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tapentadol two 100-mg TRF

Phase 1

Healthy Volunteer | Small molecule | Other |Johnson & Johnson|Last Updated: Jan 31, 2014

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment52
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01309425A Study to Compare the Dose-proportionality of Tapentadol (CG5503) in Healthy Japanese and Korean Male VolunteersPHASE1 COMPLETED 52Feb 1, 2011May 1, 2011Jan 31, 2014 -
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Study Endpoints
Primary Endpoints
Pharmacokinetic profile, as measured by Cmax, AUC, tmax, kel, t1/2
Two days
Secondary Endpoints
Number of participants with adverse events
Time of screening to end of treatment (up to 9.5 weeks)
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
Treatment Arms
ArmTypeDescription
001EXPERIMENTALtapentadol (CG5503) ER 25-mg TRF 25mg TRF single oral dose
002EXPERIMENTALtapentadol (CG5503) ER 50-mg TRF 50mg TRF single oral dose
003EXPERIMENTALtapentadol (CG5503) ER 100-mg TRF 100mg TRF single oral dose
004EXPERIMENTALtapentadol (CG5503) ER two 100-mg TRF 200mg TRF single oral dose
Interventions
NameTypeDescription
tapentadol (CG5503) ER two 100-mg TRFDRUG200mg TRF single oral dose
tapentadol (CG5503) ER 50-mg TRFDRUG50mg TRF single oral dose
tapentadol (CG5503) ER 25-mg TRFDRUG25mg TRF single oral dose
tapentadol (CG5503) ER 100-mg TRFDRUG100mg TRF single oral dose
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Eligibility Criteria
Age Range20 Years — 45 Years
SexMALE
Healthy VolunteersYes

Inclusion Criteria: * Healthy Japanese and Korean male volunteers, inclusive * Body mass index (BMI) between 18.5 and 25 kg/m², inclusive, and a body weight of not less than 50 kg * Japanese volunteers must have resided outside of Japan for no more than 5 years, and their parents and maternal and p...

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