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Human regular U-500 insulin

Phase 3

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Eli Lilly and Company|Last Updated: May 20, 2020

Target and mechanism

ModalitySmall molecule

Also known as Human regular U-500 insulin (CSII)

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLEDDMC
Total Trials1
Total Enrollment420

FDA Designations

No designations recorded

Clinical trial landscape

Human regular U-500 insulin · 1 trial · 1 indication

Phase 3 1
NCT02561078An Administration Method Study of Human Regular U-500 Insulin (LY041001) in Participants With Type 2 Diabetes MellitusType 2 Diabetes Mellitus
COMPLETED420 Analytics
PHASE3COMPLETED
An Administration Method Study of Human Regular U-500 Insulin (LY041001) in Participants With Type 2 Diabetes Mellitus
Type 2 Diabetes MellitusUnlock trial analytics

Study Endpoints

Primary Endpoints

Change From Baseline in Hemoglobin A1c (HbA1c)
Baseline, 26 Weeks

HbA1c is the glycosylated fraction of hemoglobin A. HbA1c is measured primarily to identify average plasma glucose concentration over prolonged periods of time. Least Squares (LS) mean was determined by mixed-model repeated measures (MMRM) model with baseline of response, glucagon-like peptide-1 (GLP-1) or sodium-glucose cotransporter 2 (SGLT2) use, U-500R at entry, treatment, time and treatment by time interaction.

Secondary Endpoints

Change From Baseline in Fasting Plasma Glucose (FPG)
Baseline, 26 Weeks
Percentage of Participants With HbA1c <7.0%
26 Weeks
Percentage of Participants With HbA1c <7.5%
26 Weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Human regular U-500 insulin administered by CSIIEXPERIMENTALHuman regular U-500 insulin administered by CSII and titrated based on blood glucose readings for 26 weeks with a 2-week MDI lead-in.
Human regular U-500 insulin administered by MDIACTIVE_COMPARATORHuman regular U-500 insulin administered subcutaneously (SC) by MDI three times a day and titrated based on blood glucose readings for 26 weeks.

Interventions

NameTypeDescription
Human regular U-500 insulin (CSII)DRUGAdministered SC
Human regular U-500 insulin (MDI)DRUGAdministered SC
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Eligibility Criteria

Age Range18 Years to 85 Years
SexALL
Healthy VolunteersNo
Study Sites57

Inclusion Criteria: * Diagnosed with type 2 diabetes mellitus (T2DM). * Current TDD \>200 but ≤600 units of non U-500R insulin (MDI or CSII) and/or U-500R by MDI with syringe and vial for ≥3 months at entry. * If TDD of U-500R and other insulins are combined, then insulin other than U-500R not t...

Countries:United StatesPuerto Rico
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