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IC83/LY2603618

Phase 1

Cancer | Small molecule | Oncology |Eli Lilly and Company|Last Updated: Oct 19, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment31
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00415636Safety and Tolerability of IC83/LY2603618 Administered After Pemetrexed 500 mg/m2 Every 21 Days in Patients With CancerPHASE1 COMPLETED 31Jan 1, 2007Jul 1, 2010Oct 19, 20181 United States
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Study Endpoints
Primary Endpoints
Number of Participants With Adverse Events (AEs)
baseline up to 24 months

Summary tables of serious AEs (SAEs) and all other non-serious adverse events (AEs) are located in the Reported Adverse Event Module.

Secondary Endpoints
Pharmacokinetic (PK) Parameter: Maximum Observed Plasma Concentration (Cmax) of IC83/LY2603618
Day 1 and Day 9 of Cycle 1
Pharmacokinetic (PK) Parameter: Area Under the IC83/LY2603618 Plasma Concentration Versus Time Curve From Time Zero to Infinity (AUC[0-∞])
Day 1 and Day 9 of Cycle 1
Percentage of Participants With Best Overall Response
baseline up to 24 months
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
LY2603618 40 mg/m^2 (4.5-hour infusion)EXPERIMENTALLY2603618 40 milligrams per square meter (mg/m\^2) was administered over the duration of 4.5 hours (30-minute bolus followed by a 4-hour infusion). Dose modifications were not allowed.
LY2603618 40 mg/m^2 (1-hour infusion)EXPERIMENTALBased on pharmacokinetic (PK) data from Cohort 1 (LY2603618 40 mg/m\^2 \[4.5-hour infusion\]), the LY2603618 40 mg/m\^2 dose in Cohort 2 (LY2603618 40 mg/m\^2 \[1-hour infusion\]) was repeated, but the dose was administered over the duration of 1 hour. Dose modifications were not allowed.
LY2603618 70 mg/m^2EXPERIMENTALBeginning with Cohort 3 (LY2603618 70 mg/m\^2), dose modifications were allowed. LY2603618 70 mg/m\^2 was administered over the course of 1 hour.
LY2603618 105 mg/m^2EXPERIMENTALCohort 4: LY2603618 105 mg/m\^2 administered over the duration of 1 hour.
LY2603618 150 mg/m^2EXPERIMENTALCohort 5: LY2603618 150 mg/m\^2 administered over the duration of 1 hour.
LY2603618 195 mg/m^2EXPERIMENTALCohort 6: LY2603618 195 mg/m\^2 administered over the duration of 1 hour.
Interventions
NameTypeDescription
IC83/LY2603618DRUG40 mg/m\^2 Day 1 and Day 9 of Cycle 1, Day 2 of subsequent cycles, unlimited 21-day cycles. Dose finding study: dose is escalated after a minimum of 6 participants receive 40 mg/m\^2.
pemetrexedDRUGpemetrexed 500 mg/m\^2, intravenous (IV), Day 8 of Cycle 1, Day 1 of subsequent cycles, unlimited 21-day cycles
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Has at least one lesion that can be evaluated by Response Evaluation Criteria In Solid Tumors (RECIST) * Has fully recovered from all toxicities due to the following: 1. Local radiation therapy that ended at least 14 days prior to Cycle 1, Day 1. 2. Surgery. * Has a life ...

Countries:United States
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