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ethinyl estradiol and levonorgestrel; exenatide

Phase 1

Type 2 Diabetes Mellitus | Small molecule | Metabolic |AstraZeneca PLC|Last Updated: Aug 18, 2015

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment38

FDA Designations

No designations recorded

Clinical trial landscape

ethinyl estradiol and levonorgestrel; exenatide · 1 trial · 1 indication

Phase 1 1
NCT00254800The Effects of Exenatide on Oral Contraceptive Pharmacokinetics in Healthy FemalesType 2 Diabetes Mellitus
COMPLETED38 Analytics
PHASE1COMPLETED
The Effects of Exenatide on Oral Contraceptive Pharmacokinetics in Healthy Females
Type 2 Diabetes MellitusUnlock trial analytics

Study Endpoints

Primary Endpoints

Assessment of Pharmacokinetics profile of exenatide measured by AUC and Cmax
Day 8 and Day 22 of each treatment period hours of sampling: Predose, 0.5, 1,1.5, 2, 2.5, 3, 3.5, 4, 4.5, 5, 6,8, 10, 12, 16, 24, 48

To evaluate the effect of exenatide on the multiple-dose pharmacokinetics of a combination oral contraceptive when administered one hour prior or 30 minutes after the exenatide dose.

Secondary Endpoints

Assessment of Pharmacokinetics profile of exenatide measured by AUC and Cmax
Day 8 and Day 22 of each treatment period hours of sampling: Predose, 0.5, 1,1.5, 2, 2.5, 3, 3.5, 4, 4.5, 5, 6,8, 10, 12, 16, 24, 48
Safety and Tolerability assessment by Adverse events, clinical laboratory evaluations, vital signs, ECG blood glucose, body weight, physical examination and exenatide antibodies.
Baseline through Day 84
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Sequence 1EXPERIMENTALOral contraceptive 1 hour prior to exenatide/oral contraceptive 30 minutes after exenatide/oral contraceptive alone
Sequence 2EXPERIMENTALOral contraceptive 30 minutes after exenatide/oral contraceptive alone/oral contraceptive 1 hour prior to exenatide
Sequence 3EXPERIMENTALOral contraceptive alone/oral contraceptive 1 hour prior to exenatide/oral contraceptive 30 minutes after exenatide

Interventions

NameTypeDescription
ethinyl estradiol and levonorgestrel; exenatideDRUGOral contraceptive is ethinyl estradiol (30 μg) and levonorgestrel (150 μg) one time daily, per 28-day treatment period; Study drug (exenatide 10 mcg) is subcutaneously injected twice daily
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Eligibility Criteria

Age Range18 Years to 45 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Pre-menopausal female of child-bearing potential. * Body Mass Index (BMI) between 19 and 35 kg/m\^2, inclusive. Exclusion Criteria: * On implanted contraceptives for 6 months, or injectable contraceptives for 12 months prior to the study. * Evidence of diabetes mellitus. * P...

Countries:United Kingdom
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Frequently asked questions about ethinyl estradiol and levonorgestrel; exenatide

What is ethinyl estradiol and levonorgestrel; exenatide used for?

Ethinyl estradiol and levonorgestrel; exenatide is being studied for use in Type 2 Diabetes Mellitus. It is a combination of an oral contraceptive (ethinyl estradiol and levonorgestrel) and exenatide, a medication for diabetes. The drug is in Phase 1 clinical development as a small molecule therapy.

What does ethinyl estradiol and levonorgestrel; exenatide target?

The specific molecular target of ethinyl estradiol and levonorgestrel; exenatide is not disclosed in available information. The drug combines an oral contraceptive with exenatide, which is known to affect glucose metabolism, but the precise target for this combination has not been specified.

Who makes ethinyl estradiol and levonorgestrel; exenatide?

AstraZeneca PLC (ticker: AZN) is developing ethinyl estradiol and levonorgestrel; exenatide. The company is conducting clinical research on this combination therapy for Type 2 Diabetes Mellitus.

What phase is ethinyl estradiol and levonorgestrel; exenatide in?

Ethinyl estradiol and levonorgestrel; exenatide is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed.

What clinical trials is ethinyl estradiol and levonorgestrel; exenatide in?

Ethinyl estradiol and levonorgestrel; exenatide has one completed clinical trial, NCT00254800, titled 'The Effects of Exenatide on Oral Contraceptive Pharmacokinetics in Healthy Females.' This Phase 1 study enrolled 38 healthy female participants in the United Kingdom and was completed.

Is ethinyl estradiol and levonorgestrel; exenatide the same as Ethinyl estradiol/Levonorgestrel (EE/LEVO)?

Yes, ethinyl estradiol and levonorgestrel; exenatide is also known as Ethinyl estradiol/Levonorgestrel (EE/LEVO) and Ethinyl estradiol/Levonorgestrel. These names refer to the same combination product being developed by AstraZeneca.