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Paliperidone, formulation

Phase 1

Psychotic Disorders | Small molecule | Psychiatry |Johnson & Johnson|Last Updated: Oct 29, 2015

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment305

FDA Designations

No designations recorded

Clinical trial landscape

Paliperidone, formulation · 1 trial · 4 indications

Phase 1 1
NCT02087579Parallel Group, Multiple Dose Pharmacokinetics Study of Five Antipsychotic Medications in Psychiatric ParticipantsPsychotic Disorders
COMPLETED305 Analytics
PHASE1COMPLETED
Parallel Group, Multiple Dose Pharmacokinetics Study of Five Antipsychotic Medications in Psychiatric Participants
Psychotic DisordersUnlock trial analytics

Study Endpoints

Primary Endpoints

Aripiprazole concentration in venous and capillary plasma
14 time points over 3 days postdose

Venous blood samples will be collected at 8 scheduled time points after dosing and compared to fingerstick-based capillary blood samples collected at 6 scheduled time points after dosing.

Paliperidone concentration in venous and capillary plasma
14 time points over 3 days postdose
Olanzapine concentration in venous and capillary plasma
14 time points over 3 days postdose
Quetiapine concentration in venous and capillary plasma
14 time points over 3 days postdose
Risperidone concentration in venous and capillary plasma
14 time points over 3 days postdose

Secondary Endpoints

Number of participants with an adverse event as a measure of safety
Participants will be followed for the duration of hospital stay, an expected average of 3 days
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Cohort A: AripiprazoleEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort B: OlanzapineEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort C: PaliperidoneEXPERIMENTALAdministration of prolonged-release (extended-release) tablets or long-acting injectables (LAI) will continue at a participant's usual dose and dosing schedule.
Cohort D: QuetiapineEXPERIMENTALAdministration of oral formulation will continue at a participant's usual dose and dosing schedule.
Cohort E: RisperidoneEXPERIMENTALAdministration of oral formulation or LAI will continue at a participant's usual dose and dosing schedule.

Interventions

NameTypeDescription
Aripiprazole, oral formulationDRUGAripiprazole tablets will be administered orally (by mouth), at no dose restriction, as per the locally approved label indications.
Olanzapine, oral formulationDRUGOlanzapine tablets will be administered orally, at no dose restriction as per the locally approved label indications.
Paliperidone, oral formulationDRUGPaliperidone prolonged-release/extended-release (XR) formulation tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Paliperidone, LAIDRUGPaliperidone long-acting injectable (LAI) i.e., paliperidone palmitate injections, will be administered per the locally approved label indications.
Quetiapine, oral formulationDRUGQuetiapine immediate-release (IR) formulation or extended-release (XR) formulation tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Risperidone, oral formulationDRUGRisperidone tablets will be administered orally, at no dose restriction, as per the locally approved label indications.
Risperidone, LAIDRUGRisperidone LAI injections will be administered will be administered per the locally approved label indications.
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Eligibility Criteria

Age Range18 Years to 70 Years
SexALL
Healthy VolunteersNo
Study Sites24

Inclusion Criteria: * Must be clinically stable as per the investigator's judgment (no suicidal behavior or current significant suicidal judgment based on C-SSRS rating scale) * No hospitalization for exacerbation of psychiatric symptoms during 3 months before screening * Receiving treatment with a...

Countries:United StatesArgentinaBelgiumBrazilBulgariaGermanySpain
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Frequently asked questions about Paliperidone, formulation

What is Paliperidone used for?

Paliperidone is an investigational small molecule being developed by Johnson & Johnson (JNJ) for psychiatric conditions including schizoaffective disorder, affective psychosis, bipolar disorder, and schizophrenia. It is currently in Phase 3 clinical development, though all 27 listed trials have been completed.

Who makes Paliperidone?

Paliperidone is developed by Johnson & Johnson, traded as JNJ on the stock exchange. The company is conducting clinical research on this small molecule for psychiatric indications such as schizophrenia and schizoaffective disorder.

What phase is Paliperidone in?

Paliperidone is in Phase 3 clinical development. It remains investigational and has not been reported as FDA approved. All 27 clinical trials associated with the drug are completed, with no active trials currently listed.

What clinical trials is Paliperidone in?

Paliperidone has completed trials including NCT00791622 (QT interval study in schizophrenia and schizoaffective disorder), NCT00796640 (pharmacokinetics in schizophrenia), NCT01060228 (drug interaction with valproic acid), and NCT02634463 (immunoassay development). These trials enrolled a total of 7,564 participants.

Is Paliperidone the same as Risperidone?

Paliperidone is not the same as risperidone, but it is related. One completed trial (NCT02634463) collected samples from participants taking either aripiprazole, olanzapine, paliperidone, or risperidone to develop antipsychotic immunoassays, indicating they are distinct compounds studied together.