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Nitazoxanide

Phase 1

Moderate Hepatic Impairment | Small molecule | Gastrointestinal |Genfit SA Sponsored ADR|Last Updated: Oct 28, 2022

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment25

FDA Designations

No designations recorded

Clinical trial landscape

Nitazoxanide · 2 trials · 6 indications

Phase 1 2
NCT05368935Nitazoxanide Pharmacokinetic Parameters in Renal Impaired SubjectsRenal Impairment
COMPLETED77 Analytics
NCT05116826Nitazoxanide Pharmacokinetic Parameters in Hepatic Impaired PatientsModerate Hepatic Impairment
COMPLETED25 Analytics
PHASE1COMPLETED
Nitazoxanide Pharmacokinetic Parameters in Renal Impaired Subjects
Renal ImpairmentUnlock trial analytics
PHASE1COMPLETED
Nitazoxanide Pharmacokinetic Parameters in Hepatic Impaired Patients
Moderate Hepatic ImpairmentUnlock trial analytics

Study Endpoints

Primary Endpoints

Maximum observed plasma concentration (Cmax)
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24 hours (Day 8); 48 hours (Day 9); 72 hours (Day 10) and 96 hours (Day 11) post-dose

Plasma pharmacokinetic (PK) parameters of NTZ active metabolite expressed in terms of unbound as well as total concentrations at steady-state in subjects with mild, moderate and severe renal impairment compared to healthy volunteers

Area under the plasma concentration time curve (AUC) from time zero to the time of the last quantifiable concentration (AUC0-t)
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24 (Day 8); 48 (Day 9); 72 (Day 10) and 96 (Day 11) hours post-dose

Plasma pharmacokinetic parameters of NTZ active metabolite expressed in terms of unbound as well as total concentrations at steady-state in subjects with mild, moderate and severe renal impairment compared to healthy volunteers

AUC from time zero to 12h (AUC0-12)
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24 hours (Day 8); 48 hours (Day 9); 72 hours (Day 10) and 96 hours (Day 11) post-dose

Plasma pharmacokinetic parameters of NTZ active metabolite expressed in terms of unbound as well as total concentrations at steady-state in subjects with mild, moderate and severe renal impairment compared to healthy volunteers

Area under the plasma concentration time curve (AUC) from time zero to 12h (AUC0-12)
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24; and 48 hours post dose

In participants with moderate and severe hepatic impairment compared to healthy volunteers

AUC from time zero to the time of the last quantifiable concentration (AUC0-t)
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24; and 48 hours post dose

In participants with moderate and severe hepatic impairment compared to healthy volunteers

Maximum observed plasma concentration (Cmax),
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18; 24; and 48 hours post dose

In participants with moderate and severe hepatic impairment compared to healthy volunteers

Secondary Endpoints

Time of the maximum observed plasma concentration (Tmax) for NTZ and its major active metabolite
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18 hours; 24 hours (Day 8); 48 hours (Day 9) ; 72 hours (Day 10) and 96 hours (Day 11) post-dose
Apparent plasma terminal elimination half-life (t1/2) for the NTZ and its major active metabolite
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18 hours; 24 hours (Day 8); 48 hours (Day 9) ; 72 hours (Day 10) and 96 hours (Day 11) post-dose
Unbound fraction in plasma defined as total concentration/unbound concentration (fu) for the NTZ and its major active metabolite
Day 1: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10 and 12 hours post dose; Day 2-6: pre-dose; Day 7: pre-dose; 1; 2; 3; 4; 5; 6; 7; 8; 10; 12; 14; 16; 18 hours; 24 hours (Day 8); 48 hours (Day 9) ; 72 hours (Day 10) and 96 hours (Day 11) post-dose
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Healthy Control Match (RF ≥ 90 mL/min)EXPERIMENTAL500 mg Twice Daily for 7 days
Mild Renal Impairment (RF ≥ 60 to < 90 mL/min)EXPERIMENTAL500 mg Twice Daily for 7 days
Moderate Renal Impairment (RF ≥ 30 to < 60 mL/min)EXPERIMENTAL500 mg Twice Daily for 7 days
Severe Renal Impairment (RF < 30 mL/min and not on dialysis)EXPERIMENTAL500 mg Twice Daily for 7 days
Healthy Control Match (Normal hepatic function)EXPERIMENTALNTZ 500 mg twice a day for 7 days
Moderate Child-Pugh B (Moderate hepatic impairment)EXPERIMENTALNTZ 500 mg twice a day for 7 days
Severe Child-Pugh C (Severe hepatic impairment)EXPERIMENTALNTZ 500 mg twice a day for 7 days

Interventions

NameTypeDescription
NitazoxanideDRUG500 mg Twice Daily for 7 days
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Eligibility Criteria

Age Range18 Years to 80 Years
SexALL
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: 1. Males or females, between 18 and 80 years of age, inclusive 2. With a minimum body weight of ≥ 50.0 kg for males and ≥ 45.0 kg for females and within a BMI range of 18.0 to 40.0 kg/m\^2, inclusive 3. Females participating in this study must be of non-childbearing potential or...

Countries:United States
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Frequently asked questions about Nitazoxanide

What is Nitazoxanide used for in Renal Impairment and Moderate Hepatic Impairment?

Nitazoxanide is being studied for use in patients with Renal Impairment and Moderate Hepatic Impairment. It is a small molecule being developed by Genfit SA for gastrointestinal conditions. The drug is currently in Phase 1 clinical development, with studies focused on understanding its pharmacokinetic parameters in these patient populations.

What does Nitazoxanide target?

Nitazoxanide is a small molecule therapeutic being developed for gastrointestinal conditions. The specific molecular target of Nitazoxanide is not disclosed in the available information. The ongoing Phase 1 studies are designed to evaluate its pharmacokinetic parameters in patients with renal and hepatic impairment.

Who makes Nitazoxanide?

Nitazoxanide is being developed by Genfit SA, which trades under the ticker GNFT. The company is conducting Phase 1 clinical trials to evaluate the drug's pharmacokinetics in patients with renal impairment and moderate hepatic impairment. Genfit is focused on developing this small molecule for gastrointestinal therapeutic applications.

What phase is Nitazoxanide in?

Nitazoxanide is in Phase 1 clinical development. It is an investigational drug being studied for use in patients with renal impairment and moderate hepatic impairment. The drug has completed one Phase 1 trial with 77 participants, and it is not yet approved by regulatory authorities.

What clinical trials is Nitazoxanide in?

Nitazoxanide has been studied in two completed Phase 1 clinical trials. NCT05116826 evaluated pharmacokinetic parameters in patients with moderate and severe hepatic impairment, enrolling 25 participants. NCT05368935 assessed pharmacokinetics in subjects with renal impairment, enrolling 77 participants. Both trials were conducted in the United States.

Is Nitazoxanide the same as any other drug?

Nitazoxanide is the primary name for this drug candidate being developed by Genfit SA. No alternative names for Nitazoxanide have been identified in the available information. The drug is being studied under its current name in clinical trials for renal and hepatic impairment indications.