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LY2584702 Reference Formulation

Phase 1

Healthy Participants | Small molecule | Other |Eli Lilly and Company|Last Updated: Jan 22, 2019

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment29
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01372085Single Dose Study in Healthy Participants to Investigate the Safety and Absorption of LY2584702PHASE1 COMPLETED 29Jun 1, 2011Sep 1, 2011Jan 22, 20191 Singapore
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Study Endpoints
Primary Endpoints
Pharmacokinetics: Maximum Observed Plasma Concentration (Cmax)
Part A: Day 1 and Part B: Periods 1 to 4, Day 1 [Predose, 1 hour (h), 3 h, 4 h, 6 h, 10 h, 24 h, 48 h postdose]

The Cmax following a single oral dose of LY2584702 test formulation \[TF (tablet)\] or reference formulation \[RF (capsule)\] is reported.

Secondary Endpoints
Pharmacokinetics, Area Under the Concentration-Time Curve (AUC)
Part A: Day 1 and Part B: Periods 1 to 4, Day 1 [Predose, 1 hour (h), 3 h, 4 h, 6 h, 10 h, 24 h, 48 h postdose]
Part B: Baseline-Adjusted Change-From-Predose in the Concentration of Lipids (Total Cholesterol)
Part B: Baseline [Periods 1 and 4a (Day -1)], Periods 3, 4a (Day 1). Lipid concentration measurements were performed at time point 0 and 1 hour (h), 3 h, 4 h, 6 h, 10 h, and 24 h.
Part A: QT Interval Corrected by Fridericia's Formula (QTcF) Change From Baseline to Day 1
Part A: Baseline [Day 1 (Predose)] and Day 1 (3 h, 4 h, 6 h, and 24 h postdose)
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part A: 25 mg RFEXPERIMENTALA single 25 mg dose of LY2584702 RF
Part A: PlaceboPLACEBO_COMPARATORPlacebo taken orally
Part B: Sequence 1EXPERIMENTALA single 10 mg dose of LY2584702 TF during the first intervention period, followed by placebo in the second intervention period, followed by a single dose of 50 mg TF in the third intervention period, followed by either an open-label single dose of 50 mg TF after a high fat breakfast (Period 4a) OR placebo or escalated dose of TF in the fasted state (Period 4b). There will be a washout period of at least 3 days between periods.
Part B: Sequence 2EXPERIMENTALPlacebo during the first intervention period, followed by a single dose of 50 mg RF in the second intervention period, followed by a single dose of 50 mg TF in the third intervention period, followed by either an open-label single dose of 50 mg TF after a high fat breakfast (Period 4a) OR placebo or escalated dose of TF in the fasted state (Period 4b). There will be a washout period of at least 3 days between periods.
Part B: Sequence 3EXPERIMENTALA single 10 mg dose of LY2584702 TF during the first intervention period, followed by a single dose of 50 mg RF in the second intervention period, followed by a single dose of 50 mg TF in the third intervention period, followed by either an open-label single dose of 50 mg TF after a high fat breakfast (Period 4a) OR placebo or escalated dose of TF in the fasted state (Period 4b). There will be a washout period of at least 3 days between periods.
Part B: Sequence 4EXPERIMENTALA single 10 mg dose of LY2584702 TF during the first intervention period, followed by a single dose of 50 mg RF in the second intervention period, followed by placebo in the third intervention period, followed by either an open-label single dose of 50 mg TF after a high fat breakfast (Period 4a) OR placebo or escalated dose of TF in the fasted state (Period 4b). There will be a washout period of at least 3 days between periods.
Interventions
NameTypeDescription
LY2584702 Reference FormulationDRUGAdministered orally
LY2584702 Test FormulationDRUGAdministered orally
PlaceboDRUGAdministered orally
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Eligibility Criteria
Age Range21 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: Male participants: • Agree to use a reliable method of birth control during the study and for at least 1 month following the last dose of study drug Female participants: • Women not of childbearing potential due to surgical sterilization (hysterectomy or bilateral oophorectom...

Countries:Singapore
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