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GW842166X

Phase 1

Pain, Inflammatory | Small molecule | Pain |GSK plc|Last Updated: Aug 7, 2017

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment6

FDA Designations

No designations recorded

Clinical trial landscape

GW842166X · 1 trial · 1 indication

Phase 1 1
NCT00511524An Imaging Study to Investigate the Distribution of GW842166X in the Brain.Pain, Inflammatory
COMPLETED6 Analytics
PHASE1COMPLETED
An Imaging Study to Investigate the Distribution of GW842166X in the Brain.
Pain, InflammatoryUnlock trial analytics

Study Endpoints

Primary Endpoints

Rate at which the drug crosses from plasma to brain (ki)using images from the scan
throughout the study

Secondary Endpoints

Safety of drug
after taking the drug pre-dose, 2hr, 4hr, 6hr, 10hr, 24hr, follow-up.
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Subjects receiving GW842166EXPERIMENTALSubjects will receive single oral dose of 400 milligram (mg) un-labeled GW842166X. After 2-5 hours subjects will receive \[carbonyl-\^11C\]GW842166.

Interventions

NameTypeDescription
GW842166XDRUGGW842166X will available with dose strength of 100 mg capsules. Four 100mg GW842166X capsules will be used for the 400 mg oral dose of GW842166X.
[carbonyl-^11C]GW842166DRUG\[carbonyl-\^11C\]GW842166 will b available as Intravenous solution.
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Eligibility Criteria

Age Range50 Years to 80 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male aged 50 to 80yrs inclusive at the screening visit. * subjects with negative HIV and hepatitis B and C test results within 3 months of study start. Exclusion Criteria: * A negative Allens test on arm to be used for arterial cannulation. * Any contraindications to MRI sca...

Countries:Sweden
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Competitive Landscape -Inflammatory Disorders 8 trials (matched to "Pain, Inflammatory")

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Frequently asked questions about GW842166X

What is GW842166X used for?

GW842166X is an investigational small molecule being developed for pain and inflammatory conditions. It is a Phase 1 drug candidate that has been studied in a completed clinical trial. The drug is not approved and remains in clinical development.

Who makes GW842166X?

GW842166X is being developed by GSK plc, a pharmaceutical company listed on the stock exchange under the ticker GSK. The drug is currently in Phase 1 clinical development for pain and inflammatory indications.

What phase is GW842166X in?

GW842166X is in Phase 1 clinical development. It has completed one Phase 1 trial, which was an imaging study to investigate the distribution of the drug in the brain. The drug is investigational and not yet approved.

What clinical trials is GW842166X in?

GW842166X has one completed clinical trial, NCT00511524, titled "An Imaging Study to Investigate the Distribution of GW842166X in the Brain." This Phase 1 study enrolled 6 healthy male volunteers aged 50 years and older in Sweden.

Is GW842166X the same as any other drug?

GW842166X is the drug name used in clinical development. No alternative names have been reported for this investigational compound. It is being studied by GSK plc for pain and inflammatory conditions.