Recent Updates
Recently added Catalysts

Part 1 TPST-1120

Phase 1

Hepatocellular Carcinoma | Small molecule | Oncology |Tempest Therapeutics, Inc.|Last Updated: Jul 3, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment38
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03829436TPST-1120 as Monotherapy and in Combination With Nivolumab in Subjects With Advanced CancersPHASE1 COMPLETED 38Mar 20, 2019Sep 7, 2022Jul 3, 202311 United States
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Incidence of dose limiting toxicities (DLTs) of TPST-1120 as a single agent and in combination with nivolumab.
From start of treatment to end of treatment, up to 36 months
Incidence of treatment-emergent adverse events as assessed by NCI-CTCAE v5.0 of TPST-1120 as a single agent and in combination with nivolumab.
From start of treatment to end of treatment, up to 36 months
Identify the maximum tolerated dose
From start of treatment to end of treatment, up to 36 months

Incidence of dose limiting toxicities (DLTs) of TPST-1120 as a single agent and in combination with nivolumab.

Secondary Endpoints
Assess pharmacokinetics: Maximum serum concentration (Cmax)
Day 1, 2, 8 of Cycle 1 and Day 1 of Cycle 3 (cycle can be 21 or 28 days, depending on cohort assignment)
Assess pharmacokinetics: Area under the curve (AUC)
Day 1, 2, 8 of Cycle 1 and Day 1 of Cycle 3, Day 1 of Cycles 5+ (cycle can be 21 or 28 days, depending on cohort assignment)
Objective response rate
From start of treatment to end of treatment, up to 36 months
Unlock Study Endpoints
Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part 1 TPST-1120EXPERIMENTALSubjects will receive escalating doses of TPST-1120 administered orally twice daily continuously until MTD is reached or until disease progression
Part 2 TPST-1120 + nivolumabEXPERIMENTALSubjects will receive escalating doses of TPST-1120 administered orally twice daily in combination with nivolumab administered intravenously every 28 days until MTD is reached for TPST-1120 or until disease progression.
Part 3 TPST-1120EXPERIMENTALSelected dose of TPST-1120 administered orally twice daily until disease progression
Part 4 TPST-1120 + nivolumabEXPERIMENTALSelected dose of TPST-1120 administered orally twice daily in combination with nivolumab administered intravenously every 28 days until MTD is reached for TPST-1120 or until disease progression
Interventions
NameTypeDescription
Part 1 TPST-1120DRUGSubjects will receive escalating doses of TPST-1120 administered orally twice daily continuously until MTD is reached or until disease progression
Part 2 TPST-1120 + nivolumabDRUGSubjects will receive escalating doses of TPST-1120 administered orally twice daily
Part 3 TPST-1120DRUGSelected dose of TPST-1120 administered orally twice daily until disease progression
Part 4 TPST-1120 + nivolumabDRUGSelected dose of TPST-1120 administered orally twice daily in combination with nivolumab administered intravenously every 28 days until MTD is reached for TPST-1120 or until disease progression
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites11

Inclusion Criteria * Eastern Cooperative Oncology Group performance status of 0-1 at enrollment * Progressive disease or previously untreated tumors for which no standard therapy exists or treatment naïve at the time of study entry are eligible * Have at least one measurable lesion according to REC...

Countries:United States
Unlock Eligibility Criteria