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TAK-792

Phase 1

Healthy Male Adults Participants | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Mar 19, 2019

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment72

FDA Designations

No designations recorded

Clinical trial landscape

TAK-792 · 1 trial · 1 indication

Phase 1 1
NCT02448719Single-Dose Phase 1 Study of TAK-792Healthy Male Adults Participants
COMPLETED72 Analytics
PHASE1COMPLETED
Single-Dose Phase 1 Study of TAK-792
Healthy Male Adults ParticipantsUnlock trial analytics

Study Endpoints

Primary Endpoints

Percentage of Participants Who Experience at Least One Treatment Emergent Adverse Event (TEAE)
Baseline up to Day 8
Number of Participants With TEAE Related to Vital Signs
Baseline up to Day 5

Vital signs included body temperature (infra-axillary measurement), supine blood pressure (systolic and diastolic) after the participant has rested for at least 5 minutes, respiratory rate, and pulse (beats per minute \[bpm\]).

Number of Participants With TEAE Related to Body Weight
Baseline up to Day 5
Number of Participants With TEAE Related to Electrocardiograms (ECG)
Baseline up to Day 5
Number of Participants With TEAEs Related to Laboratory Tests
Baseline up to Day 5

Reported TEAE Related to Laboratory Tests are following; Occult blood positive, Alanine aminotransferase increased, Aspartate aminotransferase increased, Blood bilirubin increased, Blood creatine phosphokinase increased, Blood glucose increased, Blood triglycerides increased, Blood urine present, Protein urine present, and White blood cell count increased.

Number of Participants With TEAE Related to Gastrointestinal Symptom Rating Scale (GSRS)
Baseline up to Day 5

The gastrointestinal (GI) symptoms (abdominal pain, heartburn, acid regurgitation, hunger pains, nausea, borborygmus, abdominal distension, eructation, increased flatus, constipation, diarrhoea, loose stools, hard stools, urgent need for defecation, and feeling of incomplete evacuation) using GSRS questionnaires at each assessment point. The GSRS a 15-item self-administered questionnaire that assesses the impact of GI symptoms during the past week on a scale from 1 (no discomfort at all) to 7 (very severe discomfort). Possible overall scores range from 1 to 7, with lower scores indicating a better quality of life with respect to GI symptoms. TEAEs related to GSRS were reported as follows: Diarrhoea, Constipation, Faeces hard, and Faeces soft.

Secondary Endpoints

AUC(0-96): Area Under the Plasma Concentration-time Curve From Time 0 to 96 Hours Postdose for TAK-792F and Its Metabolites M-I and M-II
Day 1: pre-dose and at multiple timepoints (0.5, 1, 1.5, 2, 3, 4, 6, 8, 10, 12, 16, 24, 36, 48, 72, 96 hours post dose; up to 96 hours) post-dose
AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to Time of the Last Quantifiable Concentration for TAK-792F and Its Metabolites M-I and M-II
Day 1: pre-dose and at multiple timepoints (0.5, 1, 1.5, 2, 3, 4, 6, 8, 10, 12, 16, 24, 36, 48, 72, 96 hours post dose; up to 96 hours) post-dose
Cmax: Maximum Observed Plasma Concentration for TAK-792F and Its Metabolites M-I and M-II
Day 1: pre-dose and at multiple timepoints (0.5, 1, 1.5, 2, 3, 4, 6, 8, 10, 12, 16, 24, 36, 48, 72, 96 hours post dose; up to 96 hours) post-dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Cohort 1-activeEXPERIMENTALSingle oral administration of TAK-792 30 milligram (mg) in Japanese participants
Cohort 1-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 30 mg placebo in Japanese participants
Cohort 2-activeEXPERIMENTALSingle oral administration of TAK-792 100 mg in Japanese participants
Cohort 2-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 100 mg placebo in Japanese participants
Cohort 3-activeEXPERIMENTALSingle oral administration of TAK-792 250 mg in Japanese participants
Cohort 3-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 250 mg placebo in Japanese participants
Cohort 4-activeEXPERIMENTALSingle oral administration of TAK-792 500 mg in Japanese and Caucasian participants
Cohort 4-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 500 mg placebo in Japanese and Caucasian participants
Cohort 5-activeEXPERIMENTALSingle oral administration of TAK-792 750 mg in Japanese and Caucasian participants
Cohort 5-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 750 mg placebo in Japanese and Caucasian participants
Cohort 6-activeEXPERIMENTALSingle oral administration of TAK-792 1250 mg in Japanese and Caucasian participants
Cohort 6-placeboPLACEBO_COMPARATORSingle oral administration of TAK-792 1250 mg placebo in Japanese and Caucasian participants

Interventions

NameTypeDescription
TAK-792 30 mgDRUGTAK-792 30 mg was administered in the morning after a fast.
TAK-792 30 mg placeboDRUGTAK-792 30 mg placebo was administered in the morning after a fast.
TAK-792 100 mgDRUGTAK-792 100 mg was administered in the morning after a fast.
TAK-792 100 mg placeboDRUGTAK-792 100 mg placebo was administered in the morning after a fast.
TAK-792 250 mgDRUGTAK-792 250 mg was administered in the morning after a fast.
TAK-792 250 mg placeboDRUGTAK-792 250 mg placebo was administered in the morning after a fast.
TAK-792 500 mgDRUGTAK-792 500 mg was administered in the morning after a fast or after breakfast.
TAK-792 500 mg placeboDRUGTAK-792 500 mg placebo was administered in the morning after a fast or after breakfast.
TAK-792 750 mgDRUGTAK-792 750 mg was administered in the morning after a fast.
TAK-792 750 mg placeboDRUGTAK-792 750 mg placebo was administered in the morning after a fast.
TAK-792 1250 mgDRUGTAK-792 1250 mg was administered in the morning after a fast.
TAK-792 1250 mg placeboDRUGTAK-792 1250 mg placebo was administered in the morning after a fast.
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Eligibility Criteria

Age Range20 Years to 45 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. In the opinion of the investigator or sub-investigator, the participant is capable of understanding and complying with protocol requirements. 2. The participant signs and dates a written, informed consent form and any required privacy authorization prior to the initiation of ...

Countries:Japan
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Frequently asked questions about TAK-792

What is TAK-792 used for?

TAK-792 is an investigational small molecule being studied in healthy male adult participants. It is not approved for any disease and remains in clinical development. The completed Phase 1 trial evaluated its safety and tolerability in healthy volunteers, with no therapeutic indication established yet.

Who makes TAK-792?

TAK-792 is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company sponsored the single-dose Phase 1 study of the drug in Japan.

What phase is TAK-792 in?

TAK-792 is in Phase 1 clinical development. A single-dose Phase 1 study has been completed, and the drug remains investigational. It has not been approved by regulatory authorities, and its safety and efficacy are still being evaluated in early-stage trials.

What clinical trials is TAK-792 in?

TAK-792 has one completed clinical trial, NCT02448719, titled "Single-Dose Phase 1 Study of TAK-792." This Phase 1 study enrolled 72 healthy male adult participants in Japan and was placebo-controlled, randomized, and double-blind.

Is TAK-792 FDA approved?

TAK-792 is not FDA approved. It is an investigational drug that has completed a Phase 1 clinical trial in healthy volunteers. The drug is still in clinical development, and no approval status has been granted for any indication.