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Niraparib

Phase 2

Endometrial Carcinoma | Small molecule | Oncology |Zai Lab Limited|Last Updated: Jan 5, 2024

Target and mechanism

Molecular targetPARP2, PARP1
Target classInhibitor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDBiomarker
Total Trials1
Total Enrollment83

FDA Designations

No designations recorded

Clinical trial landscape

Niraparib · 1 trial · 2 indications

Phase 2 1
NCT04716686Niraparib Monotherapy as Maintain and Recurrent Treatment of Endometrial Serous CarcinomaEndometrial Carcinoma
RECRUITING83 Analytics
PHASE2RECRUITING
Niraparib Monotherapy as Maintain and Recurrent Treatment of Endometrial Serous Carcinoma
Endometrial CarcinomaUnlock trial analytics

Study Endpoints

Primary Endpoints

PFS%(1 year)
assessed up to 12 months

for maintenance therapy arm

Objective Response Rate (ORR)
assessed up to 30months]

for maintenance therapy arm

Secondary Endpoints

PFS%(2 year)
assessed up to 24 months
Overall Survival (OS)
assessed up to 30 months
Median PFS
assessed up to 30 months
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Niraparib as maintenance therapy for Endometrial Serous CarcinomaEXPERIMENTALFor patients with baseline weight ≥ 77 kg and baseline platelets ≥ 150000/uL, a starting dose of 300 mg QD will be given; other patients will be given a starting dose of 200 mg QD. One treatment cycle is 28 days; follow-up and evaluation will be conducted every 2 cycles until the disease progression or patients cannot tolerate.
Niraparib as recurrent therapy for Endometrial CarcinomaEXPERIMENTALFor patients with baseline weight ≥ 77 kg and baseline platelets ≥ 150000/uL, a starting dose of 300 mg QD will be given; other patients will be given a starting dose of 200 mg QD. One treatment cycle is 28 days; follow-up and evaluation will be conducted every 2 cycles until the disease progression or patients cannot tolerate.

Interventions

NameTypeDescription
NiraparibDRUGPatients received oral niraparib 200/300 mg QD and every cycle (28 days) thereafter until disease progression.
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Eligibility Criteria

Age Range18 Years to N/A
SexFEMALE
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Women aged 18 or above * Histological confirmation of serous endometrial cancer or other types of endometrial cancer * FIGO stage III-IV * ESC Patients have received at least 6 cycles of first-line platinum containing chemotherapy after surgery and achieved CR, PR or SD; ESC p...

Countries:China
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Frequently asked questions about Niraparib

What is Niraparib used for in Endometrial Carcinoma?

Niraparib is being studied as a monotherapy for the maintenance and recurrent treatment of endometrial serous carcinoma, a type of endometrial cancer. It is currently in Phase 2 clinical development for this indication, with an ongoing trial enrolling 83 female patients aged 18 years and older in China.

What does Niraparib target?

Niraparib is a PARP inhibitor, belonging to the -parib class of drugs. It targets poly (ADP-ribose) polymerase (PARP) enzymes, which are involved in DNA repair. By inhibiting PARP, Niraparib may interfere with cancer cell repair mechanisms, potentially leading to cell death in tumors with certain genetic biomarkers.

Who is developing Niraparib?

Niraparib is being developed by Zai Lab Limited, a biopharmaceutical company traded on the NASDAQ under the ticker symbol ZLAB. The company is conducting a Phase 2 clinical trial of Niraparib for endometrial serous carcinoma in China.

What phase is Niraparib in for endometrial cancer?

Niraparib is in Phase 2 clinical development for endometrial carcinoma, specifically for the maintenance and recurrent treatment of endometrial serous carcinoma. The drug is investigational and has not been approved for this indication. The ongoing Phase 2 trial is currently recruiting participants.

What clinical trials is Niraparib in?

Niraparib is being evaluated in a single active Phase 2 clinical trial with the identifier NCT04716686. The trial, titled 'Niraparib Monotherapy as Maintain and Recurrent Treatment of Endometrial Serous Carcinoma,' is recruiting 83 female participants in China. The study is controlled but not randomized or double-blinded, and it uses biomarker selection.