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AZD5153

Phase 1

Malignant Solid Tumors | Small molecule | Oncology |AstraZeneca PLC|Last Updated: May 6, 2021

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment49
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03205176AZD5153 in Patients With Relapsed or Refractory Solid Tumors, Including LymphomasPHASE1 COMPLETED 49Jun 30, 2017Apr 8, 2021May 6, 20214 United States, Canada
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Study Endpoints
Primary Endpoints
Incidence of dose-limiting toxicity (DLT).
From the first dose of study treatment up to last day of cycle 1 (21 days)

DLTs will be determined from monitoring adverse events (AEs), and abnormal laboratory tests (clinical chemistry, hematology, and urinalysis), physical examinations, vital signs (blood pressure and pulse), and electrocardiogram (ECG).

Secondary Endpoints
Peak plasma concentration (Cmax)
Samples for single dose PK will be collected at prespecified time points on Day 1, Cycle 1 pre-dose on Day 2. Multiple-dose PK will be assessed from samples taken on Days 15 and 16 of Cycle 1.
The urine concentration of AZD5153 and its co-former (if appropriate).
Urine will be collected pre-dose (spot sample), and volumetrically from 0-6, 6-12, 12-24 hours on Day 1 and Day 15 of Cycle 1.
The effect of AZD 5153 on QTc interval.
ECGs will be performed at prespecified time points on Days 1 and 2 and 15 and 16 of Cycle 1.
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
AZD5153 MonotherapyEXPERIMENTALPatients will be enrolled in cohorts of up to 6 patients each in a dose escalating scheme to determine maximum tolerated dose (MTD). AZD5153 will be taken once per day (QD) or two times per day (BID) for 21 days as an oral capsule. Once the MTD is finalized, patients may be enrolled into an expansion cohort at the MTD.
AZD5153 + Olaparib Combination TherapyEXPERIMENTALPatients will be enrolled in cohorts of up to 6 patients each in a dose escalating scheme to determine MTD. AZD5153 will be taken as oral capsules BID in combination with 300 mg olaparib BID for 21 days.
Interventions
NameTypeDescription
AZD5153DRUGAZD5153 is to be taken as oral capsules once or twice per day each day in 21 day cycles. Dosing will continue until disease progression or other study discontinuation criteria are met.
OlaparibDRUGOlaparib, 300 mg, will be taken BID as oral capsules.
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Eligibility Criteria
Age Range18 Years — 130 Years
SexALL
Healthy VolunteersNo
Study Sites4

Inclusion Criteria for all Patients: 1. Patient must be able to understand the nature of the study and provide a signed and dated, written informed consent prior to any study specific procedures, sampling or analyses. 2. Patients should have the ability and willingness to comply with the study and ...

Countries:United StatesCanada
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