Recent Updates
Recently added Catalysts

GW842166X

Phase 1

Pain, Inflammatory | Small molecule | Pain |GSK plc|Last Updated: Aug 7, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
UNCONTROLLEDBiomarker
Total Trials1
Total Enrollment6
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00511524An Imaging Study to Investigate the Distribution of GW842166X in the Brain.PHASE1 COMPLETED 6Jun 26, 2007Jul 4, 2007Aug 7, 20171 Sweden
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Rate at which the drug crosses from plasma to brain (ki)using images from the scan
throughout the study
Secondary Endpoints
Safety of drug
after taking the drug pre-dose, 2hr, 4hr, 6hr, 10hr, 24hr, follow-up.
Unlock Study Endpoints
Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Subjects receiving GW842166EXPERIMENTALSubjects will receive single oral dose of 400 milligram (mg) un-labeled GW842166X. After 2-5 hours subjects will receive \[carbonyl-\^11C\]GW842166.
Interventions
NameTypeDescription
GW842166XDRUGGW842166X will available with dose strength of 100 mg capsules. Four 100mg GW842166X capsules will be used for the 400 mg oral dose of GW842166X.
[carbonyl-^11C]GW842166DRUG\[carbonyl-\^11C\]GW842166 will b available as Intravenous solution.
Unlock Study Design Details
Eligibility Criteria
Age Range50 Years — 80 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male aged 50 to 80yrs inclusive at the screening visit. * subjects with negative HIV and hepatitis B and C test results within 3 months of study start. Exclusion Criteria: * A negative Allens test on arm to be used for arterial cannulation. * Any contraindications to MRI sca...

Countries:Sweden
Unlock Eligibility Criteria
Competitive Landscape -Inflammatory Disorders 9 trials