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LY2409021 Reference Form

Phase 1

Healthy Volunteers | Small molecule | Other |Eli Lilly and Company|Last Updated: Mar 11, 2019

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment35

FDA Designations

No designations recorded

Clinical trial landscape

LY2409021 Reference Form · 1 trial · 1 indication

Phase 1 1
NCT01354496A Study of LY2409021 Formulations and the Effect of FoodHealthy Volunteers
COMPLETED35 Analytics
PHASE1COMPLETED
A Study of LY2409021 Formulations and the Effect of Food
Healthy VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

Pharmacokinetics, Area Under the Concentration-Time Curve (AUC): Medium Test Form to Reference Form
Periods 1, 2, 3 (predose, 0.5, 1, 2, 4, 6, 8, 10, 12, 18, 24, 36, 48, 72, 96, 144, 192, 240, 288, and 336 hours postdose)

AUC from time 0 to infinity (AUC0-∞).

Pharmacokinetics, Maximum Concentration (Cmax): Medium Test Form to Reference Form
Periods 1, 2, 3 (predose, 0.5, 1, 2, 4, 6, 8, 10, 12, 18, 24, 36, 48, 72, 96, 144, 192, 240, 288, and 336 hours postdose)

Secondary Endpoints

Pharmacokinetics, Area Under the Concentration-Time Curve (AUC): Standardized High Fat Meal to Fasting
Periods 1, 2, 3 (predose, 0.5, 1, 2, 4, 6, 8, 10, 12, 18, 24, 36, 48, 72, 96, 144, 192, 240, 288, and 336 hours postdose)
Pharmacokinetics, Maximum Concentration (Cmax): Standardized High Fat Meal to Fasting
Periods 1, 2, 3 (predose, 0.5, 1, 2, 4, 6, 8, 10, 12, 18, 24, 36, 48, 72, 96, 144, 192, 240, 288, and 336 hours postdose)
Pharmacokinetics, Time to Maximum Concentration (Tmax)
Periods 1, 2, 3 (predose, 0.5, 1, 2, 4, 6, 8, 10, 12, 18, 24, 36, 48, 72, 96, 144, 192, 240, 288, and 336 hours postdose)
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Cohort 1 - LY2409021 reference formEXPERIMENTALA 20 milligram (mg) LY2409021 dose, reference form administered orally in the fasted state
Cohort 1 - LY2409021 medium test form fedEXPERIMENTALSingle 20 mg LY2409021 test form with medium particle size administered orally immediately after ingestion of a standardized high-fat meal
Cohort 1 - LY2409021 medium test form fastedEXPERIMENTALSingle 20 mg LY2409021 test form with medium particle size administered orally in the fasted state
Cohort 2 - LY2409021 low test form fastedEXPERIMENTALSingle 20 mg LY2409021 test form with low particle size administered orally in the fasted state
Cohort 2 - LY2409021 medium test form fastedEXPERIMENTALSingle 20 mg LY2409021 test form with medium particle size administered orally in the fasted state
Cohort 2 - LY2409021 high test form fastedEXPERIMENTALSingle 20 mg LY2409021 test form with high particle size administered orally in the fasted state

Interventions

NameTypeDescription
LY2409021 Reference FormDRUGAdministered orally
LY2409021 Test-Med Formulation (medium particle size)DRUGAdministered orally
LY2409021 Test-High Formulation (high particle size)DRUGAdministered orally
LY2409021 Test-Low Formulation (low particle size)DRUGAdministered orally
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Eligibility Criteria

Age Range21 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Must be healthy male or a healthy female who cannot become pregnant * Must have body mass index (BMI) of 18.5 to 32 kilograms per meter squared (kg/m²), inclusive * Blood pressure as well as blood and urine laboratory test results must be acceptable for the study * The veins m...

Countries:Singapore
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Frequently asked questions about LY2409021 Reference Form

What is LY2409021 used for?

LY2409021 is an investigational small molecule being studied in healthy volunteers. It is not approved for any disease and remains in clinical development. The only completed trial evaluated its formulations and the effect of food in healthy participants.

Who makes LY2409021?

LY2409021 is being developed by Eli Lilly and Company, traded on the New York Stock Exchange under the ticker LLY. The company sponsored a Phase 1 study of the drug in healthy volunteers.

What phase is LY2409021 in?

LY2409021 is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and no trials are currently active.

What clinical trials is LY2409021 in?

LY2409021 has one completed clinical trial, NCT01354496, titled "A Study of LY2409021 Formulations and the Effect of Food." This Phase 1 study enrolled 35 healthy volunteers in Singapore and was a controlled, randomized trial.

Is LY2409021 FDA approved?

LY2409021 is not FDA approved. It is an investigational small molecule that has only been studied in a Phase 1 clinical trial involving healthy volunteers. The drug remains in clinical development and has not been authorized for any medical use.