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Paliperidone, formulation

Phase 1

Psychotic Disorders | Small molecule | Psychiatry |Johnson & Johnson|Last Updated: Oct 29, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLED
Total Trials1
Total Enrollment305
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02087579Parallel Group, Multiple Dose Pharmacokinetics Study of Five Antipsychotic Medications in Psychiatric ParticipantsPHASE1 COMPLETED 305Feb 1, 2014Dec 1, 2014Oct 29, 201524 United States, Argentina +5
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Study Endpoints
Primary Endpoints
Aripiprazole concentration in venous and capillary plasma
14 time points over 3 days postdose

Venous blood samples will be collected at 8 scheduled time points after dosing and compared to fingerstick-based capillary blood samples collected at 6 scheduled time points after dosing.

Paliperidone concentration in venous and capillary plasma
14 time points over 3 days postdose
Olanzapine concentration in venous and capillary plasma
14 time points over 3 days postdose
Quetiapine concentration in venous and capillary plasma
14 time points over 3 days postdose
Risperidone concentration in venous and capillary plasma
14 time points over 3 days postdose
Secondary Endpoints
Number of participants with an adverse event as a measure of safety
Participants will be followed for the duration of hospital stay, an expected average of 3 days
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Cohort A: AripiprazoleEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort B: OlanzapineEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort C: PaliperidoneEXPERIMENTALAdministration of prolonged-release (extended-release) tablets or long-acting injectables (LAI) will continue at a participant's usual dose and dosing schedule.
Cohort D: QuetiapineEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort E: RisperidoneEXPERIMENTALAdministration of oral formulation or LAI will continue at a participant's usual dose and dosing schedule.
Interventions
NameTypeDescription
Aripiprazole, oral formulationDRUGAripiprazole tablets will be administered orally (by mouth), at no dose restriction, as per the locally approved label indications.
Olanzapine, oral formulationDRUGOlanzapine tablets will be administered orally, at no dose restriction as per the locally approved label indications.
Paliperidone, oral formulationDRUGPaliperidone prolonged-release/extended-release (XR) formulation tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Paliperidone, LAIDRUGPaliperidone long-acting injectable (LAI) i.e., paliperidone palmitate injections, will be administered per the locally approved label indications.
Quetiapine, oral formulationDRUGQuetiapine immediate-release (IR) formulation or extended-release (XR) formulation tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Risperidone, oral formulationDRUGRisperidone tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Risperidone, LAIDRUGRisperidone LAI injections will be administered will be administered per the locally approved label indications.
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites24

Inclusion Criteria: * Must be clinically stable as per the investigator's judgment (no suicidal behavior or current significant suicidal judgment based on C-SSRS rating scale) * No hospitalization for exacerbation of psychiatric symptoms during 3 months before screening * Receiving treatment with a...

Countries:United StatesArgentinaBelgiumBrazilBulgariaGermanySpain
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