Recent Updates
Recently added Catalysts

JNJ-48816274

Phase 1

Healthy | Small molecule | Other |Johnson & Johnson|Last Updated: Apr 27, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials1
Total Enrollment90
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02852395A Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of JNJ-48816274PHASE1 COMPLETED 90Aug 13, 2016May 2, 2018Apr 27, 20252 United Kingdom
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Number of Participants with Treatment Emergent Adverse Events as a Measure of Safety and Tolerability
Up to 14 days after last dose in Part 1 (approximately 5.5 weeks)
Area Under the Plasma Concentration-Time Curve From Time Zero to Time 't' (AUC[0-t])
Days 1-2 in Part 1
Maximum Observed Plasma Concentration (Cmax)
Day 1 in Part 1
Time to Reach the Maximum Plasma Concentration (Tmax)
Day 1 in Part 1
Elimination Half Life (t1/2)
Days 1-2 in Part 1
Mean Karolinska Sleepiness Scale score
Day 1 in Part 1

A 1-item questionnaire completed by participants to rate their degree of sleepiness on a scale of 1 to 9, ranging from 'extremely alert' (1) to 'very sleepy, great effort to keep awake, fighting sleep' (9).

Secondary Endpoints
Mean Total Sleep Time by 8-hour overnight Polysomnography
Part 2: Days 1-2 of each of 3 or 4 crossover periods
Mean Latency to Persistent Sleep by 8-hour overnight Polysomnography
Part 2: Days 1-2 of each of 3 or 4 crossover periods
Mean Leeds Sleep Evaluation Questionnaire (LSEQ) Score
Part 2: Day 2 of each of 3 or 4 crossover periods
Unlock Study Endpoints
Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part 1 Single DoseEXPERIMENTALPart 1 single daytime oral dose of JNJ-48816274 or placebo. Doses of JNJ-48816274 will start at 5 milligram (mg) and increase sequentially to a maximum dose of 250 mg.
Part 2 Crossover Sleep StudyEXPERIMENTALPart 2 single nighttime oral dose of JNJ-48816274 or placebo administered during each of 3 or 4 crossover periods separated by 7-9 days. The doses of JNJ-48816274 will be selected based on data from Part 1 (not to exceed 250 mg).
Part 3 Repeated Dose (Optional)EXPERIMENTALPart 3 daytime oral dose of JNJ-48816274 or placebo administered once daily for 7 consecutive days. Doses will be determined based on data from Part 1, and may increase sequentially (not to exceed 250 mg/day).
Interventions
NameTypeDescription
JNJ-48816274DRUGOral dose; dose range of 5 mg up to 250 mg
PlaceboDRUGOral dose; appearance matched to JNJ-48816274
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Must be healthy as assessed by medical history and safety evaluations performed at screening * Has a body mass index between 18 and 30 kilogram per square meter (kg/m2) and body weight not less than 50 kg * Must be willing and able to abide by the prohibitions and restrictions...

Countries:United Kingdom
Unlock Eligibility Criteria