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BKM120

Phase 2

Brain Metastases | Small molecule | Oncology |McKesson Corporation|Last Updated: Feb 7, 2022

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment10

FDA Designations

No designations recorded

Clinical trial landscape

BKM120 · 1 trial · 3 indications

Phase 2 1
NCT02000882STAR Cape+BKM120 MBC With Brain MetBrain Metastases
COMPLETED10 Analytics
PHASE2COMPLETED
STAR Cape+BKM120 MBC With Brain Met
Brain MetastasesUnlock trial analytics

Study Endpoints

Primary Endpoints

Clinical Benefit Rate (CBR)
until disease progression (assessed by RECIST 1.1), unacceptable toxicity, death, or discontinuation from study for any other reason, up to 2 years from date of patient registration

CBR in the patients following WBRT or SRS or both will be the primary endpoint and is calculated as the total number of responders (CR or PR, assessed by RECIST 1.1) plus stable disease greater than or equal to 24 weeks (CR + PR + SD ≥ 24 weeks) divided by the total number of evaluable patients. Complete Response (CR): Disappearance of all target lesions. Any pathological lymph nodes (whether target or non-target) must have reduction in short axis to \<10 mm. Partial Response (PR): At least a 30% decrease in the sum of diameters of target lesions, taking as reference the baseline sum diameters.

Secondary Endpoints

Objective Response Rate (ORR)
until disease progression (assessed by RECIST 1.1), unacceptable toxicity, death, or discontinuation from study for any other reason, up to 2 years from date of patient registration
Median Time to Progression
until disease progression (assessed by RECIST 1.1), unacceptable toxicity, death, or discontinuation from study for any other reason, up to 2 years from date of patient registration
Median Overall Survival
up to 2 years from date of patient registration
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BKM120 plus CapecitabineEXPERIMENTALBKM120 will be administered at a dose of 100 mg orally (PO) daily. Capecitabine will be administered at a dose of 1000 mg/m2 orally (PO) twice a day (rounded down to the nearest 500 mg pill) 14 days on and 7 days off. For patients with HER2+ MBC only, standard every 3-weekly trastuzumab (6 mg/kg IV) will be added to the capecitabine/BKM120.

Interventions

NameTypeDescription
BKM120DRUG -
capecitabineDRUG -
TrastuzumabDRUG -
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Eligibility Criteria

Age Range18 Years to N/A
SexFEMALE
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. Age ≥ 18 years 2. Female 3. Histologically and/or cytologically confirmed diagnosis of inoperable metastatic breast cancer 4. ER+/HER2- OR HER2+ OR triple-negative breast cancer, assessed as ER-, PgR-, and HER2-negative by local laboratory testing; HER2 negative status (based...

Countries:United States
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Frequently asked questions about BKM120

What is BKM120 used for?

BKM120 is an investigational small molecule being studied for the treatment of brain metastases in patients with metastatic breast cancer. It is a Phase 2 oncology drug that was evaluated in a completed clinical trial in the United States.

Who makes BKM120?

BKM120 is being developed by McKesson Corporation, which trades under the ticker symbol MCK. The company conducted a Phase 2 clinical trial of the drug in patients with brain metastases from breast cancer.

What phase is BKM120 in?

BKM120 is in Phase 2 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities and is still being studied for safety and efficacy in clinical trials.

What clinical trials is BKM120 in?

BKM120 was studied in a single completed Phase 2 clinical trial with the identifier NCT02000882, titled 'STAR Cape+BKM120 MBC With Brain Met.' The trial enrolled 10 female patients aged 18 years and older with brain metastases and metastatic breast cancer in the United States.

Is BKM120 the same as STAR Cape?

No, BKM120 is not the same as STAR Cape. STAR Cape is the name of the clinical trial, not an alternative name for the drug. The trial combined BKM120 with capecitabine, a chemotherapy agent, to treat metastatic breast cancer with brain metastases.