGtofacitinib ointment 20 mg/g BID (twice daily) for 12 weeks
tofacitinib ointment 10 mg/gDRUGtofacitinib ointment 10 mg/g BID (twice daily) for 12 weeks
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Eligibility Criteria

Age Range18 Years to 60 Years
SexALL
Healthy VolunteersNo
Study Sites5

Inclusion Criteria: * Have a clinical diagnosis of atopic dermatitis (also known as atopic eczema) for at least 6 months prior to Day 1 that has been clinically stable for at least 1 month prior to Day 1 and is confirmed to be atopic dermatitis according to the criteria of Hanifin and Rajka. * Have...

Countries:CanadaUnited StatesDenmarkPoland
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Frequently asked questions about Tofacitinib/g

What is CP-690-550 used for?

CP-690-550, also known as tofacitinib, is an investigational small molecule being studied for the treatment of psoriasis, juvenile idiopathic arthritis, rheumatoid arthritis, psoriatic arthritis, and ankylosing spondylitis. It is in Phase 2 clinical development for these immunology indications.

What does CP-690-550 target?

CP-690-550 is a kinase inhibitor, belonging to the -tinib class of drugs. It targets kinases, which are enzymes involved in cell signaling pathways. By inhibiting these kinases, it modulates immune responses relevant to the autoimmune and inflammatory conditions it is being studied for.

Who makes CP-690-550?

CP-690-550 is being developed by Pfizer, Inc., a biopharmaceutical company. Pfizer is the sponsor of the clinical trials for this drug, which is also known as tofacitinib.

What phase is CP-690-550 in?

CP-690-550 is in Phase 2 clinical development for its investigational indications. It is not approved by the FDA and remains under study. The drug is being evaluated in clinical trials to assess its safety and efficacy for conditions such as rheumatoid arthritis and psoriasis.

What clinical trials is CP-690-550 in?

CP-690-550 has completed four Phase 1 clinical trials, including NCT01599377, NCT02487433, NCT04111614, and NCT04403776. These trials enrolled healthy volunteers to study bioequivalence, food effects, and pharmacokinetics of different formulations. No active trials are currently listed.

Is CP-690-550 the same as tofacitinib?

Yes, CP-690-550 is also known as tofacitinib. The drug is referred to by both names in clinical research and development contexts. Pfizer is developing this compound under the name tofacitinib.