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Ga-PSMA-11

Phase 1

Metastatic Neuroendocrine Prostate Cancer | Small molecule | Oncology |Novartis AG|Last Updated: Jul 24, 2026

Target and mechanism

Molecular targetPSMA
Target classProtein
ModalitySmall molecule

Also known as [68Ga]Ga-PSMA-11

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment31

FDA Designations

No designations recorded

Clinical trial landscape

Ga-PSMA-11 · 1 trial · 1 indication

Phase 1 1
NCT06379217NEPC Study: An Exploratory Safety and Efficacy Study With PSMA, SSTR2 and GRPR Targeted Radioligand Therapy in Metastatic Neuroendocrine Prostate Cancer.Metastatic Neuroendocrine Prostate Cancer
ACTIVE NOT_RECRUITING31 Analytics
PHASE1ACTIVE NOT_RECRUITING
NEPC Study: An Exploratory Safety and Efficacy Study With PSMA, SSTR2 and GRPR Targeted Radioligand Therapy in Metastatic Neuroendocrine Prostate Cancer.
Metastatic Neuroendocrine Prostate CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Number/extent of lesions with at least a moderate uptake of any of the Radioligand Imaging (RLI)
Baseline (baseline imaging is performed during the 42 day screening period)

Number/extent of lesions with at least a moderate update of any of the RLIs according to visual assessment scoring scale on each corresponding targeted PET/CT scan based on blinded independent central review (BICR) assessment.

Percentage changes in quantitative PET parameters.
Post-Baseline (from date of baseline imaging scans to post-baseline scans, at least 6 weeks after receiving the first cycle of radioligand treatment)

Percentage changes in quantitative PET/CT parameters (SUVmax, SUVmean, SUVpeak, target-positive Tumor Volume (target -TV), Total Lesion (target (TL-target)\] and changes in number of target-positive lesions (as per visual assessment) on each corresponding target PET/CT based on BICR.

Secondary Endpoints

Overall Response Rate (ORR)
From date of assignment to one of the treatment arms until date of radiographic progression or date of death from any cause, whichever comes first, assessed up to approximately 31 months
Disease Control Rate (DCR)
From date of assignment to one of the treatment arms until date of radiographic progression or date of death from any cause, whichever comes first, assessed up to approximately 31 months
Duration of response (DOR)
From first documented evidence of CR or PR (the response prior to confirmation) until time of documented disease progression or death due to any cause, whichever comes first, assessed up to approximately 31 months
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
PSMA-predominant Neuroendocrine prostate cancer (NEPC)EXPERIMENTAL -
Somatostatin Receptor 2 (SSTR2)-predominant NEPCEXPERIMENTAL -
Gastrin Releasing Peptide Receptor (GRPR)-predominant NEPCEXPERIMENTAL -

Interventions

NameTypeDescription
[68Ga]Ga-PSMA-11DRUG\[68Ga\]Ga-PSMA-11 will be administered as a single intravenous dose of approximately 150 MBq (4 mCi) to be administered during baseline imaging and at any time ≥ 6 weeks after first RLT dose. Sites should consider doing PET/CT imaging with RLT corresponding RLI as the first of three PET/CT scans. Administered dose should not be lower than 111 MBq (3 mCi) or higher than 259 MBq (7 mCi)
[68Ga]GA-DOTA-TATEDRUG\[68Ga\]Ga-DOTA-TATE will be administered as a single intravenous dose to be administered during baseline imaging and at any time ≥ 6 weeks after first RLT dose. Sites should consider doing PET/CT imaging with RLT corresponding RLI as the first of three PET/CT scans. within a range of 100-200MBq (2.7-5.4 mCi)
[68Ga]Ga-NeoBDRUG\[68Ga\]Ga-NeoB will be administered as a single intravenous dose to be administered during baseline imaging and at any time ≥ 6 weeks after first RLT dose. Sites should consider doing PET/CT imaging with RLT corresponding RLI as the first of three PET/CT scans. within a range of 150-250 MBq (4.1-6.8 mCi).
[177Lu]Lu-PSMA-617DRUG\[177Lu\]Lu-PSMA-617 will be administered as an intravenous infusion at a dose of 7.4 GBq (200mCi) (+/- 10%), every 6 weeks for 6 cycles.
[177Lu]Lu-DOTA-TATEDRUG\[177Lu\]Lu-DOTA-TATE will be administered as an intravenous infusion at a dose of 7.4 GBq (200mCi) (+/- 10%) every 6 weeks for 6 cycles.
[177Lu]Lu-NeoBDRUG\[177Lu\]Lu-NeoB will be administered as an intravenous infusion at a dose of 9.25 GBq (250mCi) every 6 weeks for 6 cycles
L-Lysine HCl-L-Arginine HCl, 2.5 %,DRUGsterile solution for infusion Lysine HCl-Arginine HCl, 2.5 % (1L)
Gonadotropin-releasing hormone (GnRH) analoguesDRUGAnatomical Therapeutic Chemical \[ATC\] code L02AE
GnRH antagonistsDRUGabarelix, degarelix, or relugolix
Antiemetics & antinauseantsDRUGATC code A04A
MetoclopramideDRUGATC code A03FA01
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Eligibility Criteria

Age Range18 Years to 100 Years
SexMALE
Healthy VolunteersNo
Study Sites9

Key Inclusion criteria: * Participants must have metastatic prostate cancer with neuroendocrine differentiation as determined by at least one of the following: * Histologically small cell or neuroendocrine cancer from a primary prostate or metastatic biopsy confirmed by local laboratory. * Exp...

Countries:United StatesFranceGermanySpainUnited Kingdom
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Recent Changes (Last 90 Days)

LOWJul 24, 2026NCT06379217primaryCompletionDate: changed
LOWJul 24, 2026NCT06379217primaryCompletionDate: changed
LOWJul 10, 2026NCT06379217lastUpdatePostDate: changed
LOWJul 10, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 10, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 10, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 4, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 4, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 4, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 4, 2026NCT06379217lastUpdatePostDate: changed
LOWJun 4, 2026NCT06379217lastUpdatePostDate: changed

Frequently asked questions about Ga-PSMA-11

What is Ga-PSMA-11 used for in metastatic neuroendocrine prostate cancer?

Ga-PSMA-11 is an investigational small molecule being studied for use in metastatic neuroendocrine prostate cancer. It is a PSMA-targeted radioligand therapy currently in Phase 1 clinical development. The drug is being evaluated in an exploratory safety and efficacy study for this condition.

What does Ga-PSMA-11 target?

Ga-PSMA-11 targets PSMA, a protein that is expressed on prostate cancer cells. By binding to PSMA, the drug is designed to deliver radiation therapy directly to cancer cells. This targeted approach is being investigated for the treatment of metastatic neuroendocrine prostate cancer.

Who makes Ga-PSMA-11?

Ga-PSMA-11 is being developed by Novartis AG, a global healthcare company traded on the New York Stock Exchange under the ticker symbol NVS. The company is conducting clinical trials to evaluate the safety and efficacy of this investigational drug in metastatic neuroendocrine prostate cancer.

What phase is Ga-PSMA-11 in?

Ga-PSMA-11 is in Phase 1 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities and is still being studied in clinical trials. The current trial is an exploratory safety and efficacy study in patients with metastatic neuroendocrine prostate cancer.

What clinical trials is Ga-PSMA-11 in?

Ga-PSMA-11 is being studied in a Phase 1 clinical trial with the identifier NCT06379217. This trial is titled 'NEPC Study: An Exploratory Safety and Efficacy Study With PSMA, SSTR2 and GRPR Targeted Radioligand Therapy in Metastatic Neuroendocrine Prostate Cancer.' The study is active but not recruiting, with an enrollment of 31 patients.

Is Ga-PSMA-11 the same as [68Ga]Ga-PSMA-11?

Yes, Ga-PSMA-11 is also known as [68Ga]Ga-PSMA-11. Both names refer to the same investigational drug being developed by Novartis AG for the treatment of metastatic neuroendocrine prostate cancer. The drug is a PSMA-targeted radioligand therapy currently in Phase 1 clinical trials.