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TD-5202

Phase 1

Healthy | Small molecule | Other |Theravance Biopharma, Inc.|Last Updated: Jan 14, 2021

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLEDDMC
Total Trials1
Total Enrollment56

FDA Designations

No designations recorded

Clinical trial landscape

TD-5202 · 1 trial · 1 indication

Phase 1 1
NCT04044339Single and Multiple Ascending Dose, First-in- Human Study in Healthy SubjectsHealthy
COMPLETED56 Analytics
PHASE1COMPLETED
Single and Multiple Ascending Dose, First-in- Human Study in Healthy Subjects
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

To assess the safety and tolerability of SAD of TD-5202 by assessing the number, severity and type of treatment emergent adverse events
Day 1 through Day 8
To assess the safety and tolerability of MAD of TD-5202 by assessing the number, severity and type of treatment emergent adverse events
Day 1 through Day 17
Pharmacokinetics (PK) of TD-5202 when given as an SAD: AUC
Day 1 through Day 4

Area under the plasma concentration-time curve (AUC)

Pharmacokinetics (PK) of TD-5202 when given as a SAD: Cmax
Day 1 through Day 4

Maximum observed concentration (Cmax)

Pharmacokinetics (PK) of TD-5202 when given as a SAD: Tmax
Day 1 through Day 4

Time to reach maximum observed concentration (Tmax)

PK of TD-5202 when given as an SAD: CL/F
Day 1 through Day 4

Oral Clearance (CL/F)

PK of TD-5202 when given as an SAD: Vz/F
Day 1 through Day 4

Terminal Phase Volume of Distribution(Vz/F)

PK of TD-5202 when given as an SAD: Kel
Day 1 through Day 4

Elimination Rate (Kel)

PK of TD-5202 when given as an SAD: t 1/2
Day 1 through Day 4

Halflife (t 1/2)

PK of TD-5202 when given as an MAD: AUC
Day 1 and Day 10

Area under the plasma concentration-time curve (AUC)

PK of TD-5202 when given as an MAD: Cmax
Day 1 and Day 10

Maximum observed concentration (Cmax)

PK of TD-5202 when given as an MAD: Tmax
Day 1 and Day 10

Time to reach maximum observed concentration (Tmax)

PK of TD-5202 when given as an MAD: C trough
Day 2, 4, 6, 8

concentration at trough (after multiple dosing usually after reaching steady state) (C trough)

PK of TD-5202 when given as an MAD: Css
Day 10

concentration at steady state (Css)

PK of TD-5202 when given as an MAD: CL/Fss
Day 10

Oral clearance at steady state (CL/Fss)

PK of TD-5202 when given as an MAD: Cmin
Day 10

Concentration minimum (after single dosing) (Cmin)

PK of TD-5202 when given as an MAD: Vz/Fss
Day 10

Terminal phase volume of distribution at steady state (Vz/Fss)

PK of TD-5202 when given as an MAD: Kel
Day 10

Elimination Rate (Kel)

PK of TD-5202 when given as an MAD: t 1/2
Day 10

Halflife (t 1/2)

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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
TD-5202 for SAD (Part A)EXPERIMENTAL6 out of 8 subjects per cohort (up to 4 cohorts) will be randomized to receive TD-5202
Placebo for SAD (Part A)PLACEBO_COMPARATOR2 out of 8 subjects per cohort (up to 4 cohorts) will be randomized to receive placebo
TD-5202 for MAD (Part B)EXPERIMENTAL6 out of 8 subjects per cohort (up to 3 cohorts) will be randomized to receive TD-5202
Placebo for MAD (Part B)PLACEBO_COMPARATOR2 out of 8 subjects per cohort (up to 3 cohorts) will be randomized to receive placebo.

Interventions

NameTypeDescription
TD-5202DRUGStudy Drug to be administered orally
PlaceboDRUGPlacebo to be administered orally
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Eligibility Criteria

Age Range19 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male or female, 19 - 55 years old * Willing and able to give informed consent and comply with the study * Medically healthy with no clinically significant medical history * Body mass index (BMI) 18 to 32 kg/m2 and weighs at least 50 kg * Women of child bearing potential must h...

Countries:United States
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Frequently asked questions about TD-5202

What is TD-5202?

TD-5202 is an investigational small molecule being developed by Theravance Biopharma, Inc. (TBPH). It is currently in Phase 1 clinical development. The drug has been studied in healthy volunteers, and its therapeutic area is classified as Other.

What is TD-5202 used for?

TD-5202 is being studied for use in healthy subjects. It is an investigational small molecule in Phase 1 clinical development. The drug has not been approved for any indication and is still in early-stage clinical trials.

Who makes TD-5202?

TD-5202 is being developed by Theravance Biopharma, Inc., a biopharmaceutical company traded on the NASDAQ under the ticker TBPH. The company is conducting clinical trials to evaluate the safety and tolerability of this investigational small molecule.

What phase is TD-5202 in?

TD-5202 is in Phase 1 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities. The drug is being studied in healthy volunteers to assess its safety, tolerability, and pharmacokinetics.

What clinical trials is TD-5202 in?

TD-5202 has one completed Phase 1 clinical trial, identified as NCT04044339. This was a first-in-human study titled "Single and Multiple Ascending Dose, First-in-Human Study in Healthy Subjects." The trial enrolled 56 participants in the United States and was randomized, double-blind, and placebo-controlled.

Is TD-5202 FDA approved?

No, TD-5202 is not FDA approved. It is an investigational drug currently in Phase 1 clinical development. The drug has been studied in a completed Phase 1 trial in healthy volunteers, but it has not received regulatory approval for any use.