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TAK-875 and Glimepiride

Phase 1

Pharmacokinetics | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Sep 13, 2012

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment28

FDA Designations

No designations recorded

Clinical trial landscape

TAK-875 and Glimepiride · 1 trial · 1 indication

Phase 1 1
NCT01496443TAK-875 Glimepiride Drug-Interaction StudyPharmacokinetics
COMPLETED28 Analytics
PHASE1COMPLETED
TAK-875 Glimepiride Drug-Interaction Study
PharmacokineticsUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax: Maximum Observed Plasma Concentration Pharmacokinetic Parameter for TAK-875
Day 17 and Day 18.

Maximum observed plasma concentration (Cmax) is the peak plasma concentration of a drug after administration, obtained directly from the plasma concentration-time curve.

Cmax: Maximum Observed Plasma Concentration Pharmacokinetic Parameter for Glimepiride
Day 1 and Day 18.

Maximum observed plasma concentration (Cmax) is the peak plasma concentration of a drug after administration, obtained directly from the plasma concentration-time curve.

Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) Pharmacokinetic Parameter for TAK-875
Day 17 and Day 18.

Time to reach the maximum plasma concentration (Cmax), equal to time (hours) to Cmax.

Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) Pharmacokinetic Parameter for Glimepiride
Day 1 and Day 18.

Time to reach the maximum plasma concentration (Cmax), equal to time (hours) to Cmax

AUC(0-tlqc): Area Under the Plasma Concentration-Time Curve From Time 0 to the Time of the Last Quantifiable Concentration Pharmacokinetic Parameter for Glimepiride
Day 1 and Day 18.

(AUC(0-tlqc) is a measure of total plasma exposure to the drug from Time 0 to Time of the Last Quantifiable Concentration (AUC\[0-tlqc\]).

AUC(0-inf): Area Under the Plasma Concentration-time Curve from Time 0 to Infinity Pharmacokinetic Parameter for Glimepiride
Day 1 and Day 18.

AUC(0-inf) is measure of area under the plasma concentration-time curve from time 0 to infinity after drug administration.

AUC(0-24): Area Under the Plasma Concentration-Time Curve From Time 0 to 24 Hours Postdose Pharmacokinetic Parameter for TAK-875
Day 17 and Day 18.

AUC(0-24) is measure of area under the curve over the dosing interval (tau) (AUC(0-tau\]), where tau is the length of the dosing interval - 24 hours in this study).

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Study Design & Arms

AllocationNA
MaskingSINGLE
ModelSINGLE_GROUP

Treatment Arms

ArmTypeDescription
TAK-875 & Glimepiride QDEXPERIMENTALTAK-875 50 mg, tablets, orally and glimepiride 2 mg, capsules, orally and glimepiride placebo matching capsules, orally, once daily on dosing days for up to 19 days.

Interventions

NameTypeDescription
TAK-875 and GlimepirideDRUG -
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Eligibility Criteria

Age Range18 Years to 68 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. In the opinion of the investigator, the participant is capable of understanding and complying with protocol requirements. 2. The participant or, when applicable, the participant's legally acceptable representative signs and dates a written, informed consent form and any requi...

Countries:United States
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Frequently asked questions about TAK-875 and Glimepiride

What is TAK-875 used for?

TAK-875 is an investigational small molecule being developed for the treatment of type 2 diabetes mellitus. It has been studied in diabetic patients, with clinical trials focusing on its efficacy and safety in this population. The drug is in Phase 3 clinical development.

Who makes TAK-875?

TAK-875 is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company has conducted multiple clinical trials of the drug in Japan and the United States.

What phase is TAK-875 in?

TAK-875 is in Phase 3 clinical development. It has completed three Phase 3 trials in Japan, including a double-blind comparative study, a long-term study, and an open-label study. The drug is investigational and not yet approved.

What clinical trials is TAK-875 in?

TAK-875 has completed three Phase 3 trials in Japan: NCT01433393, a double-blind comparative study with 192 patients; NCT01433406, a long-term study with 1222 patients; and NCT01433419, an open-label study with 333 patients. A Phase 1 drug-interaction study, NCT01496443, was also completed in the United States.

Is TAK-875 the same as any other drug?

TAK-875 is not known to have alternative names. It is a distinct investigational compound developed by Takeda Pharmaceutical Company Limited for type 2 diabetes mellitus.