Recent Updates
Recently added Catalysts

Insulin Lispro

Phase 3

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Eli Lilly and Company|Last Updated: Sep 8, 2025

Target and mechanism

ModalitySmall molecule

Also known as Insulin lispro (Humalog), Insulin Lispro (Humalog), Lispro, Insulin Lispro (U100), Lispro SC, Lispro Prandial Insulin

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment122

FDA Designations

No designations recorded

Clinical trial landscape

Insulin Lispro · 5 trials · 4 indications

Phase 3 1Phase 1 4
NCT01474538Safety and Efficacy Study of Insulin Lispro Versus Insulin Aspart in Participants With Type 2 Diabetes on Insulin Pump TherapyType 2 Diabetes Mellitus
COMPLETED122 Analytics
PHASE3COMPLETED
Safety and Efficacy Study of Insulin Lispro Versus Insulin Aspart in Participants With Type 2 Diabetes on Insulin Pump Therapy
Type 2 Diabetes MellitusUnlock trial analytics

Study Endpoints

Primary Endpoints

Glycosylated Hemoglobin A1C (HbA1c) at Endpoint
After 16 weeks of each treatment (Periods1 and 2)

Hemoglobin A1c (HbA1c) is a form of hemoglobin which is measured primarily to identify the average plasma glucose concentration over the last 8-12 weeks. Least Squares (LS) means were adjusted for treatment, period, sequence, thiazolidinedione use (Yes/No), baseline HbA1c (\>8% or ≤8%) and participants.

Number of Participants Who Show a Decrease or Suspension of Basal Insulin Delivery in Response to Hypoglycemia Challenges
Up to 4 hours post challenge
Number of Participants Who Show an Increase of Basal Insulin Delivery in Response to the Hyperglycemia Challenge
Up to 4 hours post challenge
Number of Participants Who Show a Resumption of Auto Mode Following Restored Continuous Glucose Monitoring (CGM) Connectivity
Up to 4 hours post challenge
Part A and Part B: Pharmacokinetics (PK): Area Under The Concentration Curve Zero to Infinity (AUC[0-∞])
-30, 0 (Predose), 5, 10, 15, 20, 25, 30, 35, 40, 45, 50, 55, 60, 70, 90, 120, 150,180, 240, and 300 Minutes

Primary outcome measure is based on the PK area under the concentration curve from 0 to infinity with a measurable concentration.

Pharmacokinetic Parameter: Area Under the Serum Insulin Concentration Versus Time Curve From Zero to Time of Return to Baseline (AUC0-tlast)
Day 1, predose through 8 hours post dose in each period.
Pharmacokinetic Parameter: Maximum Serum Insulin Concentration (Cmax)
Day 1, predose through 8 hours post dose in each period
Pharmacokinetic Parameter: Area Under the Curve(AUC)
Zero to infinity [AUC(0-∞)]
Pharmacokinetics: Area under the concentration curve (AUC)
Baseline up to 8 hours post administration of study drug
Pharmacokinetics: Maximum concentration (Cmax)
Baseline up to 8 hours post administration of study drug
Pharmacokinetics: Time of maximum concentration (Tmax)
Baseline up to 8 hours post administration of study drug

Secondary Endpoints

Total Daily Insulin Dose
Week 16 of each treatment (Periods 1 and 2)
Rate of Hypoglycemic Events Per 30 Days
Baseline through 16 weeks of each treatment (Periods 1 and 2)
Change From Baseline in Weight
Baseline, Week 16 of treatment Periods 1 and 2
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Insulin Lispro, then Insulin AspartACTIVE_COMPARATORInsulin lispro \[100 units/milliliter (U/mL)\] administered by continuous subcutaneous insulin infusion (CSII) pump for 16 weeks in Treatment Period 1, followed by insulin aspart (100 U/mL) administered by CSII pump for 16 weeks in Treatment Period 2.
Insulin Aspart, then Insulin LisproACTIVE_COMPARATORInsulin aspart (100 U/mL) administered by CSII pump for 16 weeks in Treatment Period 1, followed by insulin lispro (100 U/mL) administered by CSII pump for 16 weeks in Treatment Period 2.
AID System Containing Insulin LisproEXPERIMENTALThe AID system is comprised of a continuous subcutaneous insulin infusion (CSII) pump component with a hybrid closed-loop control (HCLC) algorithm, and a continuous glucose monitor (CGM) component.
Part A: Lispro (A)EXPERIMENTALFormulation A: Single dose of lispro administered subcutaneously (SC) in one of five periods.
Part A: Lispro (B)EXPERIMENTALFormulation B: Single dose of lispro administered SC in one of five periods.
Part A: Lispro (C)EXPERIMENTALFormulation C: Single dose of lispro administered SC in one of five periods.
Part A: Lispro (D)EXPERIMENTALFormulation D: Single dose of lispro administered SC in one of five periods.
Part A: Lispro (Reference)EXPERIMENTALReference formulation: Single dose of lispro administered SC in one of five periods.
Part B: LisproEXPERIMENTALFormulation selected from Part A. Single dose of lispro administered SC in one of four periods.
Insulin Lispro AACTIVE_COMPARATORInsulin Lispro A 20 units (U) of strength 200 units per milliliter (U/mL) (U-200)administered subcutaneously (SC) once in two of four study periods.(Two doses of test \[T\]).
Insulin Lispro BEXPERIMENTALInsulin Lispro B 20 units (U) of strength 100 U/mL (U-100) administered SC once in two of four study periods.(Two doses of reference \[R\]).
Insulin LisproACTIVE_COMPARATOR15 international units (IU) insulin lispro administered once subcutaneously (SC) during 1 of 3 dosing periods. There is a minimum 7 day washout between dosing periods.
BC106 Insulin LisproEXPERIMENTAL15 up to 30 IU BC106 insulin lispro administered once SC during 2 of 3 dosing periods. There is a minimum 7 day washout between dosing periods.

Interventions

NameTypeDescription
Insulin LisproDRUGInsulin lispro (100 U/mL) administered by CSII pump
Insulin AspartDRUGInsulin aspart (100 U/mL) administered by CSII pump
AID SystemDEVICEAID system
LisproDRUGAdministered SC
BC106 insulin lisproDRUGAdministered SC
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 85 Years
SexALL
Healthy VolunteersNo
Study Sites12

Inclusion Criteria: * Have type 2 diabetes (per World Health Organization \[WHO\] Classification of Diabetes) * Have been treated with CSII therapy using a rapid-acting analog for the previous 6 months * Have a screening A1C less than or equal to 9.0% (no lower limit for A1C) * Have a body mass ind...

Countries:United StatesSingapore
Unlock Eligibility Criteria