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Denosumab CP4

Phase 1

Healthy Volunteer | Small molecule | Other |Amgen Inc.|Last Updated: Dec 29, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials1
Total Enrollment146
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02053753Bioequivalence Study of Denosumab CP4 Drug Product and Commercially Available Denosumab CP2 Drug ProductPHASE1 COMPLETED 146Feb 1, 2014Aug 1, 2014Dec 29, 20172 United States
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Study Endpoints
Primary Endpoints
Maximum Observed Drug Concentration (Cmax) of Denosumab
Day 1 predose up to day 127

Serum denosumab concentration-time data were analyzed by non-compartmental methods. Serum concentrations below the LLOQ (20.0 ng/mL) were set to 0 before data analysis.

Area Under the Drug Concentration-time Curve From Time 0 to 18 Weeks Post-dose (AUC0-18 Weeks) of Denosumab
Day 1 predose up to day 127

Serum denosumab concentration-time data were analyzed by non-compartmental methods. Serum concentrations below the LLOQ (20.0 ng/mL) were set to 0 before data analysis.

Secondary Endpoints
Time to Maximum Observed Concentration (Tmax) of Denosumab
Day 1 predose up to day 127
Half-life (T1/2) of Denosumab
Day 1 predose up to day 127
Area Under the Serum C-telopeptide (CTX1) Percent Inhibition-Time Curve From Time 0 to 18 Weeks Post-dose (AUEC0-18 Weeks)
Day 1 predose up to day 127
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Drug Product CP4EXPERIMENTALParticipants received a single dose of 120 mg denosumab manufactured using the new CP4 process subcutaneously on day 1.
Drug Product CP2EXPERIMENTALParticipants received a single dose of 120 mg denosumab manufactured using the current CP2 process subcutaneously on day 1.
Interventions
NameTypeDescription
Denosumab CP4DRUGDenosumab produced by a process referred to as CP4, administered subcutaneously.
Denosumab CP2DRUGDenosumab produced by a process referred to as CP2, administered subcutaneously.
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites2

Key Inclusion: * Healthy male and female, ages ≥ 18 to ≤ 65 years (inclusive) * Body weight \> 60 to \< 100 kg at time of screening * Clinically acceptable physical exams and laboratory tests (blood hematology, blood chemistry, urinalysis) and no history or evidence of any clinically significant me...

Countries:United States
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