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AG221

Phase 1

Healthy Volunteers | Small molecule | Other |Agios Pharmaceuticals, Inc.|Last Updated: Dec 14, 2015

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment30

FDA Designations

No designations recorded

Clinical trial landscape

AG221 · 1 trial · 1 indication

Phase 1 1
NCT02218346Food Effect Study of AG-221 in Healthy Male SubjectsHealthy Volunteers
COMPLETED30 Analytics
PHASE1COMPLETED
Food Effect Study of AG-221 in Healthy Male Subjects
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Study Endpoints

Primary Endpoints

Pharmacokinetic (PK) profile of AG-221
Blood samples will be drawn prior to the single-dose administration of AG-221 (within 30 minutes) on Day 1 of each period, and at the following time points post dose: 1, 2, 3, 4, 6, 9, 12, 18, 24, 48, 96, 168, 240, 336, and 504 hours.

Serial blood sampling at specified time points for determination of plasma concentration-time profiles and PK parameters of AG-221.

Incidence of adverse events
105 days
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Treatment A (unfed)ACTIVE_COMPARATORTreatment A: Single oral dose of AG-221 mesylate at Hour 0 on Day 1, following a 10-hour overnight fast.
Treatment B (fed)ACTIVE_COMPARATORTreatment B: Single oral dose of AG-221 mesylate at Hour 0 on Day 1, 30 minutes after the start of a high-fat breakfast.

Interventions

NameTypeDescription
AG221DRUGAG221 in fed and fasted conditions
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Eligibility Criteria

Age Range18 Years to 56 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Healthy adult male subjects 18 to 56 years of age, inclusive, at Screening. 2. Subjects who are able to understand and sign informed consent prior to the conduct of any protocol-specific screening procedures. 3. Subjects must be willing and able to complete all study assessme...

Countries:United States
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Frequently asked questions about AG221

What is AG221 used for?

AG221 is an investigational small molecule being studied in healthy volunteers. It is not approved for any disease and is in Phase 1 clinical development. The only completed trial evaluated its effects in healthy male subjects.

Who makes AG221?

AG221 is being developed by Agios Pharmaceuticals, Inc., a biopharmaceutical company traded on the NASDAQ under the ticker AGIO. The company conducted a Phase 1 study of AG221 in healthy volunteers.

What phase is AG221 in?

AG221 is in Phase 1 clinical development. One Phase 1 trial has been completed, and there are no active trials currently listed. The drug remains investigational and has not been approved by regulatory authorities.

What clinical trials is AG221 in?

AG221 has one completed clinical trial, NCT02218346, titled 'Food Effect Study of AG-221 in Healthy Male Subjects.' This Phase 1 study enrolled 30 healthy male participants in the United States and was completed.

Is AG221 the same as AG-221?

Yes, AG221 is also referred to as AG-221 in clinical trial documentation. The completed study NCT02218346 uses the name AG-221 in its title, confirming that both names refer to the same investigational drug.