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Ezetimibe

Phase 3

Hyperlipidemia | Small molecule | Metabolic |Amgen Inc.|Last Updated: Nov 29, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindACTIVE_CONTROLLEDDMC
Total Trials1
Total Enrollment511
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01984424Goal Achievement After Utilizing an Anti-PCSK9 Antibody in Statin Intolerant Subjects-3PHASE3 COMPLETED 511Dec 10, 2013Nov 21, 2017Nov 29, 201858 United States, Australia +11
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Study Endpoints
Primary Endpoints
Percent Change From Baseline in LDL-C at the Mean of Weeks 22 and 24
Baseline and weeks 22 and 24
Percent Change From Baseline in LDL-C at Week 24
Baseline and week 24
Secondary Endpoints
Change From Baseline in LDL-C at the Mean of Weeks 22 and 24
Baselie and weeks 22 and 24
Change From Baseline in LDL-C at Week 24
Baseline and week 24
Percentage of Participants Who Achieved a Mean LDL-C at Weeks 22 and 24 of Less Than 70 mg/dL
Weeks 22 and 24
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part A: Atorvastatin 20 mg => PlaceboOTHERParticipants received atorvastatin 20 mg orally for 10 weeks (period 1) followed by placebo orally for 10 weeks (period 2), separated by a 2-week washout period.
Part A: Placebo => Atorvastatin 20 mgOTHERParticipants received placebo orally for 10 weeks (period 1) followed by atorvastatin 20 mg orally for 10 weeks (period 2), separated by a 2-week washout period.
Part B: EzetimibeACTIVE_COMPARATORParticipants received 10 mg ezetimibe orally only a day and placebo to evolocumab by subcutaneous injection once a month for 24 weeks.
Part B: EvolocumabEXPERIMENTALParticipants received 420 mg evolocumab by subcutaneous injection once a month and placebo to ezetimibe orally once a day for 24 weeks.
Part C: Open-label EvolocumabEXPERIMENTALParticipants who completed part B and were eligible to proceed to open-label extension part C and could choose quarterly between evolocumab 420 mg once a month or evolocumab 140 mg every 2 weeks for up to 2 years.
Interventions
NameTypeDescription
AtorvastatinDRUGAtorvastatin was supplied as over-encapsulated 20 mg tablets
Placebo to AtorvastatinDRUGPlacebo matching to atorvastatin supplied as over-encapsulated tablets
Placebo to EzetimibeOTHERPlacebo matching to Ezetimibe supplied as over-encapsulated tablets.
EzetimibeDRUGEzetimibe was supplied as 10 mg tablets, over-encapsulated for blinding.
Placebo to EvolocumabOTHERPlacebo matching to evolocumab supplied as single-use prefilled autoinjector/pen(s)
EvolocumabDRUGEvolocumab supplied as single-use prefilled autoinjector/pen(s)
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Eligibility Criteria
Age Range18 Years — 80 Years
SexALL
Healthy VolunteersNo
Study Sites58

Inclusion Criteria: * Male or female ≥ 18 to ≤ 80 years of age * Subject not at LDL-C goal * History of statin intolerance * Lipid lowering therapy has been stable prior to enrolment for at least 4 weeks * Fasting triglycerides ≤ 400 mg/dL Exclusion Criteria: * New York Heart Association (NYHA) I...

Countries:United StatesAustraliaCanadaCzechiaDenmarkFranceGermanyItalyNetherlandsNew ZealandNorwaySouth AfricaUnited Kingdom
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