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BMS-986141

Phase 2

Thrombosis | Small molecule | Cardiovascular |Bristol-Myers Squibb Company|Last Updated: Dec 14, 2018

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLEDDMC
Total Trials2
Total Enrollment164

FDA Designations

No designations recorded

Clinical trial landscape

BMS-986141 · 3 trials · 2 indications

Phase 2 1Phase 1 2
NCT02671461Safety and Efficacy Study of a Protease Activated Receptor-4 Antagonist Being Tested to Reduce the Chances of Having Additional Strokes or "Mini Strokes"Thrombosis
COMPLETED16 Analytics
PHASE2COMPLETED
Safety and Efficacy Study of a Protease Activated Receptor-4 Antagonist Being Tested to Reduce the Chances of Having Additional Strokes or "Mini Strokes"
ThrombosisUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Participants With Composite of Symptomatic Ischemic Stroke by Day 28 and Unrecognized Brain Infarction Assessed by MRI at Day 28
28 Days

The incidence of a composite of symptomatic ischemic stroke by Day 28 and unrecognized brain infarction assessed by MRI at Day 28 was to be reported by arm in all treated participants.

Percentage of Participants With Composite of Adjudicated Major Bleeding and Adjudicated Clinically Relevant Non-major (CRNM) Bleeding During the Treatment Period
Up to 90 days

The percentage of participants with composite of major bleeding and CRNM bleeding was to be reported. Point estimates and 95% CIs for event rates were to be presented by treatment, together with point estimates and 95% CIs for the difference of event rates between each BMS-986141 arm and placebo.

Maximum observed concentration (Cmax)
Days 1-21
Area under the concentration-time curve from time zero extrapolated to infinite time (AUC(INF))
Days 1-21
Area under the concentration-time curve from time zero to the time of the last quantifiable concentration (AUC (0-T))
Days 1-21
Safety measured by number of subjects who experience SAEs, deaths, AEs leading to discontinuation, and potential clinically significant changes in ECG parameters, vital signs, laboratory tests and physical examinations
Up to 30 days post discontinuation of dosing or last participation in the study

Serious adverse event (SAE) Adverse event (AE) Electrocardiogram (ECG)

Tolerability measured by number of subjects who experience SAEs, deaths, AEs leading to discontinuation, and potential clinically significant changes in ECG parameters, vital signs, laboratory tests and physical examinations
Up to 30 days post discontinuation of dosing or last participation in the study
Safety measured by percent of subjects who experience SAEs, deaths, AEs leading to discontinuation, and potential clinically significant changes in ECG parameters, vital signs, laboratory tests and physical examinations
Up to 30 days post discontinuation of dosing or last participation in the study
Tolerability measured by percent of subjects who experience SAEs, deaths, AEs leading to discontinuation, and potential clinically significant changes in ECG parameters, vital signs, laboratory tests and physical examinations
Up to 30 days post discontinuation of dosing or last participation in the study

Secondary Endpoints

Percentage of Participants With Major Adverse Cardiovascular Events (MACE)
90 days
Percentage of Participants With Adjudicated Symptomatic Recurrent Stroke (Including Fatal and Non-fatal)
Day 28
Percentage of Participants With Composite of Unrecognized Brain Infarction Assessed by MRI at Day 28 and MACE at Day 90
Day 90
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BMS-986141 0.8mgEXPERIMENTALBMS-986141 0.8mg orally (tablets) and Aspirin (ASA) 75 to 162 mg orally (tablets)
BMS-986141 4.8mgEXPERIMENTALBMS-986141 4.8mg orally (tablets) and ASA 75 to 162 mg orally (tablets)
PlaceboPLACEBO_COMPARATORPlacebo orally (tablets) and ASA 75 to 162 mg orally (tablets)
BMS-986141 and DilitazemEXPERIMENTAL -
Part A Panel 1: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 2: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 3: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 4: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 5: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 6: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo single dose by mouth as specified
Part A Panel 7: BMS-986141EXPERIMENTALSingle dose by mouth as specified
Part A Panel 8: BMS-986141EXPERIMENTALSingle dose by mouth as specified
Part B Panel 1: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part B Panel 2: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part B Panel 3: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part C Panel 1: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part C Panel 2: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part C Panel 3: BMS-986141 or PlaceboEXPERIMENTALBMS-986141 or Placebo by mouth as specified
Part D Panel 1: BMS-986141 and AspirinEXPERIMENTALBMS-986141 and Aspirin by mouth as specified
Part D Panel 1: Placebo matching BMS-986141 and AspirinPLACEBO_COMPARATORBMS-986141 placebo and Aspirin by mouth as specified
Part E Panel 1: BMS-986141 and ItraconazoleEXPERIMENTALBMS-986141 and Itraconazole by mouth as specified

Interventions

NameTypeDescription
BMS-986141DRUG -
AspirinDRUG -
PlaceboOTHER -
DilitazemDRUGSingle dose BMS-986141 and Multiple doses of Dilitazem
ItraconazoleDRUG -
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites33

For more information regarding BMS clinical trial participation, please visit www.BMSStudyConnect.com Inclusion Criteria: * Male or female, age 18 or older * Must have had a very recent stroke or transient ischemic attack ("mini stroke") that can be confirmed by the study doctor * Able to be assig...

Countries:United StatesJapan
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Frequently asked questions about BMS-986141

What is BMS 986141 used for?

BMS 986141 is an investigational small molecule being developed for cardiovascular conditions including atherothrombotic diseases, ischemic stroke, and thrombosis. It is currently in clinical development and has not been approved by the FDA. The drug is being studied to potentially reduce the chances of additional strokes or mini strokes.

What does BMS 986141 target?

BMS 986141 is a protease activated receptor-4 (PAR-4) antagonist, as indicated by the clinical trial title. It works by targeting this receptor, which is involved in platelet activation and thrombosis. By blocking PAR-4, the drug aims to reduce thrombotic events in conditions like ischemic stroke and atherothrombotic diseases.

Who makes BMS 986141?

BMS 986141 is being developed by Bristol-Myers Squibb Company, which trades under the ticker BMY on the stock exchange. The company is conducting clinical trials to evaluate the safety, tolerability, pharmacokinetics, and pharmacodynamics of this investigational drug in various patient populations.

What phase is BMS 986141 in?

BMS 986141 is in Phase 1 of clinical development, according to the overall phase designation. However, one completed trial (NCT02671461) was a Phase 2 study. The drug is investigational and not yet approved by regulatory authorities. All listed trials for BMS 986141 have been completed.

What clinical trials is BMS 986141 in?

BMS 986141 has been studied in four completed clinical trials. NCT02341638 was a Phase 1 single and multiple ascending dose study in healthy subjects. NCT02671461 was a Phase 2 safety and efficacy study in patients with thrombosis. NCT02922452 and NCT02957448 were Phase 1 drug interaction studies with diltiazem and rifampin, respectively.

Is BMS 986141 the same as BMS-986141?

Yes, BMS 986141 and BMS-986141 refer to the same drug. The hyphenated version is used in clinical trial titles, while the non-hyphenated form appears in other contexts. Both names identify the same investigational protease activated receptor-4 antagonist being developed by Bristol-Myers Squibb.