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TAK-418

Phase 1

Healthy Participants | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Sep 9, 2019

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment40

FDA Designations

No designations recorded

Clinical trial landscape

TAK-418 · 1 trial · 1 indication

Phase 1 1
NCT03228433A Study to Evaluate Safety, Tolerability and Pharmacokinetics of Ascending Oral Single Dose of TAK-418 in Healthy ParticipantsHealthy Participants
COMPLETED40 Analytics
PHASE1COMPLETED
A Study to Evaluate Safety, Tolerability and Pharmacokinetics of Ascending Oral Single Dose of TAK-418 in Healthy Participants
Healthy ParticipantsUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Participants Reporting One or More Treatment-emergent Adverse Events (TEAEs)
Baseline Up to Day 184
Number of Participants Who Discontinued Due to an Adverse Event (AE)
Baseline Up to Day 184
Number of Participants Who Meet the Markedly Abnormal Criteria for Neurological Assessment Measurements at Least Once Post Dose
Baseline Up to Day 184
Number of Participants Who Meet the Markedly Abnormal Criteria for Safety Laboratory Tests at Least Once Post Dose
Baseline Up to Day 184
Number of Participants Who Meet the Markedly Abnormal Criteria for Vital Sign Measurements at Least Once Post Dose
Baseline Up to day 184
Number of Participants Who Meet the Markedly Abnormal Criteria for Safety 12-lead Electrocardiogram (ECG) Parameters at Least Once Post Dose
Baseline Up to Day 14

Secondary Endpoints

AUClast: Area Under the Plasma Concentration-time Curve From Time 0 to the Time of the Last Quantifiable Concentration of TAK-418F (TAK-418 Free Base)
Day 1 pre-dose and at multiple time points (up to 72 hours) post-dose
AUC∞: Area Under the Plasma Concentration-time Curve From Time 0 to Infinity for TAK-418F
Day 1 pre-dose and at multiple time points (up to 72 hours) post-dose
Cmax: Maximum Observed Plasma Concentration for TAK-418F
Day 1 pre-dose and at multiple time points (up to 72 hours) post-dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelSEQUENTIAL
PurposeOTHER

Treatment Arms

ArmTypeDescription
Cohort 1: TAK-418 5 mgEXPERIMENTALTAK-418 5 milligram (mg), capsule, orally, once on Day 1.
Cohort 2: TAK-418 15 mgEXPERIMENTALTAK-418 15 mg, capsule, orally, once on Day 1. Actual dose of TAK-418 may vary based on safety, tolerability and PK data from previous Cohorts.
Cohort 3: TAK-418 30 mg Fasted + TAK-418 30 mg FedEXPERIMENTALTAK-418 30 mg, capsule, in fasted state, orally, once on Day 1, followed by a 28-day washout period, further followed by TAK-418 30 mg, capsule, in fed state, orally, once on Day 1. Actual dose of TAK-418 may vary based on safety, tolerability and PK data from previous Cohorts.
Cohort 4: TAK-418 40 mgEXPERIMENTALTAK-418 40 mg, capsule, orally, once on Day 1. Actual dose of TAK-418 may vary based on safety, tolerability and PK data from previous Cohorts.
Cohort 5: TAK-418 60 mgEXPERIMENTALTAK-418 60 mg, capsule, orally, once on Day 1. Actual dose of TAK-418 may vary based on safety, tolerability and PK data from previous Cohorts.
Cohorts 1-5: PlaceboPLACEBO_COMPARATORTAK-418 placebo-matching, capsule, orally, once on Day 1.

Interventions

NameTypeDescription
TAK-418DRUGTAK-418 Capsule.
TAK-418 PlaceboDRUGTAK-418 placebo-matching capsules.
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Is a male or female participants with a body mass index (BMI) within the range of 18.5 -30.0 kilogram per square meter (kg/m\^2) at the Screening Visit. 2. Is a nonsmoker who has not used tobacco or nicotine-containing products (example, nicotine patch) for at least 6 months ...

Countries:United States
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Frequently asked questions about TAK-418

What is TAK-418 used for?

TAK-418 is an investigational small molecule being studied in healthy participants. It is currently in Phase 1 clinical development, with a completed trial evaluating its safety, tolerability, and pharmacokinetics after ascending oral single doses. TAK-418 is not approved by the FDA and remains under investigation.

Who makes TAK-418?

TAK-418 is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company is conducting clinical research on this investigational small molecule in healthy participants.

What phase is TAK-418 in?

TAK-418 is in Phase 1 clinical development. A Phase 1 trial has been completed, and the drug remains investigational. It has not been approved by the FDA and is still in the early stages of clinical testing.

What clinical trials is TAK-418 in?

TAK-418 has one completed clinical trial, NCT03228433, titled "A Study to Evaluate Safety, Tolerability and Pharmacokinetics of Ascending Oral Single Dose of TAK-418 in Healthy Participants." This Phase 1 study enrolled 40 participants in the United States and was placebo-controlled and double-blind.

Is TAK-418 FDA approved?

No, TAK-418 is not FDA approved. It is an investigational drug currently in Phase 1 clinical development. The completed trial focused on safety, tolerability, and pharmacokinetics in healthy participants, and the drug has not yet progressed to later-stage trials or regulatory approval.