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TAK-438ASA

Phase 1

Healthy Volunteers | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Nov 19, 2019

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment276

FDA Designations

No designations recorded

Clinical trial landscape

TAK-438ASA · 1 trial · 1 indication

Phase 1 1
NCT03456960A Study to Evaluate the Bioequivalence (BE) and the Food Effect of TAK-438ASA TabletHealthy Volunteers
COMPLETED276 Analytics
PHASE1COMPLETED
A Study to Evaluate the Bioequivalence (BE) and the Food Effect of TAK-438ASA Tablet
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Study Endpoints

Primary Endpoints

Study 1, AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to the Time of the Last Quantifiable Concentration for Free Base of TAK-438 (TAK-438F)
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, Cmax: Maximum Observed Plasma Concentration for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to the Time of the Last Quantifiable Concentration for Unchanged Aspirin
Day 1 pre-dose and at multiple time points (up to 12 hours) post-dose
Study 1, Cmax: Maximum Observed Plasma Concentration for Unchanged Aspirin
Day 1 pre-dose and at multiple time points (up to 12 hours) post-dose

Secondary Endpoints

Study 1, AUC∞: Area Under the Plasma Concentration-time Curve From Time 0 to Infinity for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, MRT (Infinity,ev): Mean Residence Time From Time 0 to Infinity for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Pilot phase of Study 1,TAK-438ASA + TAK-438 and AspirinEXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in the Pilot phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 2 in the Pilot phase of Study 1 (Day 16).
Pilot phase of Study 1,TAK-438 and Aspirin + TAK-438ASAEXPERIMENTALOne TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 1 in the Pilot phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by, one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in the Pilot phase of Study 1 (Day 16).
Pivotal phase of Study 1, TAK-438ASA + TAK-438 and AspirinEXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in the Pivotal phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 2 in the Pivotal phase of Study 1 (Day 16).
Pivotal phase of Study 1, TAK-438 and Aspirin + TAK-438ASAEXPERIMENTALOne TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 1 in the Pivotal phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in the Pivotal phase of Study 1 (Day 16).
Study 2,TAK-438ASA (Fasted + Fed condition)EXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in Study 2 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally 30 minutes after breakfast, on Day 1 of Period 2 in Study 2 (Day 16).
Study 2,TAK-438ASA (Fed + Fasted condition)EXPERIMENTALOne TAK-438ASA tablet, orally 30 minutes after breakfast, on Day 1 of Period 1 in Study 2 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in Study 2 (Day 16).

Interventions

NameTypeDescription
TAK-438ASADRUGTAK-438ASA tablet.
TAK-438DRUGTAK-438 tablet.
AspirinDRUGAspirin enteric-coated tablet.
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Eligibility Criteria

Age Range20 Years to 60 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. In the opinion of the investigator or sub-investigator, participants are capable of understanding the procedures required for the study and complying with its requirements. 2. Participants sign and date an informed consent form by themselves prior to the initiation of any stu...

Countries:Japan
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Frequently asked questions about TAK-438ASA

What is TAK-438ASA?

TAK-438ASA is an investigational small molecule being developed by Takeda Pharmaceutical Company Limited (TAK). It is currently in Phase 1 clinical development. The drug has been studied in healthy volunteers, with one completed clinical trial evaluating its bioequivalence and food effect.

What is TAK-438ASA used for?

TAK-438ASA is being studied for use in healthy volunteers. The completed Phase 1 trial, NCT03456960, evaluated the bioequivalence and food effect of TAK-438ASA tablet. The study enrolled 276 healthy male participants in Japan, aged 20 years and older.

Who makes TAK-438ASA?

TAK-438ASA is developed by Takeda Pharmaceutical Company Limited, a biopharmaceutical company listed on the stock exchange under the ticker TAK. The company is conducting clinical research on this investigational small molecule drug.

What phase is TAK-438ASA in?

TAK-438ASA is in Phase 1 clinical development. The drug is investigational and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and there are no active trials currently ongoing for this drug.

What clinical trials is TAK-438ASA in?

TAK-438ASA has one completed clinical trial, NCT03456960, titled 'A Study to Evaluate the Bioequivalence (BE) and the Food Effect of TAK-438ASA Tablet'. This Phase 1 study was conducted in Japan with 276 healthy male volunteers, and it was a controlled, randomized trial.

Is TAK-438ASA the same as TAK-438?

TAK-438ASA is a distinct drug candidate from TAK-438, as indicated by its unique name. The drug is being developed by Takeda Pharmaceutical Company Limited. The clinical trial NCT03456960 specifically evaluates TAK-438ASA tablet, not TAK-438.