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TAK-438ASA

Phase 1

Healthy Volunteers | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Nov 19, 2019

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment276
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03456960A Study to Evaluate the Bioequivalence (BE) and the Food Effect of TAK-438ASA TabletPHASE1 COMPLETED 276Mar 8, 2018Oct 12, 2018Nov 19, 20191 Japan
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Study Endpoints
Primary Endpoints
Study 1, AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to the Time of the Last Quantifiable Concentration for Free Base of TAK-438 (TAK-438F)
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, Cmax: Maximum Observed Plasma Concentration for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to the Time of the Last Quantifiable Concentration for Unchanged Aspirin
Day 1 pre-dose and at multiple time points (up to 12 hours) post-dose
Study 1, Cmax: Maximum Observed Plasma Concentration for Unchanged Aspirin
Day 1 pre-dose and at multiple time points (up to 12 hours) post-dose
Secondary Endpoints
Study 1, AUC∞: Area Under the Plasma Concentration-time Curve From Time 0 to Infinity for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
Study 1, MRT (Infinity,ev): Mean Residence Time From Time 0 to Infinity for TAK-438F
Day 1 pre-dose and at multiple time points (up to 48 hours) post-dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER
Treatment Arms
ArmTypeDescription
Pilot phase of Study 1,TAK-438ASA + TAK-438 and AspirinEXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in the Pilot phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 2 in the Pilot phase of Study 1 (Day 16).
Pilot phase of Study 1,TAK-438 and Aspirin + TAK-438ASAEXPERIMENTALOne TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 1 in the Pilot phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by, one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in the Pilot phase of Study 1 (Day 16).
Pivotal phase of Study 1, TAK-438ASA + TAK-438 and AspirinEXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in the Pivotal phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 2 in the Pivotal phase of Study 1 (Day 16).
Pivotal phase of Study 1, TAK-438 and Aspirin + TAK-438ASAEXPERIMENTALOne TAK-438 10 mg tablet and one aspirin 100 mg tablet, orally without breakfast, on Day 1 of Period 1 in the Pivotal phase of Study 1 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in the Pivotal phase of Study 1 (Day 16).
Study 2,TAK-438ASA (Fasted + Fed condition)EXPERIMENTALOne TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 1 in Study 2 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally 30 minutes after breakfast, on Day 1 of Period 2 in Study 2 (Day 16).
Study 2,TAK-438ASA (Fed + Fasted condition)EXPERIMENTALOne TAK-438ASA tablet, orally 30 minutes after breakfast, on Day 1 of Period 1 in Study 2 (Day 1), followed by a washout period (Days 2 to 15), followed by one TAK-438ASA tablet, orally without breakfast, on Day 1 of Period 2 in Study 2 (Day 16).
Interventions
NameTypeDescription
TAK-438ASADRUGTAK-438ASA tablet.
TAK-438DRUGTAK-438 tablet.
AspirinDRUGAspirin enteric-coated tablet.
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Eligibility Criteria
Age Range20 Years — 60 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. In the opinion of the investigator or sub-investigator, participants are capable of understanding the procedures required for the study and complying with its requirements. 2. Participants sign and date an informed consent form by themselves prior to the initiation of any stu...

Countries:Japan
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