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CHR-2797: Aminopeptidase inhibitor

Phase 1

Acute Myeloid Leukemia | Small molecule | Oncology |cbdMD, Inc.|Last Updated: Oct 22, 2010

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment57

FDA Designations

No designations recorded

Clinical trial landscape

CHR-2797: Aminopeptidase inhibitor · 1 trial · 3 indications

Phase 1 1
NCT00689000Safety and Anti-Disease Activity of CHR-2797 (Tosedostat) in Elderly and/or Treatment Refractory Patients With Acute Myeloid Leukemia (AML) and Multiple Myeloma (MM)Acute Myeloid Leukemia
COMPLETED57 Analytics
PHASE1COMPLETED
Safety and Anti-Disease Activity of CHR-2797 (Tosedostat) in Elderly and/or Treatment Refractory Patients With Acute Myeloid Leukemia (AML) and Multiple Myeloma (MM)
Acute Myeloid LeukemiaUnlock trial analytics

Study Endpoints

Primary Endpoints

Phase I: To determine the safety, tolerability, dose-limiting toxicity (DLT) and maximum tolerated dose (MTD) of CHR-2797 when administered orally, once daily.
first 28 days of treatment
Phase II: To evaluate the anti-leukaemia/myeloma effect of the recommended dose of single agent CHR-2797.
End of study

Secondary Endpoints

Phase I and II: To determine trough levels of CHR-2797 when administered orally, once daily, at different dose levels.
End of study
Phase II: To evaluate the safety and tolerability of the recommended dose of CHR-2797 when administered orally, once daily.
End of study
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
CHR-2797 (tosedostat)EXPERIMENTALoral, once daily administration of CHR-2797 to determine safety \& anti-disease activity.

Interventions

NameTypeDescription
CHR-2797 (tosedostat): Aminopeptidase inhibitorDRUGPhase I: Once daily, oral ingestion of CHR-2797 capsules (60mg, 90mg, 130mg or 180mg) depending on cohort Phase II: Once daily, oral ingestion of 130mg CHR-2797 (recommended dose from Phase I) until progressive disease or withdrawal from the study
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Signed, informed consent. * Patients with AML, MDS (subtype RAEB-1 or RAEB-2), or MM whose disease has relapsed or is refractory to front line and/ or salvage therapy; elderly patients (≥ 60 years) with AML, MDS, MM who are not candidates for chemotherapy and for whom other th...

Countries:United Kingdom
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Frequently asked questions about CHR-2797: Aminopeptidase inhibitor

What is CHR-2797 used for in Acute Myeloid Leukemia?

CHR-2797, also known as tosedostat, is an investigational small molecule being studied for the treatment of Acute Myeloid Leukemia (AML). It is an aminopeptidase inhibitor in Phase 1 clinical development. The drug is intended for elderly and/or treatment refractory patients with AML, as well as those with multiple myeloma and myelodysplastic syndrome.

What does CHR-2797 target?

CHR-2797 targets aminopeptidases, which are enzymes involved in protein processing. By inhibiting these enzymes, the drug aims to disrupt cellular processes in cancer cells. This mechanism is being explored as a potential therapeutic approach for Acute Myeloid Leukemia and other hematologic malignancies.

Who makes CHR-2797?

CHR-2797 is being developed by cbdMD, Inc., a company traded under the ticker YCBD. The drug is in Phase 1 clinical development for Acute Myeloid Leukemia. It is a small molecule therapeutic being investigated for its potential anti-disease activity in hematologic cancers.

What phase is CHR-2797 in?

CHR-2797 is in Phase 1 clinical development. It is an investigational drug, not yet approved by regulatory authorities. The Phase 1 trial has been completed, having enrolled 57 participants. The study focused on safety and anti-disease activity in patients with Acute Myeloid Leukemia and related conditions.

What clinical trials is CHR-2797 in?

CHR-2797 has one completed clinical trial, identified as NCT00689000. This Phase 1 study evaluated the safety and anti-disease activity of CHR-2797 (tosedostat) in elderly and/or treatment refractory patients with Acute Myeloid Leukemia and Multiple Myeloma. The trial was conducted in the United Kingdom and enrolled 57 participants.

Is CHR-2797 the same as tosedostat?

Yes, CHR-2797 is also known as tosedostat. The clinical trial NCT00689000 refers to the drug as CHR-2797 (tosedostat). This aminopeptidase inhibitor is being investigated for Acute Myeloid Leukemia and other hematologic conditions, and is currently in Phase 1 development.