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JNJ-64991524

Phase 1

Healthy | Small molecule | Other |Johnson & Johnson|Last Updated: Jan 24, 2019

Target and mechanism

ModalitySmall molecule

Also known as JNJ-64991524 Dose Level 1

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLEDDMC
Total Trials1
Total Enrollment86

FDA Designations

No designations recorded

Clinical trial landscape

JNJ-64991524 · 1 trial · 1 indication

Phase 1 1
NCT03346122A Study to Investigate the Safety, Tolerability and Pharmacokinetics of JNJ-64991524 in Healthy ParticipantsHealthy
COMPLETED86 Analytics
PHASE1COMPLETED
A Study to Investigate the Safety, Tolerability and Pharmacokinetics of JNJ-64991524 in Healthy Participants
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Study Endpoints

Primary Endpoints

Part 1: Single Ascending Dose (SAD): Number of Participants with Treatment Emergent Adverse Events (AEs) as a Measure of Safety and Tolerability
Up to Day 20

An adverse event is any untoward medical event that occurs in a participant administered an investigational product, and it does not necessarily indicate only events with clear causal relationship with the relevant investigational product. Treatment-emergent were events between administration of study drug and up to Day 20 that were absent before treatment or that worsened relative to pre-treatment state.

Part 2: Multiple Ascending Dose (MAD): Number of Participants with Treatment Emergent Adverse Events as a Measure of Safety and Tolerability
Up to Day 28

An adverse event is any untoward medical event that occurs in a participant administered an investigational product, and it does not necessarily indicate only events with clear causal relationship with the relevant investigational product. Treatment-emergent were events between administration of study drug and up to Day 28 that were absent before treatment or that worsened relative to pre-treatment state.

Number of Participants with Abnormalities in Vital Signs, Physical Examinations, Electrocardiogram (ECG), Cardiac Telemetry and Clinically Significant Laboratory Findings
Pre-dose, up to Day 20 (SAD) and up to Day 28 (MAD)

Number of participants with abnormalities in vital signs, physical examinations, ECG, cardiac telemetry and clinically significant laboratory findings will be measured.

Secondary Endpoints

Plasma Concentration of JNJ-64991524
Pre-dose, up to Day 20 (SAD) and up to Day 28 (MAD)
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeOTHER

Treatment Arms

ArmTypeDescription
Cohort 1:JNJ-64991524 Dose Level (DL) 1 or Placebo(SAD Part 1)EXPERIMENTALParticipants will receive a single oral dose (Dose level 1) of either JNJ-64991524 or placebo capsules after an overnight fast (at least 10 hours) on Day 1 of Part 1.
Cohort 2: JNJ-64991524 DL 2 or Placebo (SAD Part 1)EXPERIMENTALParticipants will receive a single oral dose (Dose level 2) of either JNJ-64991524 or placebo capsules after an overnight fast (at least 10 hours) on Day 1 of Part 1.
Cohort 3: JNJ-64991524 DL 3 or Placebo (SAD Part 1)EXPERIMENTALParticipants will receive a single oral dose (Dose level 3) of either JNJ-64991524 or placebo capsules after an overnight fast (at least 10 hours) on Day 1 of Part 1.
Cohort 4:JNJ-64991524 DL 4 or Placebo (SAD Part 1:Fasted-Fed)EXPERIMENTALParticipants will receive a single oral dose (Dose level 4) of either JNJ-64991524 or placebo capsules in a fasted condition on Day 1 and fed condition, on Day 7.
Cohort 5: JNJ-64991524 DL 5 or Placebo (SAD Part 1)EXPERIMENTALParticipants will receive a single oral dose (Dose level 5) of JNJ-64991524 or placebo after an overnight fast (at least 10 hours) on Day 1 of Part 1.
Cohort 6: JNJ-64991524 DL 6 or Placebo (SAD Part 1)EXPERIMENTALParticipants will receive a single oral dose (Dose level 6) of JNJ-64991524 or placebo after an overnight fast (at least 10 hours) on Day 1 of Part 1.
Cohort 1: JNJ-64991524 DL 7 or Placebo (MAD Part 2)EXPERIMENTALParticipants will receive an oral dose (Dose level 7) JNJ-64991524 or placebo capsules once daily for 14 days in fasted or fed condition in Part 2. Fasted/fed condition will be determined based on tolerability and pharmacokinetics (PK) from Part 1.
Cohort 2: JNJ-64991524 DL 8 or Placebo (MAD Part 2)EXPERIMENTALParticipants will receive an oral dose (Dose level 8) JNJ-64991524 or placebo capsules once daily for 14 days in fasted or fed condition in Part 2. Fasted/fed condition will be determined based on tolerability and PK from Part 1.
Cohort 3: JNJ-64991524 DL 9 or Placebo (MAD Part 2)EXPERIMENTALParticipants will receive an oral dose (Dose level 9) JNJ-64991524 or placebo capsules once daily for 14 days in fasted or fed condition in Part 2. Fasted/fed condition will be determined based on tolerability and PK from Part 1.
Cohort 4: JNJ-64991524 DL 6 or Placebo (MAD Part 2)EXPERIMENTALParticipants will receive an oral dose (Dose level 6) of JNJ-64991524 or placebo capsules once daily for 14 days in fasted or fed condition in Part 2. Fasted/fed condition will be determined by tolerability and PK from Part 1.

Interventions

NameTypeDescription
JNJ-64991524 Dose Level 1DRUGParticipants will receive JNJ-64991524 at a Dose Level 1 in SAD Part 1 of study.
JNJ-64991524 Dose Level 2DRUGParticipants will receive JNJ-64991524 at a Dose Level 2 in SAD Part 1 of study.
JNJ-64991524 Dose Level 3DRUGParticipants will receive JNJ-64991524 at a Dose Level 3 in SAD Part 1 of study.
JNJ-64991524 Dose Level 4DRUGParticipants will receive JNJ-64991524 at a Dose Level 4 in SAD Part 1 of study.
JNJ-64991524 Dose Level 5DRUGParticipants will receive JNJ-64991524 at a dose of Dose Level 5 in SAD Part 1 of study.
JNJ-64991524 Dose Level 6DRUGParticipants will receive JNJ-64991524 at a Dose Level 6 in SAD Part 1 and MAD part 2 of study.
PlaceboDRUGParticipants will receive matching placebo in all cohorts on Day 1 in Part 1 and Part 2 of the study.
JNJ-64991524 Dose Level 7DRUGParticipants will receive JNJ-64991524 at a dose of Dose Level 7 in MAD Part 2 of study for 14 days.
JNJ-64991524 Dose Level 8DRUGParticipants will receive JNJ-64991524 at a Dose Level 8 in MAD Part 2 of study for 14 days.
JNJ-64991524 Dose Level 9DRUGParticipants will receive JNJ-64991524 at a Dose Level 9 in MAD Part 2 of study for 14 days.
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Eligibility Criteria

Age Range18 Years to 60 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Weigh at least 50 kilogram (kg), and have a body mass index (BMI) of 18 kg/ meter (m)\^2 to 30 kg/m\^2, inclusive, at screening * Be otherwise healthy on the basis of physical examination, medical history, vital signs, and 12-lead ECG performed at screening and Day-1. This det...

Countries:Belgium
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