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GRPR PET/CT

Phase 1

Malignancies Multiple | Unknown | Oncology |Eli Lilly and Company|Last Updated: Sep 18, 2026

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment60

FDA Designations

No designations recorded

Clinical trial landscape

GRPR PET/CT · 1 trial · 1 indication

Early Phase 1 1
NCT07828678PET/CT Imaging of GRPR Expression in Various TumorsMalignancies Multiple
NOT YET_RECRUITING60 Analytics
EARLY_PHASE1NOT YET_RECRUITING
PET/CT Imaging of GRPR Expression in Various Tumors
Malignancies MultipleUnlock trial analytics

Study Endpoints

Primary Endpoints

Per-Patient GRPR PET/CT Detection Rate
After the PET/CT imaging is completed

Proportion of participants with at least one GRPR-positive lesion on \[⁶⁸Ga\]-LY4257529 PET/CT. Detection rate will be calculated as the number of participants with at least one GRPR-positive lesion divided by the total number of participants in the relevant cancer cohort.

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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeDIAGNOSTIC

Treatment Arms

ArmTypeDescription
[⁶⁸Ga]-GRPR PET/CTEXPERIMENTALParticipants with breast cancer or other selected GRPR-expressing malignancies will receive a single intravenous administration of approximately 170 MBq ±20% of \[⁶⁸Ga\]-LY4257529, followed by PET/CT imaging approximately 50-70 minutes after injection. All participants undergo the same imaging intervention.

Interventions

NameTypeDescription
GRPR PET/CTDIAGNOSTIC_TEST\[⁶⁸Ga\]-LY4257529 is an investigational gastrin-releasing peptide receptor (GRPR)-targeted PET radiopharmaceutical. Participants will receive approximately 170 MBq ±20% (4.6 mCi ±20%) intravenously. PET/CT imaging will begin approximately 50-70 minutes after administration to evaluate GRPR-targeted tumor uptake and distribution.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo

Inclusion Criteria: Age 18 years or older Able to understand and provide written informed consent Diagnosis of a breast cancer or other tumor known or suspected to express GRPR, including: ER-positive/HER2-negative breast cancer Invasive lobular breast cancer Head and neck squamous cell carcinoma...

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Recent Changes (Last 90 Days)

LOWSep 19, 2026NCT07828678NEW_TRIAL: changed
LOWSep 19, 2026NCT07828678NEW_TRIAL: changed
LOWSep 19, 2026NCT07828678NEW_TRIAL: changed