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Hydrocodone bitartrate

Phase 1

Hepatic Impairment | Small molecule | Gastrointestinal |Teva Pharmaceutical Industries Limited|Last Updated: Apr 24, 2012

Target and mechanism

ModalitySmall molecule

Also known as Hydrocodone bitartrate extended-release tablet, Hydrocodone Bitartrate extended-release tablet

Success Probability

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Market & Valuation

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Trial Design

CONTROLLEDBiomarker
Total Trials1
Total Enrollment16

FDA Designations

No designations recorded

Clinical trial landscape

Hydrocodone bitartrate · 2 trials · 2 indications

Phase 1 2
NCT01319279A Study to Evaluate the Pharmacokinetics of the Hydrocodone Extended-Release Tablet (CEP-33237) in Subjects With Normal Hepatic Function and Subjects With Moderate Hepatic ImpairmentHepatic Impairment
COMPLETED16 Analytics
NCT01319266A Study to Assess the Pharmacokinetics of the Hydrocodone Extended-Release Tablet (CEP-33237) in Subjects With Normal Renal Function and Subjects With Varying Degrees of Renal ImpairmentRenal Impairment
COMPLETED55 Analytics
PHASE1COMPLETED
A Study to Evaluate the Pharmacokinetics of the Hydrocodone Extended-Release Tablet (CEP-33237) in Subjects With Normal Hepatic Function and Subjects With Moderate Hepatic Impairment
Hepatic ImpairmentUnlock trial analytics
PHASE1COMPLETED
A Study to Assess the Pharmacokinetics of the Hydrocodone Extended-Release Tablet (CEP-33237) in Subjects With Normal Renal Function and Subjects With Varying Degrees of Renal Impairment
Renal ImpairmentUnlock trial analytics

Study Endpoints

Primary Endpoints

Pharmacokinetics (AUC and Cmax) after a single dose
7 days
Maximum observed plasma drug concentration (Cmax)
Between baseline and 144 hours following drug administration
Area under the plasma drug concentration-by-time curve (AUC) from time 0 to infinity (AUC0-∞)
Between baseline and 144 hours following drug administration

Secondary Endpoints

Safety (occurrence of adverse events, labs, ECG, physical exam, vital signs, oxygen saturation)
throughout the 37 day study period (includes screening, drug administration and pharmacokinetics sampling period, and follow-up)
Assess the safety of a single 45-mg dose of the hydrocodone bitartrate extended release tablet
Safety will be assessed from the start of study drug administration through the follow-up visit 48 to 72 hours after discharge from the study center.
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Normal Hepatic FunctionEXPERIMENTALIntervention Drug: Hydrocodone bitartrate extended-release tablet
Moderate Hepatic ImpairmentEXPERIMENTALIntervention Drug: Hydrocodone bitartrate extended-release tablet
Normal Renal FunctionEXPERIMENTALSubjects with normal renal function
Mild Renal ImpairmentEXPERIMENTALSubjects with mild renal impairment (defined by an estimated creatinine clearance of \> 50 and up to 80 mL/min)
Moderate Renal ImpairmentEXPERIMENTALSubjects with moderate renal impairment (defined by an estimated creatinine clearance of 30-50 mL/min)
Severe Renal ImpairmentEXPERIMENTALSubjects with severe renal impairment (defined by an estimated creatinine clearance of less than 30 mL/min)
End Stage Renal Disease (ESRD)EXPERIMENTALSubjects with ESRD (defined as being on hemodialysis for at least 6 months prior to enrollment and be receiving standard in-center dialysis treatments three times a week)

Interventions

NameTypeDescription
Hydrocodone bitartrate extended-release tabletDRUG15 mg (single dose)
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. All subjects: * Written informed consent is obtained 2. Subjects with normal hepatic function: * The subject is in generally good health (age-appropriate) as determined by medical and psychiatric history, physical examination, ECG, serum chemistry, hematology, coagula...

Countries:United States
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