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TV-46046-mL

Phase 1

Pregnancy | Small molecule | Endocrine |Teva Pharmaceutical Industries Limited|Last Updated: Feb 12, 2024

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLEDDMC
Total Trials1
Total Enrollment12

FDA Designations

No designations recorded

Clinical trial landscape

TV-46046-mL · 1 trial · 2 indications

Phase 1 1
NCT02817464Study to Evaluate Suppression of Ovulation and Pharmacokinetics of Medroxyprogesterone Acetate Following Administration of TV-46046 in Women With Ovulatory CyclePregnancy
COMPLETED12 Analytics
PHASE1COMPLETED
Study to Evaluate Suppression of Ovulation and Pharmacokinetics of Medroxyprogesterone Acetate Following Administration of TV-46046 in Women With Ovulatory Cycle
PregnancyUnlock trial analytics

Study Endpoints

Primary Endpoints

Part 1: Serum Medroxyprogesterone Acetate (MPA) Concentration at Day 1
Day 1

'Overall number of participants analyzed' = participants evaluable for this outcome measure.

Part 1: Serum MPA Concentration at Day 7
Day 7
Part 1: Serum MPA Concentration at Day 28
Day 28
Part 1: Serum MPA Concentration at Day 91
Day 91
Part 1: Serum MPA Concentration at Day 182
Day 182
Part 1: Serum MPA Concentration at Day 210
Day 210
Part 1: Maximum Observed Serum Concentration (Cmax) of MPA
Day 0 up to Week 52
Part 1: Observed Serum Drug Concentration at Day 182 (C182) of MPA
Day 182
Part 1: Time to Reach Cmax (Tmax) of MPA
Day 0 up to Week 52
Part 1: Area Under the Serum Drug Concentration by Time Curve From Time 0 to Day 182 (AUC0-182) of MPA
Day 0 up to Day 182
Part 1: Area Under the Serum Drug Concentration by Time Curve From Time 0 to Day 210 (AUC0-210) of MPA
Day 0 up to Day 210
Part 1: Area Under the Serum Drug Concentration by Time Curve From Time 0 to Infinity (AUC0-∞) of MPA
Day 0 up to Week 52
Part 1: Apparent Terminal Half-life (t1/2) of MPA
Day 0 up to Week 52
Part 2: Time to Ovulation
Day 0 up to Week 78

Ovulation was defined as a single elevated serum progesterone ≥4.7 ng/mL.

Secondary Endpoints

Part 1: Time to Ovulation
Day 0 up to Week 78
Part 2: Cmax of MPA
Day 0 up to Week 52
Part 2: Tmax of MPA
Day 0 up to Week 52
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelSINGLE_GROUP
PurposeOTHER

Treatment Arms

ArmTypeDescription
TV-46046 - 1EXPERIMENTAL -
TV-46046 - 2EXPERIMENTAL -

Interventions

NameTypeDescription
TV-46046 - 400 mg/mLDRUGA single subcutaneous injection in the abdomen of undiluted TV-46046 - 400 mg/mL
TV-46046 - 200 mg/mLDRUGA single subcutaneous injection in the abdomen of saline-diluted TV-46046 - 200 mg/mL
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Eligibility Criteria

Age Range18 Years to 40 Years
SexFEMALE
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * has regular menstrual cycle (24 to 35 days) * is at low risk of pregnancy (ie, sterilized, in exclusively same-sex partnership, in monogamous relationship with vasectomized partner, or using non-hormonal IUD) * is in good general health as determined by a medical history and p...

Countries:United States
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Frequently asked questions about TV-46046-mL

What is TV-46046 used for?

TV-46046 is an investigational small molecule being developed for contraception and pregnancy prevention. It is a long-acting injectable formulation of medroxyprogesterone acetate intended for use in women of reproductive age. The drug is currently in Phase 1 clinical development and is not yet approved by regulatory authorities.

Who makes TV-46046?

TV-46046 is being developed by Teva Pharmaceutical Industries Limited, a company publicly traded under the ticker symbol TEVA. The drug is an investigational product candidate in the company's endocrine therapeutic area pipeline, focused on women's reproductive health and contraception.

What phase is TV-46046 in?

TV-46046 is in Phase 1 clinical development. Three Phase 1 trials have been completed, with a total of 87 participants enrolled across studies conducted in the United States and the Dominican Republic. The drug remains investigational and has not received regulatory approval for any indication.

What clinical trials is TV-46046 in?

TV-46046 has completed three Phase 1 clinical trials: NCT02817464 evaluated suppression of ovulation and pharmacokinetics in 12 women with ovulatory cycles; NCT03700658 assessed injection pain and local tolerability in 27 women; and NCT04682353 studied pharmacokinetics in 60 healthy women of reproductive age. All trials were completed.

How does TV-46046 work?

TV-46046 is a small molecule formulation of medroxyprogesterone acetate, a progestin hormone. It works by delivering a sustained release of medroxyprogesterone acetate to suppress ovulation, thereby preventing pregnancy. The drug is administered via subcutaneous injection to provide long-acting contraceptive effects.

Is TV-46046 the same as medroxyprogesterone acetate?

TV-46046 is a proprietary long-acting injectable formulation of medroxyprogesterone acetate, not the same as standard immediate-release versions. It is designed to provide sustained drug release over an extended period. The active pharmaceutical ingredient is medroxyprogesterone acetate, but TV-46046 is a distinct product candidate in development.