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TIMP-GLIA

Phase 2

Celiac Disease | Small molecule | Gastrointestinal |Takeda Pharmaceutical Company Limited|Last Updated: Aug 12, 2020

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLEDDMC
Total Trials2
Total Enrollment57

FDA Designations

No designations recorded

Clinical trial landscape

TIMP-GLIA · 2 trials · 1 indication

Phase 2 1Phase 1 1
NCT03738475Study of the Safety, Pharmacodynamics, Efficacy, and PK of TIMP-GLIA in Subjects With Celiac DiseaseCeliac Disease
COMPLETED34 Analytics
PHASE2COMPLETED
Study of the Safety, Pharmacodynamics, Efficacy, and PK of TIMP-GLIA in Subjects With Celiac Disease
Celiac DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Change From Baseline in Interferon-Gamma Spot Forming Units (IFN-gamma SFUs) in a Gliadin-specific Enzyme-linked Immunospot (ELISpot) at Day 20
Baseline (Day 15/Day 1), Day 20

The spots formed by interferon-gamma-secreting T-cells were counted with an automated ELISPOT analyzer. The average spot-forming units (SFU) per antigen was calculated. A response was considered positive when the average SFU in wells with a given peptide was at least twice that of the average SFU in the no-peptide control wells. Baseline (Day 15/Day 1) was defined as Day 15 (or Day 1 if enough blood was not available on Day 15). Peripheral blood mononuclear cell is PBMC.

Number of Participants Reporting One or More Treatment-emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs)
From Day 1 up to Day 180
Number of Participants With Grade 3 or Higher TEAEs and Drug-related Adverse Events
From Day 1 up to Day 180

AE Grades will be evaluated as per National Cancer Institute Common Terminology Criteria for Adverse Event (NCI CTCAE), version 4.0. Grade 1 scaled as Mild; Grade 2 scaled as Moderate; Grade 3 scaled as severe or medically significant but not immediately life-threatening; Grade 4 scaled as life-threatening consequences; and Grade 5 scaled as death related to AE. Drug-related adverse events are those that the investigator assessed as possibly or probably related to the study treatment.

Number of Participants With Clinically Significant Physical Examination Findings
From Day 1 up to Day 60
Number of Participants With Clinically Significant Electrocardiograms (ECG) Findings
From Day 1 up to Day 60
Number of Participants With Clinically Significant Change From Baseline in Arterial Oxygen Saturation Levels
From Day 1 up to Day 60
Number of Participants With Clinically Significant Change From Baseline in Vital Signs Values
From Day 1 up to Day 60
Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 3
Baseline (Day 1 pre-dose) and Day 3

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 7
Baseline (Day 1 pre-dose) and Day 7

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 8
Baseline (Day 1 pre-dose) and Day 8

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 10
Baseline (Day 1 pre-dose) and Day 10

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 14
Baseline (Day 1 pre-dose) and Day 14

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 38
Baseline (Day 1 pre-dose) and Day 38

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C1q Binding at Day 60
Baseline (Day 1 pre-dose) and Day 60

Baseline is defined as Day 1 pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C3a and SC5B-9 Levels at 15 Minutes Post-dose on Day 1
Baseline (Day 1 pre-dose) and 15 minutes (min) post-dose on Day 1

Baseline was defined as Day 1 Pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C3a and SC5B-9 Levels at 30 Minutes Post-dose on Day 1
Baseline (Day 1 pre-dose) and 30 min post-dose on Day 1

Baseline was defined as Day 1 Pre-dose.

Part B: Change From Baseline (Day 1 Pre-dose) in C3a and SC5B-9 Levels at Day 2
Baseline (Day 1 pre-dose) and Day 2

Baseline was defined as Day 1 Pre-dose.

Number of Participants With Clinically Significant Change From Baseline in Hematology, Serum Chemistry, Coagulation, and Urinalysis
From Day 1 up to Day 60
Part A (Greater Than or Equal to [>=] 4.0 mg/kg) and Part B: Number of Participants With Clinically Significant Change From Baseline in Gliadin-Specific T-cell Proliferation and Cytokine Release Markers
Part A (>=4.0 mg/kg): Day 1 pre-dose up to 144 hours post-dose on Day 7; Part B: Day 8 pre-dose up to 144 hours post-dose on Day 14
Number of Participants With Clinically Significant Laboratory Abnormalities
From Day 1 up to Day 60

Secondary Endpoints

Change From Baseline in Gliadin-specific T Cell Proliferation by Enzyme-linked Immunosorbent Assay (ELISA) at Day 20
Baseline (Day 15/Day 1), Day 20
Change From Baseline in Gliadin-specific T Cell Cytokine Secretion by ELISA at Day 20
Baseline (Day 15/Day 1), Day 20
Change From Baseline in Gut-Homing CD4, CD8 and Gamma Delta T-cells by Mass Cytometry (CyTOF) at Day 20
Baseline (Day 15/Day 1), Day 20
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
TIMP-GLIAEXPERIMENTAL8 mg/kg up to a maximum of 650 mg administered intravenously on days 1 and 8.
PlaceboPLACEBO_COMPARATORNormal saline administered intravenously on days 1 and 8.
Part A, Cohort 1: 0.1 mg/kgEXPERIMENTALTIMP-GLIA 0.1 mg/kg, infusion, intravenously, once on Day 1.
Part A, Cohort 2: 0.5 mg/kgEXPERIMENTALTIMP-GLIA 0.5 mg/kg, infusion, intravenously, once on Day 1.
Part A, Cohort 3: 1.0 mg/kgEXPERIMENTALTIMP-GLIA 1.0 mg/kg, infusion, intravenously, once on Day 1.
Part A, Cohort 4: 2.0 mg/kgEXPERIMENTALTIMP-GLIA 2.0 mg/kg, infusion, intravenously, once on Day 1.
Part A, Cohort 5: 4.0 mg/kgEXPERIMENTALTIMP-GLIA 4.0 mg/kg, infusion, intravenously, once on Day 1.
Part A, Cohort 6: 8.0 mg/kgEXPERIMENTALTIMP-GLIA 8.0 mg/kg, infusion, intravenously, once on Day 1.
Part B, Cohort 1: 2.0 mg/kgEXPERIMENTALTIMP-GLIA 2.0 mg/kg, infusion, intravenously, once on Days 1 and 8.
Part B, Cohort 2: 4.0 mg/kgEXPERIMENTALTIMP-GLIA 4.0 mg/kg, infusion, intravenously, once on Days 1 and 8.
Part B, Cohort 3: 8.0 mg/kgEXPERIMENTALTIMP-GLIA 8.0 mg/kg, infusion, intravenously, once on Days 1 and 8.

Interventions

NameTypeDescription
TIMP-GLIADRUG8 mg/kg up to a maximum of 650 mg administered intravenously on days 1 and 8.
PlaceboDRUGAdministered intravenously on days 1 and 8.
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Eligibility Criteria

Age Range18 Years to 70 Years
SexALL
Healthy VolunteersNo
Study Sites8

Key Inclusion Criteria: 1. Male or nonpregnant female, ages 18 to 70 years inclusive, at Screening Visit. 2. Biopsy-confirmed CD (intestinal histology showing villous atrophy). 3. Positive for human leukocyte antigen (HLA)-DQ2 or HLA-DQ2/DQ8 - results will be obtained at Screening if unknown or res...

Countries:United States
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Frequently asked questions about TIMP-GLIA

What is TIMP-GLIA used for in celiac disease?

TIMP-GLIA is an investigational small molecule being developed for the treatment of celiac disease. It is designed to address the gastrointestinal condition, though its exact mechanism of action has not been disclosed. The drug is currently in clinical development and has not been approved by regulatory authorities.

Who is developing TIMP-GLIA?

TIMP-GLIA is being developed by Takeda Pharmaceutical Company Limited, a global biopharmaceutical company listed on the New York Stock Exchange under the ticker TAK. Takeda is conducting clinical trials to evaluate the safety, tolerability, pharmacokinetics, pharmacodynamics, and efficacy of TIMP-GLIA in adult patients with celiac disease.

What phase is TIMP-GLIA in?

TIMP-GLIA is in Phase 2 clinical development for celiac disease. It has completed a Phase 1 study and a Phase 2 study, both of which have finished. The drug remains investigational and is not yet approved for commercial use.

What clinical trials has TIMP-GLIA been studied in?

TIMP-GLIA has been evaluated in two completed clinical trials in the United States. The first, NCT03486990, was a Phase 1 study of safety, tolerability, and pharmacokinetics in 23 adults with celiac disease. The second, NCT03738475, was a Phase 2 study of safety, pharmacodynamics, efficacy, and pharmacokinetics in 34 adults with celiac disease.

Is TIMP-GLIA FDA approved?

TIMP-GLIA is not FDA approved. It is an investigational drug that has completed Phase 1 and Phase 2 clinical trials for celiac disease. The drug is still in clinical development and has not received marketing authorization from the U.S. Food and Drug Administration or any other regulatory agency.