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ICI35, 868

Phase 2

Gastrointestinal Endoscopy | Small molecule | Gastrointestinal |AstraZeneca PLC|Last Updated: Dec 19, 2011

Target and mechanism

ModalitySmall molecule

Also known as ICI35,868 (propofol), ICI35,868 (Diprivan)

Success Probability

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Market & Valuation

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Trial Design

RandomizedPLACEBO_CONTROLLED
Total Trials1
Total Enrollment123

FDA Designations

No designations recorded

Clinical trial landscape

ICI35, 868 · 1 trial · 2 indications

Phase 2 1
NCT01189604Dose Rate Range Finding Study of Propofol for minimal-to Moderate Sedation on Upper & Lower Endoscopic TestsGastrointestinal Endoscopy
COMPLETED123 Analytics
PHASE2COMPLETED
Dose Rate Range Finding Study of Propofol for minimal-to Moderate Sedation on Upper & Lower Endoscopic Tests
Gastrointestinal EndoscopyUnlock trial analytics

Study Endpoints

Primary Endpoints

Modified Observers Assessment of Alertness/Sedation (MOAA/S) Score 2 Minutes From Beginning of Maintenance Period
2 minutes from the beginning of the maintenance period

The MOAA/S is a 6-point ordinal scale measuring a patient's level of sedation. Scores range from 0 (No response to painful stimulus \[trapezius squeeze\]) to 5 (Responds readily to name spoken in normal tone \[awake\]). MOAA/S scores were classified as 0-1, 2-4 and 5.

Modified Observers Assessment of Alertness/Sedation (MOAA/S) Score 4 Minutes From Beginning of Maintenance Period
4 minutes from the beginning of the maintenance period

The MOAA/S is a 6-point ordinal scale measuring a patient's level of sedation. Scores range from 0 (No response to painful stimulus \[trapezius squeeze\]) to 5 (Responds readily to name spoken in normal tone \[awake\]). MOAA/S scores were classified as 0-1, 2-4 and 5.

Secondary Endpoints

Patient Satisfaction With Sedation Instrument (PSSI) Questionnaire
24 - 48 hours after completion of the procedure
Blood Concentrations of Propofol
At the end of the initiation period and every 2 minutes during the maintenance period
Modified Observers Assessment of Alertness/Sedation (MOAA/S) at End of Initiation Period
Last measurement in maintenance period (3 minutes for arms 1-5; 1 minute for arm 6, 5 minute for arm 7)
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Arm1 - PlaceboPLACEBO_COMPARATOR -
Arm 2 - ICI35,868 (propofol)ACTIVE_COMPARATOR -
Arm 3 - ICI35,868 (propofol)ACTIVE_COMPARATOR -
Arm 4 - ICI35,868 (propofol)ACTIVE_COMPARATOR -
Arm 5 - ICI35,868 (propofol)ACTIVE_COMPARATOR -
Arm 6 - ICI35,868 (propofol)ACTIVE_COMPARATOR -
Arm 7 - ICI35,868 (propofol)ACTIVE_COMPARATOR -

Interventions

NameTypeDescription
PlaceboDRUGInfusion of placebo, same infusion rates as for arm 2
ICI35,868 (propofol)DRUGInfusion of propofol: initiation with 0.17 mg/kg for 3 minutes followed by maintenance with 25 µg/kg/minute
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Eligibility Criteria

Age Range20 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion Criteria: * Male or female (females of child bearing potential to confirm not pregnant via test or contraception) * Be undergoing a non-emergent esophagogastroduodenoscopy (EGD) or colonoscopy, including polypectomy that shall be completed within 1 hour Exclusion Criteria: * American So...

Countries:Japan
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Frequently asked questions about ICI35, 868

What is ICI35,868?

ICI35,868 is an investigational small molecule developed by AstraZeneca PLC under the ticker AZN. It is being studied as a sedative agent for gastrointestinal endoscopy procedures, including upper and lower endoscopic tests and gastrointestinal polypectomy. It is also known by the name propofol and the brand name Diprivan.

What is ICI35,868 used for in gastrointestinal endoscopy?

ICI35,868 is being developed to provide minimal-to-moderate sedation during upper and lower endoscopic tests, including gastrointestinal polypectomy procedures. It is a small molecule sedative studied in a Phase 2 dose rate range finding trial conducted in Japan in adults aged 20 years and older.

Who makes ICI35,868?

AstraZeneca PLC, which trades under the ticker AZN, is the developer of ICI35,868. The company sponsored the clinical development work for the drug, including the Phase 2 dose rate range finding study conducted in Japan in patients undergoing gastrointestinal endoscopy.

What phase is ICI35,868 in?

ICI35,868 is in Phase 2 development. It is investigational and has not been approved. One Phase 2 trial has been completed, and no trials are currently active. That completed study enrolled 123 participants and evaluated the drug for sedation during upper and lower endoscopic tests.

What clinical trials is ICI35,868 in?

ICI35,868 has been studied in one completed Phase 2 trial, NCT01189604, titled a dose rate range finding study of propofol for minimal-to-moderate sedation on upper and lower endoscopic tests. It enrolled 123 participants in Japan, was randomized and placebo-controlled, and included patients with gastrointestinal endoscopy and gastrointestinal polypectomy conditions.

Is ICI35,868 the same as propofol or Diprivan?

Yes. ICI35,868 is also known as propofol and by the brand name Diprivan. These names refer to the same small molecule, which AstraZeneca PLC is developing for sedation during gastrointestinal endoscopy procedures such as upper and lower endoscopic tests and gastrointestinal polypectomy.