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Enzastaurin 500 milligram Once Daily

Phase 2

Glioblastoma Multiforme | Small molecule | Oncology |Eli Lilly and Company|Last Updated: Apr 5, 2019

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment60
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00509821Enzastaurin Before and Concomitant With Radiation, Followed by Enzastaurin in Participants With Newly Diagnosed GlioblastomaPHASE2 COMPLETED 60Oct 1, 2007Mar 1, 2016Apr 5, 201910 Germany
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Study Endpoints
Primary Endpoints
Percentage of Participants With Progression Free Survival at 6 Months (PFS-6)
Baseline to 6 months

PFS-6 is defined as the percentage of participants with PFS at 6 months from the date of diagnosis to the first date of objectively determined progressive disease (based on radiological assessment) or death from any cause. It is assumed that PFS follows an exponential distribution.Estimation using Kaplan-Meier technique.

Secondary Endpoints
Percentage of Participants With Overall Survival at 1 and 2 Years After Surgery
Baseline to 1 and 2 year
Response Rate
Baseline to 30 months
Change in Neurologic Status as Measured by Mini Mental Status Questionnaire, Total Score
Baseline through Week 12 .
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Enzastaurin Once Daily (QD)EXPERIMENTALEnzastaurin given orally (PO) once daily (QD). 1125 mg loading dose D(-)7 then 500 mg PO,QD with concomitant radiotherapy.
Enzastaurin Twice Daily (BID)EXPERIMENTALEnzastaurin 1125 mg loading dose D(-)7 then 250 mg twice daily (BID) PO, with concomitant radiotherapy.
Interventions
NameTypeDescription
Enzastaurin 500 milligram (mg) Once Daily (QD)DRUG1125 mg loading dose D(-)7 then 500 mg QD, oral, daily until disease progression, given with and without radiotherapy treatment.
Enzastaurin 250 mg Twice Daily (BID)DRUG1125 mg loading dose D(-)7 then 250 mg BID, oral, daily until disease progression, given with and without radiotherapy treatment.
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites10

Inclusion Criteria: * Present with newly diagnosed histologically proven supratentorial GBM. * Demonstration of an unmethylated MGMT-promotor * Participants must sign an informed consent document. Participants must be at least 18 years of age. * Estimated life expectancy of at least 12 weeks * Tumo...

Countries:Germany
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