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Oromucosal Nicotine

Phase 1

Healthy | Small molecule | Other |Johnson & Johnson|Last Updated: Feb 3, 2025

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment24

FDA Designations

No designations recorded

Clinical trial landscape

Oromucosal Nicotine · 1 trial · 1 indication

Phase 1 1
NCT03398876A Study to Assess the Nicotine Pharmacokinetics, Tolerability and Safety With a New Oral Nicotine Replacement Product in Healthy Japanese SmokersHealthy
COMPLETED24 Analytics
PHASE1COMPLETED
A Study to Assess the Nicotine Pharmacokinetics, Tolerability and Safety With a New Oral Nicotine Replacement Product in Healthy Japanese Smokers
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Part 1: Maximum Baseline Corrected Plasma Nicotine Concentration (cCmax)
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 minute (min) and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose

cCmax is defined as the maximum baseline corrected plasma nicotine concentration (cCmax).

Part 1: Baseline Corrected Area Under the Plasma Nicotine Concentration versus (vs) Time Curve Until the Last Measurable Time Point (cAUCt)
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 min and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose

cAUCt is defined as the baseline corrected area under the plasma nicotine concentration-vs time curve until the last measurable time point.

Part 1: Baseline Corrected Area Under the Plasma Nicotine Concentration-vs Time Curve Extrapolated to Infinite (cAUC[infinity])
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 min and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose

cAUC(infinity) is defined as the baseline corrected area under the plasma nicotine concentration-vs time curve extrapolated to infinite.

Part 1: Baseline Corrected Area Under the Plasma Nicotine Concentration-vs Time Curve until the Last Measurable Time Point (cAUCt)
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 min and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose

cAUCt is defined as baseline corrected area under the plasma nicotine concentration-vs time curve until the last measurable time point.

Part 2: Average Plasma Nicotine Concentration During the Last Dosing Interval/Intervals (Cav)
Predose, 2, 4, 6, 8, 10, 15, 20, 30 post last dose (last dose: Hour 11.5 for Treatment E and Hour 11 for Treatment F); 45 and 60 min post last dose for Treatment F

Cav is defined as the average plasma nicotine concentration during the last dosing interval/intervals.

Part 2: Area Under the Plasma Nicotine Concentration-vs Time Curve During the Last Dosing Interval/Intervals (AUCtau)
Predose, 2, 4, 6, 8, 10, 15, 20, 30 post last dose (last dose: Hour 11.5 for Treatment E and Hour 11 for Treatment F); 45 and 60 min post last dose for Treatment F

AUCtau is defined as the area under the plasma nicotine concentration-vs time curve during the last dosing interval/intervals.

Part 2: Maximum Plasma Nicotine Concentration During the Last Dosing Interval/Intervals (Cmax)
Predose, 2, 4, 6, 8, 10, 15, 20, 30 post last dose (last dose: Hour 11.5 for Treatment E and Hour 11 for Treatment F); 45 and 60 min post last dose for Treatment F

Cmax is defined as maximum observed plasma nicotine concentration.

Secondary Endpoints

Part 1: Area Under the Plasma Nicotine Concentration-vs Time Curve until 10 Minutes after Start of Administration [AUC10min],
Predose; 2, 4, 6, 8, 10 min postdose
Part 1: Time to Reach Maximum Observed Plasma Concentration (Tmax)
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 min and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose
Part 1: Terminal Half-Life [t1/2]
Predose; 2, 4, 6, 8, 10, 15, 20, 30, 45 and 60 min and 1.5, 2, 3, 4, 6, 8, 10, 12 hours postdose
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Part 1; Treatment Sequence ABDCEXPERIMENTALParticipants will receive Treatment A (one spray of oromucosal nicotine spray \[ONS\]) at Visit 1, then Treatment B (2 consecutive sprays of ONS at Visit 2, then Treatment D (1 cigarette \[10 puffs\]) at Visit 3, followed by Treatment C (nicotine gum) at Visit 4. The visits will be separated by a period of at least 7 calendar days.
Part 1; Treatment Sequence BCADEXPERIMENTALParticipants will receive Treatment B at Visit 1, then Treatment C at Visit 2, then Treatment A at Visit 3 followed by Treatment D at Visit 4. The visits will be separated by a period of at least 7 calendar days.
Part 1; Treatment Sequence CDBAEXPERIMENTALParticipants will receive Treatment C at Visit 1, then Treatment D at Visit 2, then Treatment B at Visit 3 followed by Treatment A at Visit 4. The visits will be separated by a period of at least 7 calendar days. The visits will be separated by a period of at least 7 calendar days.
Part 1; Treatment Sequence DACBEXPERIMENTALParticipants will receive Treatment D at Visit 1, then Treatment A at Visit 2, then Treatment C at Visit 3 followed by Treatment B at Visit 4. The visits will be separated by a period of at least 7 calendar days.
Part 2; Treatment Sequence EFEXPERIMENTALParticipants who complete Part 1 will be selected for Part 2 based on the results of genetic polymorphism test and other examinations. Selected participants will receive Treatment E (two consecutive sprays of ONS once every 30 minutes until 11.5 hours) at Visit 5, followed by Treatment F (two consecutive sprays of ONS once every 1 hour until 11 hours) at Visit 6. The visits will be separated by a period of at least 7 calendar days.
Part 2; Treatment Sequence FEEXPERIMENTALParticipants who complete Part 1 will be selected for Part 2 based on the results of genetic polymorphism test and other examinations. Selected participants will receive Treatment F at Visit 5 followed by Treatment E at Visit 6. The visits will be separated by a period of at least 7 calendar days.

Interventions

NameTypeDescription
Oromucosal Nicotine Spray (ONS)DRUGParticipants will receive oral dose of oromucosal nicotine spray (ONS).
Nicotine GumDRUGParticipants will chew nicotine gum for 30 minutes.
CigaretteOTHERParticipants will smoke one cigarette as 10 puffs for 3 minutes.
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Eligibility Criteria

Age Range20 Years to 50 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male or female Japanese participants between the ages of 20 and 50 years, inclusive. Health is defined as the absence of clinically relevant abnormalities identified by a detailed medical history, blood pressure, pulse rate measurements, 12-lead electrocardiogram (ECG)...

Countries:Japan
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Frequently asked questions about Oromucosal Nicotine

What is Oromucosal Nicotine used for?

Oromucosal Nicotine is an investigational small molecule being studied as a nicotine replacement product. It is intended for use in healthy smokers, with a completed Phase 1 trial assessing its pharmacokinetics, tolerability, and safety in healthy Japanese smokers.

Who makes Oromucosal Nicotine?

Oromucosal Nicotine is being developed by Johnson & Johnson, traded on the New York Stock Exchange under the ticker JNJ. The company conducted a Phase 1 clinical trial of the product in Japan.

What phase is Oromucosal Nicotine in?

Oromucosal Nicotine is in Phase 1 clinical development. It is investigational and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and no active trials are currently listed.

What clinical trials is Oromucosal Nicotine in?

Oromucosal Nicotine has one completed clinical trial, NCT03398876, titled 'A Study to Assess the Nicotine Pharmacokinetics, Tolerability and Safety With a New Oral Nicotine Replacement Product in Healthy Japanese Smokers.' This Phase 1 study enrolled 24 healthy participants in Japan.

Is Oromucosal Nicotine the same as nicotine replacement therapy?

Oromucosal Nicotine is a nicotine replacement product, but it is not the same as other marketed nicotine replacement therapies. It is a new oral formulation under investigation, and its specific composition and delivery method are distinct from existing products.