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TMC278, Long acting

Phase 1

Healthy | Small molecule | Other |Johnson & Johnson|Last Updated: Apr 7, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment4
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01656018A Study to Evaluate Safety, Acceptability, Pharmacokinetics, and ex Vivo Pharmacodynamics of TMC278 Long Acting Formulation in HIV-1 Seronegative ParticipantsPHASE1 COMPLETED 4Nov 1, 2012Jan 1, 2016Apr 7, 20161 United States
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Study Endpoints
Primary Endpoints
Number of participants with adverse events
Up to 280 days
Number of participants who would consider using long acting TMC278 for Human immunodeficiency virus (HIV) prevention in the future
Up to 280 days
Secondary Endpoints
TMC278 concentration in plasma
Up to 280 days
TMC278 concentration in endocervical fluid
Up to 280 days
TMC278 concentration in vaginal fluid
Up to 280 days
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Arm 1AEXPERIMENTALFemale participants will receive a single dose of long acting TMC278 1200 mg intramuscularly (IM) at baseline (Day 0) in Arm 1A.
Arm 1BEXPERIMENTALMale participants will receive a single dose of long acting TMC278 1200 mg IM at baseline in Arm 1B.
Arm 2AEXPERIMENTALFemale participants will receive a single dose of long acting TMC278 600 mg IM at baseline in Arm 2A.
Arm 2BEXPERIMENTALMale participants will receive a single dose of long acting TMC278 600 mg IM at baseline in Arm 2B.
Arm 3AEXPERIMENTALFemale participants will receive 3 bi-monthly injections of long acting TMC278 1200 mg IM at baseline, Months 2 and 4 in Arm 3A.
Arm 3BEXPERIMENTALMale participants will receive 3 bi-monthly injections of long acting TMC278 1200 mg IM at baseline, Months 2 and 4 in Arm 3B.
Arm 4AEXPERIMENTALFemale participants will receive a single dose of long acting TMC278 1200 mg IM at baseline followed by TMC278 900 mg at Months 2 and 4 in Arm 4A.
Arm 4BEXPERIMENTALMale participants will receive a single dose of long acting TMC278 1200 mg IM at baseline followed by TMC278 900 mg at Months 2 and 4 in Arm 4B.
Arm 5AEXPERIMENTALFemale participants will receive a single dose of long acting TMC278 1200 mg IM at baseline followed by TMC278 600 mg at Months 2 and 4 in Arm 5A.
Arm 5BEXPERIMENTALMale participants will receive a single dose of long acting TMC278 1200 mg IM at baseline followed by TMC278 600 mg at Months 2 and 4 in Arm 5B.
Interventions
NameTypeDescription
TMC278, Long acting (LA)DRUGTMC278 long acting will be administered IM to the participants as follows: a single dose of TMC278 600 mg will be administered at baseline in Arm 2A and Arm 2B; at Months 2 and 4 in Arm 5A and Arm 5B. A single dose of TMC278 900 mg will be administered at Months 2 and 4 in Arm 4A and Arm 4B. A single dose of TMC278 1200 mg will be administered at baseline in Arm 1A, Arm 1B; Arm 3A, Arm 3B, Arm 4A, Arm 4B, Arm 5A and Arm 5B; at Months 2 and 4 in Arm 3A and Arm 3B.
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Eligibility Criteria
Age Range18 Years — 45 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Human immunodeficiency virus type 1 (HIV-1) seronegative at screening and enrollment * Not pregnant or breastfeeding females * Agrees to protocol-defined method of contraception * Abstinence from insertion of anything in rectum (eg, medication, enema, penis, or sex toy) for 72...

Countries:United States
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